中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [3]
地理科学与资源研究所 [2]
过程工程研究所 [1]
高能物理研究所 [1]
海洋研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2024 [2]
2023 [1]
2022 [5]
学科主题
Hydrogen B... [1]
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浏览/检索结果:
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Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
;
Lyu, Xiaodong
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/05
Structure-based discovery of a new series of nucleoside-derived ring-opening PRMT5 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 19
作者:
Chen, Yuting
;
Wang, Zekun
;
Zhang, Junjie
;
Shi, Qiongyu
;
Yang, Hong
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/05/07
PRMT5
Nucleoside derivatives
Methyltransferases
Structure -activity relationship
Structure-activity relationship study of a series of nucleoside derivatives bearing sulfonamide scaffold as potent and selective PRMT5 inhibitors
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 130, 页码: 20
作者:
Chen, Yuting
;
Shi, Qiongyu
;
Yang, Hong
;
Li, Jiayi
;
Zhou, Kaixin
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2023/04/10
Epigenetic
PRMT5 inhibitor
Nucleoside derivatives
Structure-activity Relationship Prodrug
Phosphinous Acid-Phosphinito Tetra-Icosahedral Au52Nanoclusters for Electrocatalytic Oxygen Reduction
期刊论文
OAI收割
JACS Au, 2022, 卷号: 2, 期号: 11, 页码: 2617-2626
作者:
Zhuang, Shengli
;
Chen, Dong
;
Ng, Wai-Pan
;
Liu, Dongyi
;
Liu, Li-Juan
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2023/06/26
Density functional theory - Electrocatalysts - Electrolytic reduction - Gold - Ligands - Nanoclusters - Oxygen - Phosphorus
EGPI-1, a novel eIF4E/eIF4G interaction inhibitor, inhibits lung cancer cell growth and angiogenesis through Ras/MNK/ERK/eIF4E signaling pathway
期刊论文
OAI收割
CHEMICO-BIOLOGICAL INTERACTIONS, 2022, 卷号: 352, 页码: 10
作者:
Qi, Xueju
;
Zhang, Shuna
;
Chen, Zekun
;
Wang, Lijun
;
Zhu, Wenyong
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/07/18
Human lung cancer
eIF4E
EGPI-1
Anticancer
Angiogenesis
Collective neutrino oscillations in moving and polarized matter
期刊论文
OAI收割
Journal of Physics: Conference Series, 2022, 卷号: 2156, 期号: 1, 页码: 12180
作者:
Chen, Zekun
;
Kouzakov, Konstantin
;
Li, Yu-Feng,
;
Shakhov, Vadim
;
Stankevich, Konstantin,
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/11/10
Mapping Gridded Gross Domestic Product Distribution of China Using Deep Learning With Multiple Geospatial Big Data
期刊论文
OAI收割
IEEE JOURNAL OF SELECTED TOPICS IN APPLIED EARTH OBSERVATIONS AND REMOTE SENSING, 2022, 卷号: 15, 页码: 1791-1802
作者:
Chen, Yuehong
;
Wu, Guohao
;
Ge, Yong
;
Xu, Zekun
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/09/21
Economic indicators
Deep learning
Convolutional neural networks
Decoding
Encoding
Geospatial analysis
Big Data
1-km gridded gross domestic product (GDP)
China
deep learning
downscaling
geospatial big data
gross domestic product (GDP)
Mapping Gridded Gross Domestic Product Distribution of China Using Deep Learning With Multiple Geospatial Big Data
期刊论文
OAI收割
IEEE JOURNAL OF SELECTED TOPICS IN APPLIED EARTH OBSERVATIONS AND REMOTE SENSING, 2022, 卷号: 15, 页码: 1791-1802
作者:
Chen, Yuehong
;
Wu, Guohao
;
Ge, Yong
;
Xu, Zekun
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/09/21
Economic indicators
Deep learning
Convolutional neural networks
Decoding
Encoding
Geospatial analysis
Big Data
1-km gridded gross domestic product (GDP)
China
deep learning
downscaling
geospatial big data
gross domestic product (GDP)