机构

• 上海药物研究所 [14]
• 南京地理与湖泊研究所 [1]

采集方式

• OAI收割 [15]

内容类型

• 期刊论文 [15]

发表日期

• 2021 [1]
• 2020 [1]
• 2015 [1]
• 2014 [1]
• 2013 [3]
• 2012 [2]
• 更多

学科主题

筛选

浏览/检索结果: 共15条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Assessment of extrinsic and intrinsic influences on water quality variation in subtropical agricultural multipond system 期刊论文  OAI收割 ENVIRONMENTAL POLLUTION, 2021, 卷号: 276 作者:  Chen, Wenjun;  Nover, Daniel;  Xia, Yongqiu;  Zhang, Guangxin;  Yen, Haw   |  收藏  |  浏览/下载：25/0  |  提交时间：2022/03/10 The Nonclinical Pharmacokinetics and Prediction of Human Pharmacokinetics of SPH3127, a Novel Direct Renin Inhibitor 期刊论文  OAI收割 EUROPEAN JOURNAL OF DRUG METABOLISM AND PHARMACOKINETICS, 2020, 卷号: 45, 期号: 1, 页码: 15-26 作者:  Zhang, Leduo;  Mao, Yu;  Gao, Zhiwei;  Chen, Xiaoyan;  Li, Xin   |  收藏  |  浏览/下载：24/0  |  提交时间：2020/07/01 Fragment-Based Drug Discovery of 2-Thiazolidinones as BRD4 Inhibitors: 2. Structure-Based Optimization 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 3, 页码: 1281-1297 作者:  Zhao, Lele;  Wang, Yingqing;  Cao, Danyan;  Chen, Tiantian;  Wang, Qi   |  收藏  |  浏览/下载：22/0  |  提交时间：2019/01/08 A Chemical Tuned Strategy to Develop Novel Irreversible EGFR-TK Inhibitors with Improved Safety and Pharmacokinetic Profiles 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 57, 期号: 23, 页码: 9889-9900 作者:  Xia, Guangxin;  Chen, Wenteng;  Zhang, Jing;  Shao, Jiaan;  Zhang, Yong   |  收藏  |  浏览/下载：40/0  |  提交时间：2019/01/08 Design, Synthesis, and Biological Evaluation of Novel Conformationally Constrained Inhibitors Targeting EGFR 期刊论文  OAI收割 ACS MEDICINAL CHEMISTRY LETTERS, 2013, 卷号: 4, 期号: 10, 页码: 974-978 作者:  Wu, Jianwei;  Chen, Wenteng;  Xia, Guangxin;  Zhang, Jing;  Shao, Jiaan   |  收藏  |  浏览/下载：55/0  |  提交时间：2019/01/08 Anticancer  kinase inhibitor  EGFR  conformationally constrained   Design, synthesis and SAR of piperidyl-oxadiazoles as 11 beta-hydroxysteroid dehydrogenase 1 inhibitors 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 62, 页码: 1-10 作者:  Xia, Guangxin;  You, Xiaodi;  Liu, Lin   |  收藏  |  浏览/下载：15/0  |  提交时间：2019/01/08 11 beta-HSD1 inhibitor  Oxadiazole  Bioisostere  SAR  Docking   Design and Synthesis of (R)-1-Arylsulfonylpiperidine-2-carboxamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors 期刊论文  OAI收割 CHEMMEDCHEM, 2013, 卷号: 8, 期号: 4, 页码: 577-581 作者:  Xia, Guangxin;  Liu, Lin;  Liu, Haiyan;  Yu, Jianxin;  Xu, Zhenmin   |  收藏  |  浏览/下载：19/0  |  提交时间：2019/01/08 11-HSD1  diabetes  docking  inhibitors   Discovery of 2-Alkyl-1-arylsulfonylprolinamides as 11 beta-Hydroxysteroid Dehydrogenase Type 1 Inhibitors 期刊论文  OAI收割 ACS MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 3, 期号: 10, 页码: 793-798 作者:  Yu, Jianxin;  Liu, Haiyan;  Xia, Guangxin;  Liu, Lin;  Xu, Zhenmin   |  收藏  |  浏览/下载：135/0  |  提交时间：2019/01/08 metabolic syndrome  enzyme inhibitor  11 beta-hydroxysteroid dehydrogenase type 1  sulfonamide  2-alkylproline  prolinamide   Discovery of novel sulfonamides as potent and selective inhibitors against human and mouse 11 beta-hydroxysteroid dehydrogenase type 1 期刊论文  OAI收割 MOLECULAR AND CELLULAR ENDOCRINOLOGY, 2012, 卷号: 358, 期号: 1, 页码: 46-52 作者:  Xia, Guangxin;  Liu, Lin;  Xue, Mengzhu;  Liu, Haiyan;  Yu, Jianxin   |  收藏  |  浏览/下载：22/0  |  提交时间：2019/01/08 11 beta-HSD1  Inhibitor  Sulfonamide  Diabetes  Docking   Potent and novel 11 beta-HSD1 inhibitors identified from shape and docking based virtual screening 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 19, 页码: 5739-5744 作者:     |  收藏  |  浏览/下载：32/0  |  提交时间：2019/01/08 11 beta-HSD1 inhibitor  Virtual screening  Docking  Shape similarity