中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共40条,第1-10条 帮助

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Discovery of Novel Nonpeptidic and Noncovalent Small Molecule 3CLpro Inhibitors as anti-SARS-CoV-2 Drug Candidate 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 15, 页码: 12760-12783
作者:  
Jiang, Zhidong;  Feng, Bo;  Chen, Lu;  Nie, Tianqing;  Chen, Shizhao
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/09/26
Discovery and Mechanism Study of SARS-CoV-2 3C-like Protease Inhibitors with a New Reactive Group 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 18
作者:  
Ren, Pengxuan;  Li, Hui;  Nie, Tianqing;  Jian, Xiaoqin;  Yu, Changyue
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
Discovery of novel non-peptidic and non-covalent small-molecule 3CL(pro) inhibitors as potential candidate for COVID-19 treatment 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 4
作者:  
Jiang, Zhidong;  Feng, Bo;  Zhang, Yumin;  Nie, Tianqing;  Liu, Hong
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
Discovery, synthesis and mechanism study of 2,3,5-substituted [1,2,4]-thiadiazoles as covalent inhibitors targeting 3C-Like protease of SARS-CoV-2 期刊论文  OAI收割
European journal of medicinal chemistry, 2023, 卷号: 249, 页码: 115129
作者:  
Ren, Pengxuan;  Yu, Changyue;  Zhang, Ruxue;  Nie, Tianqing;  Hu, Qiaoyu
  |  收藏  |  浏览/下载:29/0  |  提交时间:2024/03/26
In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2 期刊论文  OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:  
Shang, Weijuan;  Dai, Wenhao;  Yao, Cheng;  Xu, Ling;  Tao, Xiangming
  |  收藏  |  浏览/下载:25/0  |  提交时间:2023/04/10
The p300 Inhibitor A-485 Exerts Antitumor Activity in Growth Hormone Pituitary Adenoma 期刊论文  OAI收割
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 2022, 页码: 10
作者:  
Ji, Chenxing;  Xu, Wen;  Ding, Hong;  Chen, Zhengyuan;  Shi, Chengzhang
  |  收藏  |  浏览/下载:52/0  |  提交时间:2022/06/15
Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV-2 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 4, 页码: 2794-2808
作者:  
Dai, Wenhao;  Jochmans, Dirk;  Xie, Hang;  Yang, Hang;  Li, Jian
  |  收藏  |  浏览/下载:44/0  |  提交时间:2022/08/16
Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 20
作者:  
Zhang, Rui;  Li, Heng;  Zhang, Xianglei;  Li, Jian;  Su, Haixia
  |  收藏  |  浏览/下载:45/0  |  提交时间:2021/05/24
Guidelines for the use and interpretation of assays for monitoring autophagy (4th edition) 期刊论文  OAI收割
AUTOPHAGY, 2021, 卷号: 17
作者:  
Klionsky, Daniel J.;  Abdel-Aziz, Amal Kamal;  Abdelfatah, Sara;  Abdellatif, Mahmoud;  Abdoli, Asghar
  |  收藏  |  浏览/下载:319/0  |  提交时间:2021/05/31
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease 期刊论文  OAI收割
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:  
Dai, Wenhao;  Zhang, Bing;  Jiang, Xia-Ming;  Su, Haixia;  Li, Jian
  |  收藏  |  浏览/下载:52/0  |  提交时间:2020/12/24