中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [108]
化学研究所 [1]
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OAI收割 [109]
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期刊论文 [106]
会议论文 [3]
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2026 [2]
2025 [9]
2024 [4]
2023 [4]
2022 [6]
2021 [5]
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DMetFinder: A novel mass spectrometry analysis tool for comprehensive drug metabolite detection
期刊论文
OAI收割
TALANTA, 2026, 卷号: 298, 页码: 9
作者:
Ke, Wenhao
;
Wang, Yingying
;
Zeng, Yanping
;
Hou, Haiyang
;
Zhu, Dafu
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Multiplexed Isotope-Coded Mass Spectrometry Footprinting Enables Broad Heteroatom-Residue Mapping and Uncovers Noncanonical Ligand-Binding Sites in Amyloidosis Proteins
期刊论文
OAI收割
ANALYTICAL CHEMISTRY, 2026, 页码: 13
作者:
Yang, Kuoqi
;
Zheng, Wei
;
Bai, Lin
;
Wang, Kai
;
Zhang, Jian
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Design, synthesis, and biological evaluation of KDM5B degraders against hematologic malignancy cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 296, 页码: 17
作者:
Liu, Xiaowen
;
Li, Jiarong
;
Guo, Yihao
;
Xie, Zhicheng
;
Geng, Meiyu
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Structural optimization of phthalazine derivatives for anti-HBV activities to improve oral bioavailability
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 10
作者:
Yang, Yurong
;
Xiao, Fuling
;
Zuo, Jianping
;
Yang, Li
;
Hu, Youhong
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Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
;
Xiao, Jian
;
Zeng, Yanping
;
Li, Yangsha
;
Wei, Aihuan
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Discovery of potent anti-idiopathic pulmonary fibrosis (IPF) agents based on an o-aminopyridinyl alkynyl scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 15
作者:
Wang, Yang
;
Fan, Wenhui
;
Guo, Yihao
;
Sun, Li
;
Hu, Youhong
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Discovery of novel Ebola entry inhibitors with 1,2,3,4-tetrahydroisoquinoline-3-carboxamide based on (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 123, 页码: 4
作者:
Lin, Junzhen
;
Xiao, Fuling
;
Han, Sheng
;
Hu, Youhong
;
Zuo, Jianping
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Fine structural design of 3βHSD1 inhibitors for prostate cancer
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2025, 卷号: 122, 期号: 26, 页码: 12
作者:
He, Dongyin
;
Zhang, Luyao
;
Yu, Leiye
;
Zhang, Yuhang
;
Chen, Jingjing
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Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:
Zeng, Yanping
;
Xiao, Jian
;
Shi, Li
;
Li, Yangsha
;
Xu, Yuanxin
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Diazonium-based derivatization for enhanced detection of phosphorylated metabolites by LC-MS in cells
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2025, 卷号: 255, 页码: 7
作者:
Wang, Yikang
;
Lin, Feifei
;
Zhu, Guozheng
;
Zhou, Xiaoxue
;
Hu, Youhong
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