中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [27]
采集方式
OAI收割 [27]
内容类型
期刊论文 [27]
发表日期
2022 [1]
2021 [3]
2020 [4]
2019 [3]
2018 [2]
2017 [2]
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Discovery of seneciobipyrrolidine derivatives for the amelioration of glucose homeostasis disorders through 4E-BP1/Akt/AMPK signaling activation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 228, 页码: 25
作者:
Che, Jinxin
;
Ma, Canliang
;
Lu, Jialiang
;
Chen, Binhui
;
Shi, Qiuqiu
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2022/06/15
Seneciobipyrrolidine
Phenotypic screening
Glucose homeostasis
Proteomic analysis
L6 myotubes
4E-BP1
Discovery of 1,5-Dihydro-4H-imidazol-4-one Derivatives as Potent, Selective Antagonists of CXC Chemokine Receptor 2
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 5, 页码: 836-845
作者:
Che, Jinxin
;
Wang, Zhilong
;
Shen, Zheyuan
;
Zhuang, Weihao
;
Ying, Huazhou
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2021/08/17
cancer metastasis
CXCR1
CXCR2
selectivity
antagonist
1,5-dihydro-4H-imidazol-4-one
Selectivity Comparison of Tumor-Imaging Probes Designed Based on Various Tumor-Targeting Strategies: A Proof of Concept Study
期刊论文
OAI收割
ACS applied bio materials, 2021, 卷号: 4, 期号: 3, 页码: 2058-2065
作者:
Guo, Rui-Ying
;
Wang, Han-Min
;
Dong, Xiaowu
;
Hu, Yongzhou
;
Li, Jia
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/03/15
fluorescence imaging
fluorescent probe
imaging contrast
receptor
tumor
tumor microenvironment
Bioinspired Design of Reversible Fluorescent Probes for Tracking Nitric Oxide Dynamics in Live Cells
期刊论文
OAI收割
CCS CHEMISTRY, 2021, 卷号: 3, 期号: 10, 页码: 180
作者:
Guo Ruiying
;
Zhang Yutian
;
Chanmungkalakul Supphachok
;
Guo Haoran
;
Hu Yongzhou
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/05/22
fluorescent probe
fluorescence imaging
reversible
nitric oxide
S-nitrosation
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:
Che, Jinxin
;
Huang, Feng
;
Zhang, Mengmeng
;
Xu, Gaoya
;
Qu, Bingxue
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2020/12/21
Metabolic pathways
Isocitrate dehydrogenase 2
Conformational restriction
Macrocyclic derivatives
Inhibitors
A fluorogenic probe for tracking GSH flux in developing neurons
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2020, 卷号: 56, 期号: 4, 页码: 515-518
作者:
Zong, Haichao
;
Peng, Jiayi
;
Li, Xiao-Rong
;
Liu, Meng
;
Hu, Yongzhou
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
Microenvironment-Responsive Small-Molecule Probe for Pulmonary Fibrosis Detection
期刊论文
OAI收割
ANALYTICAL CHEMISTRY, 2020, 卷号: 92, 期号: 1, 页码: 699-706
作者:
Dong, Ying
;
Li, Xiao-Rong
;
Chen, Qi
;
Guo, Rui-Ying
;
Tang, Bi-Xi
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:
Zhan, Wenhu
;
Che, Jinxin
;
Xu, Lei
;
Wu, Yizhe
;
Hu, Xiaobei
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/07/01
Pyrazole-thiophene derivatives
Akt inhibitor
Antitumor
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:
Dong, Xiaowu
;
Zhan, Wenhu
;
Zhao, Mengting
;
Che, Jinxin
;
Dai, Xiaoyang
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/07/01