中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共27条,第1-10条 帮助

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Discovery of seneciobipyrrolidine derivatives for the amelioration of glucose homeostasis disorders through 4E-BP1/Akt/AMPK signaling activation 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 228, 页码: 25
作者:  
Che, Jinxin;  Ma, Canliang;  Lu, Jialiang;  Chen, Binhui;  Shi, Qiuqiu
  |  收藏  |  浏览/下载:47/0  |  提交时间:2022/06/15
Discovery of 1,5-Dihydro-4H-imidazol-4-one Derivatives as Potent, Selective Antagonists of CXC Chemokine Receptor 2 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 5, 页码: 836-845
作者:  
Che, Jinxin;  Wang, Zhilong;  Shen, Zheyuan;  Zhuang, Weihao;  Ying, Huazhou
  |  收藏  |  浏览/下载:32/0  |  提交时间:2021/08/17
Selectivity Comparison of Tumor-Imaging Probes Designed Based on Various Tumor-Targeting Strategies: A Proof of Concept Study 期刊论文  OAI收割
ACS applied bio materials, 2021, 卷号: 4, 期号: 3, 页码: 2058-2065
作者:  
Guo, Rui-Ying;  Wang, Han-Min;  Dong, Xiaowu;  Hu, Yongzhou;  Li, Jia
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/15
Bioinspired Design of Reversible Fluorescent Probes for Tracking Nitric Oxide Dynamics in Live Cells 期刊论文  OAI收割
CCS CHEMISTRY, 2021, 卷号: 3, 期号: 10, 页码: 180
作者:  
Guo Ruiying;  Zhang Yutian;  Chanmungkalakul Supphachok;  Guo Haoran;  Hu Yongzhou
  |  收藏  |  浏览/下载:13/0  |  提交时间:2023/05/22
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:  
Che, Jinxin;  Huang, Feng;  Zhang, Mengmeng;  Xu, Gaoya;  Qu, Bingxue
  |  收藏  |  浏览/下载:58/0  |  提交时间:2020/12/21
Structure-based design, synthesis and bioactivity evaluation of macrocyclic inhibitors of mutant isocitrate dehydrogenase 2 (IDH2) displaying activity in acute myeloid leukemia cells 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 203, 页码: 19
作者:  
Che, Jinxin;  Huang, Feng;  Zhang, Mengmeng;  Xu, Gaoya;  Qu, Bingxue
  |  收藏  |  浏览/下载:40/0  |  提交时间:2020/12/21
A fluorogenic probe for tracking GSH flux in developing neurons 期刊论文  OAI收割
CHEMICAL COMMUNICATIONS, 2020, 卷号: 56, 期号: 4, 页码: 515-518
作者:  
Zong, Haichao;  Peng, Jiayi;  Li, Xiao-Rong;  Liu, Meng;  Hu, Yongzhou
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
Microenvironment-Responsive Small-Molecule Probe for Pulmonary Fibrosis Detection 期刊论文  OAI收割
ANALYTICAL CHEMISTRY, 2020, 卷号: 92, 期号: 1, 页码: 699-706
作者:  
Dong, Ying;  Li, Xiao-Rong;  Chen, Qi;  Guo, Rui-Ying;  Tang, Bi-Xi
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:  
Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:  
Dong, Xiaowu;  Zhan, Wenhu;  Zhao, Mengting;  Che, Jinxin;  Dai, Xiaoyang
  |  收藏  |  浏览/下载:37/0  |  提交时间:2020/07/01