中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [9]
南京地理与湖泊研究所 [1]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2024 [3]
2023 [1]
2022 [1]
2021 [1]
2016 [1]
2009 [1]
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学科主题
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Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 44, 期号: 11, 页码: 3476-3489
作者:
Cheng, Tingting
;
Song, Gaolei
;
Cheng, Long
;
Wang, Fan
;
Sun, Xinyu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/02/28
metabolic diseases
ATP-citrate lyase (ACLY)
lipogenesis
ACLY inhibitors
dienyldicarboxylic acid
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
Polyphenol Compound 18a Modulates UCP1-Dependent Thermogenesis to Counteract Obesity
期刊论文
OAI收割
BIOMOLECULES, 2024, 卷号: 14, 期号: 6, 页码: 21
作者:
Wen, Xueping
;
Song, Yufei
;
Zhang, Mei
;
Kang, Yiping
;
Chen, Dandan
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/08/22
18a
adipocytes
polyphenols
thermogenesis
UCP1
Development of the novel ACLY inhibitor 326E as a promising treatment for hypercholesterolemia
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 2, 页码: 739-753
作者:
Xie, Zhifu
;
Zhang, Mei
;
Song, Qian
;
Cheng, Long
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/03/27
Hypercholesterolemia
Atherosclerosis
Liver
ATP-Citrate lyase (ACLY)
Lipogenesis
Cholesterol efflux
ACLY inhibitor
Lignin-containing hydrogel matrices with enhanced adhesion and toughness for all-hydrogel supercapacitors
期刊论文
OAI收割
CHEMICAL ENGINEERING JOURNAL, 2022, 卷号: 450
作者:
Wang, Dingkun
;
Yang, Fusheng
;
Cong, Lulu
;
Feng, Wanglong
;
Wang, Chunpeng
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/19
Design and Synthesis of Alkyl Phenols Inhibitors of Death Associated Apoptotic Protein Kinase 2 (DRAK2)
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3204-3213
作者:
Zheng Zhang
;
Dai Chengqiu
;
Wu Honghong
;
Li Jingya
;
Nan Fajun
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2021/11/04
death associated apoptotic protein kinase 2
diabetes
alkylphenols
inhibitors
Design and Synthesis of Diacylglycerol Acyltransferase 1 Inhibitors Based on Aphadilactone C
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 36, 期号: 6, 页码: 1359-1367
作者:
Li Dan
;
Yin Jianpeng
;
Li Jingya
;
Nan Fajun
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
aphadilactone C
DGAT1
selective inhibitor
PF-04620110
AZD-7687
Design and Synthesis of Matrix Metalloprotease Photoaffinity Trimodular Probes
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2009, 卷号: 27, 期号: 4, 页码: 825-833
作者:
Qiu Wenwei
;
Xu Jie
;
Li Xin
;
Zhong Li
;
Li Jingya
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
trimodular probe
photoaffinity labeling
protein profiling
click chemistry
matrix metalloprotease
Click chemistry in drug discovery
期刊论文
OAI收割
Chinese Bulletin of Life Sciences, 2006, 卷号: 18, 期号: 3, 页码: 295-302
作者:
QIU WenWei
;
LI JingYa
;
LI Jia
;
NAN FaJun
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
click chemistry
combinatorial chemistry
target-guided synthesis
bioconjugate chemistry
drug discovery
Photoaffinity labeling in drug discovery
期刊论文
OAI收割
Chinese Bulletin of Life Sciences, 2005, 卷号: 17, 期号: 4, 页码: 296-303
作者:
Chou Wenwei
;
Li Jingya
;
Li Jia
;
Nan FaJun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
functional proteomics
photoaffinity labeling technology
target proteins
drug discovery