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	Discovery of novel 3-hydroxypicolinamides as selective inhibitors of HIV-1 integrase-LEDGF/p75 interaction 期刊论文 OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 125, 页码: 1051-1063 作者: Zhang, Feng-Hua; Debnath, Bikash; Xu, Zhong-Liang; Yang, Liu-Meng; Song, Li-Rui \| 收藏 \| 浏览/下载：20/0 \| 提交时间：2019/01/08 HIV-1 integrase Allosteric inhibitor LEDGF/p75 Dimerization 3-Hydroxypicolinamide
	Design and discovery of flavonoid-based HIV-1 integrase inhibitors targeting both the active site and the interaction with LEDGF/p75 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 卷号: 22, 期号: 12, 页码: 3146-3158 作者: Li, Bo-Wen; Zhang, Feng-Hua; Serrao, Erik; Chen, Huan; Sanchez, Tino W. \| 收藏 \| 浏览/下载：25/0 \| 提交时间：2019/01/08 HIV-1 integrase inhibitors Flavonoid Chelation Strand transfer LEDGF/p75
	Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase-LEDGF/p75 interaction 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 19, 页码: 5963-5972 作者: Serrao, Erik; Xu, Zhong-Liang; Debnath, Bikash; Christ, Frauke; Debyser, Zeger \| 收藏 \| 浏览/下载：25/0 \| 提交时间：2019/01/08 HIV-1 Integrase LEDGF/p75 5-carbonyl-1H-Imidazole-4-carboxamide Protein-protein interaction Antiviral PDB ID code2B4J
	Repositioning HIV-1 Integrase Inhibitors for Cancer Therapeutics: 1,6-Naphthyridine-7-carboxamide as a Promising Scaffold with Drug-like Properties 期刊论文 OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 22, 页码: 9492-9509 作者: Zeng, Li-Fan; Wang, Yong; Kazemi, Roza; Xu, Shili; Xu, Zhong-Liang \| 收藏 \| 浏览/下载：27/0 \| 提交时间：2019/01/08
	Synthesis of the pyridinyl analogues of dibenzylideneacetone (pyr-dba) via an improved Claisen-Schmidt condensation, displaying diverse biological activities as curcumin analogues 期刊论文 OAI收割 ORGANIC & BIOMOLECULAR CHEMISTRY, 2012, 卷号: 10, 期号: 6, 页码: 1239-1245 作者: Cao, Bin; Wang, Yong; Ding, Kan; Neamati, Nouri; Long, Ya-Qiu \| 收藏 \| 浏览/下载：22/0 \| 提交时间：2019/01/08
	基于1,6-二氮杂萘的聚焦型化合物库:新机理酪氨酸激酶抑制剂和HIV-1整合酶抑制剂的发现及结构优化会议论文 OAI收割作者: 王勇; 张凤华; 曾立凡; 谢华; Nouri Neamati \| 收藏 \| 浏览/下载：36/0 \| 提交时间：2019/01/08 1,6-二氮杂萘聚焦型化合物库 HIV-1整合酶酪氨酸激酶抑制剂 LEDGF/p75 c-Src激酶
	Design of HIV-1 integrase inhibitors targeting the catalytic domain as well as its interaction with LEDGF/p75: A scaffold hopping approach using salicylate and catechol groups 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 16, 页码: 4935-4952 作者: Fan, Xing; Zhang, Feng-Hua; Al-Safi, Rasha I.; Zeng, Li-Fan; Shabaik, Yumna \| 收藏 \| 浏览/下载：26/0 \| 提交时间：2019/01/08 HIV-1 integrase inhibitors 2,3-Dihydroxybenzamide Strand transfer 3 '-Process LEDGF/p75 Chelation
	Novel dimeric aryldiketo containing inhibitors of HIV-1 integrase: Effects of the phenyl substituent and the linker orientation 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 卷号: 16, 期号: 16, 页码: 7777-7787 作者: Zeng, Li-Fan; Jiang, Xiao-Hua; Sanchez, Tino; Zhang, Hu-Shan; Dayam, Raveendra \| 收藏 \| 浏览/下载：21/0 \| 提交时间：2019/01/08 HIV-1 integrase inhibitors aryl diketoacid strand transfer dimer conformationally constrained linker orientation substitution effect
	Efficient synthesis and utilization of phenyl-substituted heteroaromatic carboxylic acids as aryl diketo acid isosteres in the design of novel HIV-1 integrase inhibitors 期刊论文 OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 卷号: 18, 期号: 16, 页码: 4521-4524 作者: Zeng, Li-Fan; Zhang, Hu-Shan; Wang, Yun-Hua; Sanchez, Tino; Zheng, Yong-Tang \| 收藏 \| 浏览/下载：14/0 \| 提交时间：2019/01/08 HIV-1 integrase inhibitor bioisostere heteroaromatic carboxylic acid isoxazole isothiazole 1H-pyrazole bioavailability antiviral effect