中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [140]
新疆理化技术研究所 [13]
生物物理研究所 [1]
中国科学院大学 [1]
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期刊论文 [155]
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2024 [5]
2023 [16]
2022 [18]
2021 [16]
2020 [11]
2019 [16]
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An Improved Iodine-Catalyzed Aromatization Reaction and Its Application in the Synthesis of a Key Intermediate of Cannabidiol
期刊论文
OAI收割
SYNLETT, 2024, 页码: 6
作者:
Abduahadi, Safomuddin
;
Bonku, Emmanuel Mintah
;
Qin, Hongjian
;
Odilov, Abdullajon
;
Zhu, Fuqiang
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
methyl olivetolate
potassium persulfate
aromatization
oxidation
iodine-catalyst
cannabidiol
Identification of Dihydrobenzofuran Neolignans as Novel PDE4 Inhibitors and Evaluation of Antiatopic Dermatitis Efficacy in DNCB-Induced Mice Model
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 6, 页码: 4855-4869
作者:
Gu, Chenming
;
Liu, Jiayuan
;
Qian, Fei
;
Yu, Wenchao
;
Huang, Doudou
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Improved and ligand-free copper-catalyzed cyclization for an efficient synthesis of benzimidazoles from
o
-bromoarylamine and nitriles
期刊论文
OAI收割
RSC ADVANCES, 2024, 卷号: 14, 期号: 10, 页码: 6906-6916
作者:
Bonku, Emmanuel Mintah
;
Qin, Hongjian
;
Odilov, Abdullajon
;
Abduahadi, Safomuddin
;
Guma, Samuel Desta
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/07
Discovery of a CB2 and 5-HT1A receptor dual agonist for the treatment of depression and anxiety
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 20
作者:
Yang, Wenjiao
;
Gong, Xudong
;
Sun, Haiguo
;
Wu, Chunhui
;
Suo, Jin
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/03/06
CB2R agonist
5-HT1AR agonist
CB1R antagonist
Antidepressant
Anxiolytic
Oral Simnotrelvir for Adult Patients with Mild-to-Moderate Covid-19
期刊论文
OAI收割
NEW ENGLAND JOURNAL OF MEDICINE, 2024, 卷号: 390, 期号: 3, 页码: 230-241
作者:
Cao, Bin
;
Wang, Yeming
;
Lu, Hongzhou
;
Huang, Chaolin
;
Yang, Yumei
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
Repurposing of Rutan showed effective treatment for COVID-19 disease
期刊论文
OAI收割
FRONTIERS IN MEDICINE, 2023, 卷号: 10, 页码: 13
作者:
Salikhov, Shavkat I.
;
Abdurakhmonov, Ibrokhim Y.
;
Oshchepkova, Yuliya I.
;
Ziyavitdinov, Jamolitdin F.
;
Berdiev, Nodir Sh.
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/26
COVID-19
SARS-CoV-2
3CLpro
RdRp
Rhus coriaria
Rutan
clinical trial
An efficient synthesis of the last step key intermediate for telmisartan via Pd-catalyzed carbonylative cyclization
期刊论文
OAI收割
TETRAHEDRON, 2023, 卷号: 148, 页码: 8
作者:
Odilov, Abdullajon
;
Qin, Hongjian
;
Bonku, Emmanuel Mintah
;
Zhu, Fuqiang
;
Yang, Feipu
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/19
Telmisartan
Benzimidazole
Pd-catalyzed
Carbonylative/cyclization
Optimized Synthesis of the Key Intermediate of Telmisartan via the Cyclization of 2-Bromoarylamine with
n
-Butyronitrile
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 卷号: 27, 期号: 11, 页码: 2165-2173
作者:
Qin, Hongjian
;
Mintah Bonku, Emmanuel
;
Odilov, Abdullajon
;
Wu, Mingjun
;
Liu, Yongjian
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/02/27
bis-benzimidazole
cyclization
2-bromoarylamine
n-butyronitrile
telmisartan
design of experiments
Structure-based development and preclinical evaluation of the SARS-CoV-2 3C-like protease inhibitor simnotrelvir
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Jiang, Xiangrui
;
Su, Haixia
;
Shang, Weijuan
;
Zhou, Feng
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/25