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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [14]
武汉物理与数学研究所 [1]
采集方式
OAI收割 [15]
内容类型
期刊论文 [15]
发表日期
2023 [1]
2022 [1]
2016 [1]
2015 [2]
2014 [2]
2013 [3]
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Construction of Diversified Penta-Spiro-Heterocyclic and Fused-Heterocyclic Frameworks with Potent Antitumor Activity
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2023, 页码: 7
作者:
Liu, Qi
;
Liu, Xuyi
;
Li, Yazhou
;
Zhou, Yu
;
Zhao, Linxiang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/10/17
spiro
fused-heterocyclic frameworks
substrate- and pH- controlled strategies
C-H activation
[4+1] and [4+2] annulation
antitumor
indazolone
A substrate-controlled Ru(ii)-catalyzed C-H activation/[5+2] annulation cascade and unusual acyl migration to synthesize diverse indoline scaffolds
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2022, 页码: 6
作者:
Zheng, Miao
;
Zhou, Jianhui
;
Fang, Feifei
;
Xu, Zichao
;
Zheng, Fuqiang
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
Enantioselective N-Heterocyclic Carbene-Catalyzed [3+3] Annulation of ,-Unsaturated Esters with Methyl Ketoimine
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2016, 卷号: 358, 期号: 11, 页码: 1864-1869
作者:
Xia, Wenjing
;
Yao, Hong
;
Liu, Dan
;
Zhao, Linxiang
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
[3+3] annulation
enantioselectivity
N-heterocyclic carbenes
-lactams
-unsaturated esters
Direct access to pyrido/pyrrolo[2,1-b]quinazolin-9(1H)-ones through silver-mediated intramolecular alkyne hydroamination reactions
期刊论文
OAI收割
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 2015, 卷号: 11, 页码: 416-424
作者:
Wang, Hengshuai
;
Jiao, Shengchao
;
Chen, Kerong
;
Zhang, Xu
;
Zhao, Linxiang
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
heterocyclic molecules
intramolecular alkyne hydroamination
silver
Improved synthetic process of JNJ-40411813
期刊论文
OAI收割
Chinese Journal of Medicinal Chemistry, 2015, 卷号: 25, 期号: 4, 页码: 291-294
作者:
Jiao Shenchao
;
Xia Wenjing
;
Liu Dan
;
Zhao Linxiang
;
Zhou Yu
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
JNJ-40411813
JNJ-40411813
mGluR2 PAM
process improvement
Design, synthesis and biological evaluation of 4-fluoropyrrolidine-2-carbonitrile and octahydrocyclopenta[b]pyrrole-2-carbonitrile derivatives as dipeptidyl peptidase IV inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 86, 页码: 242-256
作者:
Ji, Xun
;
Xia, Chunmei
;
Wang, Jiang
;
Su, Mingbo
;
Zhang, Lei
  |  
收藏
  |  
浏览/下载:97/0
  |  
提交时间:2019/01/08
DPP4 inhibitors
GLP-1
Selectivity
Oral bioavailability
Oral glucose tolerance tests
hERG
Design, synthesis and biological evaluation of hetero-aromatic moieties substituted pyrrole-2-carbonitrile derivatives as dipeptidyl peptidase IV inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 75, 页码: 111-122
作者:
Ji, Xun
;
Su, Mingbo
;
Wang, Jiang
;
Deng, Guanghui
;
Deng, Sisi
  |  
收藏
  |  
浏览/下载:87/0
  |  
提交时间:2019/01/08
DPP4 inhibitors
Selectivity
Reversible kinetic characterization
Oral bioavailability
Oral glucose tolerance test
Polyoxometalate-based ionic complexes immobilized in mesoporous silicas prepared via a one-pot procedure: Efficient and reusable catalysts for H2O2-mediated alcohol oxidations in aqueous media
期刊论文
OAI收割
MICROPOROUS AND MESOPOROUS MATERIALS, 2013, 卷号: 172, 页码: 67-76
作者:
Zhao, Haihong
;
Zeng, Linxiang
;
Li, Yunlong
;
Liu, Cheng
;
Hou, Bo
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2015/06/23
Polyoxometalate
Ionic liquid
Immobilization
Mesoporous silica
Alcohol oxidation
Au(I)/Ag(I)-Catalyzed Cascade Approach for the Synthesis of Benzo[4,5]imidazo[1,2-c]pyrrolo[1,2-a]quinazolinones
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2013, 卷号: 78, 期号: 9, 页码: 4312-4318
作者:
Ji, Xun
;
Zhou, Yu
;
Wang, Jinfang
;
Zhao, Linxiang
;
Jiang, Hualiang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Application of phosphates and phosphonates prodrugs in drug research and development
期刊论文
OAI收割
Acta Pharmaceutica Sinica, 2013, 卷号: 48, 期号: 5, 页码: 621-634
作者:
Ji Xun
;
Wang Jiang
;
Zhang Lei
;
Zhao Linxiang
;
Jiang Hualiang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
prodrugs of phosphates and phosphonates
bioavailability
lipophilicity
solubility
stability
HepDirect prodrug