中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [26]
上海营养与健康研究所 [8]
水生生物研究所 [1]
西安光学精密机械研究... [1]
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OAI收割 [36]
内容类型
期刊论文 [36]
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2023 [3]
2021 [5]
2020 [6]
2019 [7]
2018 [7]
2017 [5]
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学科主题
Science & ... [5]
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Structure-Based Ligand Discovery Targeting the Transmembrane Domain of Frizzled Receptor FZD7
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
Li, Cuixia
;
Wu, Yiran
;
Wang, Wenli
;
Xu, Lu
;
Zhou, Yan
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2023/10/17
Orthogonally Engineered Albumin with Attenuated Macrophage Phagocytosis for the Targeted Visualization and Phototherapy of Liver Cancer
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 31, 页码: 17377-17388
作者:
Dou, Wei-Tao
;
Qiu, Peng
;
Shi, Yuanyuan
;
Zhu, Ling
;
Guo, Chen
  |  
收藏
  |  
浏览/下载:257/0
  |  
提交时间:2023/10/17
Cryo-EM structures of orphan GPR21 signaling complexes
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:
Xi Lin
;
Bo Chen
;
Yiran Wu
;
Yingqi Han
;
Ao Qi
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/05/22
Structures of the human cholecystokinin receptors bound to agonists and antagonists
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1230-1237
作者:
Zhang, Xuefeng
;
He, Chenglin
;
Wang, Mu
;
Zhou, Qingtong
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/03/21
Structure-Based Design of Dual-Acting Compounds Targeting Adenosine A(2A) Receptor and Histone Deacetylase as Novel Tumor Immunotherapeutic Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16573-16597
作者:
Yan, Wenzhong
;
Ling, Lijun
;
Wu, Yiran
;
Yang, Kexin
;
Liu, Ruiquan
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/06/15
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening
期刊论文
OAI收割
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:
Zhou, Qingtong
;
Guo, Wanjing
;
Dai, Antao
;
Cai, Xiaoqing
;
Vass, Marton
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2021/08/17
GLP-1R
virtual screening
allosteric modulator
drug discovery
molecular docking
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:
Lu, Yan
;
Liu, Hongyue
;
Yang, Dehua
;
Zhong, Li
;
Xin, Ye
  |  
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2021/08/17
G protein-coupled receptors: structure- and function-based drug discovery
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 27
作者:
Yang, Dehua
;
Zhou, Qingtong
;
Labroska, Viktorija
;
Qin, Shanshan
;
Darbalaei, Sanaz
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:
Ma, Mengna
;
Guo, Shimeng
;
Lin, Xi
;
Li, Shanshan
;
Wu, Yiran
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2021/05/24
A unique hormonal recognition feature of the human glucagon-like peptide-2 receptor
期刊论文
OAI收割
CELL RESEARCH, 2020, 页码: 11
作者:
Sun, Wen
;
Chen, Li-Nan
;
Zhou, Qingtong
;
Zhao, Li-Hua
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:126/0
  |  
提交时间:2020/12/24