中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共66条,第1-10条 帮助

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Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:  
Zeng, Yanping;  Xiao, Jian;  Shi, Li;  Li, Yangsha;  Xu, Yuanxin
  |  收藏  |  浏览/下载:38/0  |  提交时间:2025/04/01
BET inhibitor and CDK4/6 inhibitor synergistically inhibit breast cancer by suppressing BRD4 stability and DNA damage repair 期刊论文  OAI收割
TRANSLATIONAL ONCOLOGY, 2025, 卷号: 51, 页码: 11
作者:  
Chi, Shuaishuai;  Wei, Fan;  Li, Yangsha;  Yu, Lei;  Ma, Chuyao
  |  收藏  |  浏览/下载:9/0  |  提交时间:2025/01/06
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 20
作者:  
Wang, Yafang;  Xu, Lansong
  |  收藏  |  浏览/下载:21/0  |  提交时间:2024/10/21
Discovery of novel CDK9 inhibitor with tridentate ligand: Design, synthesis and biological evaluation 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 150, 页码: 12
作者:  
Zhong, Ye;  Xu, Jing;  Ding, Shaoyue;  Cao, Huiying;  Zhang, Yufei
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/08/22
Design, Synthesis, and Biological Evaluation of 2,4-Diaminopyrimidine Derivatives as Potent CDK7 Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 页码: 8
作者:  
Zhang, Hualin;  Tu, Yutong;  Tao, Zhaofan;  Gao, Lixin;  Huang, Shengjie
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/08/22
The anticancer potential of chemical constituents of Moringa oleifera targeting CDK-2 inhibition in estrogen receptor positive breast cancer using in-silico and in vitro approches 期刊论文  OAI收割
BMC COMPLEMENTARY MEDICINE AND THERAPIES, 2023, 卷号: 23, 期号: 1, 页码: 17
作者:  
Sultan, Rida;  Ahmed, Abrar;  Wei, Li;  Saeed, Hamid;  Islam, Muhammad
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/12/19
LINC00955 suppresses colorectal cancer growth by acting as a molecular scaffold of TRIM25 and Sp1 to Inhibit DNMT3B-mediated methylation of the PHIP promoter 期刊论文  OAI收割
BMC CANCER, 2023, 卷号: 23, 期号: 1, 页码: 20
作者:  
Ren, Ganglin;  Li, Hongyan;  Hong, Dan;  Hu, Fangyu;  Jin, Rongjia
  |  收藏  |  浏览/下载:22/0  |  提交时间:2023/12/08
Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:  
Hua, Chen;  Shena, Lijuan;  Zoua, Fengming;  Wua, Yun;  Wanga, Beilei
  |  收藏  |  浏览/下载:28/0  |  提交时间:2023/11/10
Discovery of HyT-Based Degraders of CDK9-Cyclin T1 Complex 期刊论文  OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 页码: 10
作者:  
Lin, Rongkun;  Yang, Jie;  Liu, Ting;  Wang, Mingyu
  |  收藏  |  浏览/下载:40/0  |  提交时间:2023/10/17
New Monoterpenoid Indole Alkaloids from Tabernaemontana crassa Inhibit beta-Amyloid42 Production and Phospho-Tau (Thr217) 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2023, 卷号: 24, 期号: 2, 页码: 1487
作者:  
Li,Sheng;  Han,Ling-Ling;  Huang,Ke-Pu;  Ma,Ye-Han;  Guo,Ling-Li
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/05/09