中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共13条,第1-10条 帮助

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Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:  
Zeng, Yanping;  Xiao, Jian;  Shi, Li;  Li, Yangsha;  Xu, Yuanxin
  |  收藏  |  浏览/下载:33/0  |  提交时间:2025/04/01
Unraveling the CDK9/PP2A/ERK Network in Transcriptional Pause Release and Complement Activation in KRAS-mutant Cancers 期刊论文  OAI收割
ADVANCED SCIENCE, 2024, 页码: 20
作者:  
Wang, Yafang;  Xu, Lansong;  Ling, Lijun;  Yao, Mingyue;  Shi, Shangxuan
  |  收藏  |  浏览/下载:18/0  |  提交时间:2024/10/21
Discovery of novel CDK9 inhibitor with tridentate ligand: Design, synthesis and biological evaluation 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 150, 页码: 12
作者:  
Zhong, Ye;  Xu, Jing;  Ding, Shaoyue;  Cao, Huiying;  Zhang, Yufei
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/08/22
Predicting and overcoming resistance to CDK9 inhibitors for cancer therapy 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13
作者:  
Hua, Chen;  Shena, Lijuan;  Zoua, Fengming;  Wua, Yun;  Wanga, Beilei
  |  收藏  |  浏览/下载:28/0  |  提交时间:2023/11/10
Discovery of HyT-Based Degraders of CDK9-Cyclin T1 Complex 期刊论文  OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 页码: 10
作者:  
Lin, Rongkun;  Yang, Jie;  Liu, Ting;  Wang, Mingyu;  Ke, Chongrong
  |  收藏  |  浏览/下载:40/0  |  提交时间:2023/10/17
Inhibition of the dopamine transporter promotes lysosome biogenesis and ameliorates Alzheimer's disease-like symptoms in mice 期刊论文  OAI收割
ALZHEIMERS & DEMENTIA, 2022, 页码: 15
作者:  
Yin, Limin;  Zhou, Jianhui;  Li, Tianyou;  Wang, Xinghua;  Xue, Wenlong
  |  收藏  |  浏览/下载:91/0  |  提交时间:2022/11/11
Efficient Synthesis and Docking Analysis of Selective CDK9 Inhibitor NVP-2 期刊论文  OAI收割
Pharmaceutical Fronts, 2021, 期号: 3, 页码: E50-E55
作者:  
Saidahmatov, Abdusaid;  Liang, Xue-Wu;  Shi, Yuqiang;  Han, Xu;  Liu, Hong
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/03/14
Discovery of selective CDK9 degraders with enhancing antiproliferative activity through PROTAC conversion 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 11
作者:  
Qiu, Xiaqiu;  Li, Yuanqing;  Yu, Bin;  Ren, Jie;  Huang, Huidan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2021/05/24
CDK9  Antitumor  PROTAC  AML  Degrader  
Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:  
Wang, Jubo
  |  收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
CDK9 modulates circadian clock by attenuating REV-ERB alpha activity 期刊论文  OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2019, 卷号: 513, 期号: 4, 页码: 967-973
作者:  
Ou, Jiali;  Li, Huilin;  Tang, Yun-Chi;  Qiu, Peiyuan;  Li, Qing
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/12/09