中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
化学研究所 [1]
采集方式
OAI收割 [6]
内容类型
期刊论文 [6]
发表日期
2024 [1]
2021 [1]
2019 [2]
2011 [1]
2008 [1]
学科主题
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The effect of malaria-induced alteration of metabolism on piperaquine disposition in Plasmodium yoelii infected mice and predicted in malaria patients
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS, 2024, 卷号: 64, 期号: 1, 页码: 11
作者:
Xie, Yuewu
;
Zhang, Yifan
;
Lin, Feifei
;
Chen, Xiaoyue
;
Xing, Jie
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/08/22
Malaria
Drug metabolizing enzymes
Piperaquine
Clearance
PBPK modelling
Metabolic map of the antiviral drug podophyllotoxin provides insights into hepatotoxicity
期刊论文
OAI收割
XENOBIOTICA, 2021, 页码: 13
作者:
Sun, Dongxue
;
Gao, Xiaoxia
;
Wang, Qiao
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2021/11/04
CYP
podophyllotoxin metabolism
liver microsomes
recombinant drug-metabolizing enzymes
hepatic and intestinal toxicity
Current trends in drug metabolism and pharmacokinetics
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2019, 卷号: 9, 期号: 6, 页码: 1113-1144
作者:
Li, Yuhua
;
Meng, Qiang
;
Yang, Mengbi
;
Liu, Dongyang
;
Hou, Xiangyu
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2020/07/01
Pharmacokinetics
Drug metabolism
Drug-drug interactions
Modeling
Metabolizing enzymes
Transporters
Nuclear receptors
Noncoding RNAs
currenttrendsindrugmetabolismandpharmacokinetics
期刊论文
OAI收割
actapharmaceuticasinicab, 2019, 卷号: 9, 期号: 6, 页码: 1113
作者:
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/07/01
ARYL-HYDROCARBON RECEPTOR
BLOOD-BRAIN-BARRIER
ORGANIC ANION TRANSPORTERS
CHRONIC KIDNEY-DISEASE
PREGNANE-X-RECEPTOR
P-GLYCOPROTEIN
QUANTITATIVE PREDICTION
CYTOCHROME-P450 ENZYMES
DOWN-REGULATION
IN-VIVO
Pharmacokinetics
Drug metabolism
Drug-drug interactions
Modeling
Metabolizing enzymes
Transporters
Nuclear receptors
Noncoding RNAs
An Examination of the Potential Effect of Lipids on the First-Pass Metabolism of the Lipophilic Drug Anethol Trithione
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL SCIENCES, 2011, 卷号: 100, 期号: 11, 页码: 5048-5058
作者:
Yu, Hong-Zhen
;
Han, Si-Fei
;
Li, Ping
;
Zhu, Chun-Liu
;
Zhang, Xin-Xin
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
anethol trithione
medium chain triglycerides
first-pass metabolism
hepatic metabolism
nonlinear pharmacokinetics
dose proportionality
drug metabolizing enzymes
inhibition
formulation
lipids
Function prediction for DNA-/RNA-binding proteins, GPCRs, and drug ADME-associated proteins by SVM
期刊论文
OAI收割
PROTEIN AND PEPTIDE LETTERS, 2008, 卷号: 15, 期号: 5, 页码: 463-468
作者:
Cai, Congzhong
;
Xiao, Hanguang
;
Yuan, Qianfei
;
Liu, Xinghua
;
Wen, Yufeng
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/04/09
Protein Function Prediction
Dna-binding Proteins
Rna-binding Proteins
G-protein Coupled Receptors (Gpcrs)
Drug Absorption Proteins
Drug Metabolizing Enzymes
Drug Distribution And Excretion Proteins
Support Vector Machine (Svm)