中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
上海神经科学研究所 [5]
上海生物化学与细胞生... [4]
金属研究所 [3]
昆明植物研究所 [2]
长春应用化学研究所 [2]
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OAI收割 [29]
内容类型
期刊论文 [29]
发表日期
2022 [1]
2021 [3]
2019 [1]
2018 [4]
2015 [1]
2014 [2]
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Biochemist... [4]
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浏览/检索结果:
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Necrosulfonamide Selectively Induces DNA Double-Strand Breaks in Acute Myeloid Leukemia Cells
期刊论文
OAI收割
CHEMICAL RESEARCH IN TOXICOLOGY, 2022, 卷号: 35, 期号: 3, 页码: 387-391
作者:
Chen, Shaokun
;
Lai, Weiyi
;
Li, Xiangjun
;
Wang, Hailin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/11/08
MIXED LINEAGE KINASE
INHIBITION
APOPTOSIS
PROTEIN
REPAIR
NECROPTOSIS
CANCER
DAMAGE
DEATH
Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:
Liu, Xiao
;
Yang, Su
;
Hart, Jonathan R.
;
Xu, Yingna
;
Zou, Xinyu
  |  
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2022/01/04
phosphoinositide 3-kinase (PI3K)
activation
inhibition
activity-dependent conformational changes
Alteration of the PKA-CREB cascade in the mPFC accompanying prepulse inhibition deficits: evidence from adolescent social isolation and chronic SKF38393 injection during early adolescence
期刊论文
OAI收割
BEHAVIOURAL PHARMACOLOGY, 2021, 卷号: 32, 期号: 6, 页码: 487-496
作者:
Du, Wei
;
Li, Man
;
Zhou, Hao
;
Shao, Feng
;
Wang, Weiwen
  |  
收藏
  |  
浏览/下载:66/0
  |  
提交时间:2021/09/24
adolescent social isolation
cAMP-dependent protein kinase A
cAMP-response element-binding protein
medial prefrontal cortex
prepulse inhibition
Bitter Melon and Diabetes Mellitus
期刊论文
OAI收割
FOOD REVIEWS INTERNATIONAL, 2021
作者:
Gao,Ya
;
Li,Xian
;
Huang,Yanjie
;
Chen,Jianchao
;
Qiu,Minghua
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2022/04/02
Bitter melon
diabetes mellitus
crude extracts
phyto-metabolites
hypoglycemic mechanism
MOMORDICA-CHARANTIA L.
11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE-1
ALPHA-GLUCOSIDASE INHIBITION
INSULIN-RESISTANCE
ANTIDIABETIC ACTIVITIES
GUT MICROBIOTA
STRUCTURAL-CHARACTERIZATION
PHENOLIC-COMPOUNDS
OXIDATIVE STRESS
PROTEIN-KINASE
Structural Basis for the Inhibition of the Autophosphorylation Activity of HK853 by Luteolin
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 5, 页码: 11
作者:
Jiang, Ling
;
Liu, Yixiang
;
Liu, Maili
;
Li, Conggang
;
Luo, Liang
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2019/06/24
two-component system
histidine kinase
luteolin
ATP
NMR
molecular docking
inhibition
Targeting HER2 Aberrations in Non-Small Cell Lung Cancer with Osimertinib
期刊论文
OAI收割
CLINICAL CANCER RESEARCH, 2018, 卷号: 24, 期号: 11, 页码: 2594-2604
作者:
Liu, Shengwu
;
Hai, Josephine
;
Wang, Xiaoen
;
Quinn, Max M.
;
Gao, Peng
  |  
收藏
  |  
浏览/下载:97/0
  |  
提交时间:2019/04/28
Receptor Tyrosine Kinase
Phase-ii Trial
Bromodomain Inhibition
Combination Therapy
Acquired-resistance
Domain Mutations
Bet Bromodomains
Breast-cancer
Egfr
Mutant
A novel USP9X substrate TTK contributes to tumorigenesis in non-small-cell lung cancer
期刊论文
OAI收割
THERANOSTICS, 2018, 卷号: 8, 期号: 9, 页码: 2348-2360
作者:
Chen, Xiangling
;
Yu, Chengli
;
Gao, Jing
;
Zhu, Hongwen
;
Zhou, Yanting
  |  
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2019/04/28
Deubiquitinase Inhibition
Chromosomal Instability
Ubiquitin Ligases
Stability
Expression
Kinase
Mps1
Proliferation
Degradation
Centrosome
UTX is an escape from X-inactivation tumor-suppressor in B cell lymphoma
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2018, 卷号: 9, 期号: 1, 页码: -
作者:
Li, Xiaoxi
;
Zhang, Yanli
;
Liu, Mingxian
;
Jiang, Hai
;
Zheng, Liting
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2019/04/28
Acute Lymphoblastic-leukemia
H3k27me3 Demethylase Utx
Tyrosine Kinase
Cancer
Mutations
Cytarabine
Inhibition
Landscape
Carcinoma
Genes
targetingthepi3kaktmtorsignalingpathwaybypterostilbeneattenuatesmantlecelllymphomaprogression
期刊论文
OAI收割
actabiochimicaetbiophysicasinica, 2018, 卷号: 50, 期号: 8, 页码: 782
作者:
Yu Dandan
;
Zhang Yong
;
Chen Gege
;
Xie Yongsheng
;
Xu Zhijian
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/07/01
PROTEIN-KINASE PATHWAY
CANCER IN-VITRO
TRANSDUCTION PATHWAYS
CYCLE ARREST
APOPTOSIS
ACTIVATION
PATHOGENESIS
INHIBITION
ANTICANCER
EXPRESSION
mantle cell lymphoma
pterostilbene
antiproliferative activity
PI3K/Akt/mTOR pathway
synergistic cytotoxicity
Synthesis and Anticancer Activity of 7,8-dihydroxy-4-arylcoumarins
期刊论文
OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2015, 卷号: 12, 期号: 5, 页码: 366-373
作者:
Wu, Jianrui
;
Peng, Ting
;
Chen, Fang
;
Leng, Yixin
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
Anticancer
4-Arylcoumarin
Cytotoxicity
Structure-activity relationship
Tubulin
Tyrosine kinase inhibition