中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
长春应用化学研究所 [2]
烟台海岸带研究所 [2]
西双版纳热带植物园 [1]
上海应用物理研究所 [1]
武汉植物园 [1]
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OAI收割 [15]
内容类型
期刊论文 [15]
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2024 [2]
2022 [2]
2019 [1]
2018 [1]
2016 [1]
2015 [1]
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Biochemist... [2]
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Synchrotron Radiation: A Key Tool for Drug Discovery
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 114, 页码: 10
作者:
Li, Fengcheng
;
Liu, Runze
;
Li, Wenjun
;
Xie, Mingyuan
;
Qin, Song
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/12/06
Synchrotron radiation
Drug discovery
Protein crystals
Structure determination
Ligand screening
Synchrotron Radiation: A Key Tool for Drug Discovery
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 114, 页码: 10
作者:
Li, Fengcheng
;
Liu, Runze
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/12/06
Synchrotron radiation
Drug discovery
Protein crystals
Structure determination
Ligand screening
Recent progress in fragment-based drug discovery facilitated by NMR spectroscopy
期刊论文
OAI收割
Magnetic Resonance Letters, 2022, 卷号: 2, 期号: 2, 页码: 107-118
作者:
Wang, Lei
;
Gao, Jia
;
Ma, Rongsheng
;
Liu, Yaqian
;
Liu, Mingqing
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/03/14
Fragment-based lead/drug discovery
NMR spectroscopy
Protein-ligand interaction
Complex structure
Hit-to-lead evolution
Evaluation of the binding performance of flavonoids to estrogen receptor alpha by Autodock, Autodock Vina and Surflex-Dock
期刊论文
OAI收割
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2022, 卷号: 233, 期号: 0, 页码: 113323
作者:
Xue, Qiao
;
Liu, Xian
;
Russell, Paul
;
Li, Jin
;
Pan, Wenxiao
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/11/08
PROTEIN-LIGAND DOCKING
MOLECULAR DOCKING
DISCOVERY
FRAMEWORK
DYNAMICS
AFFINITY
Advances in MS Based Strategies for Probing Ligand-Target Interactions: Focus on Soft Ionization Mass Spectrometric Techniques
期刊论文
OAI收割
FRONTIERS IN CHEMISTRY, 2019, 卷号: 7, 页码: 17
作者:
Chen, Guilin
;
Fan, Minxia
;
Liu, Ye
;
Sun, Baoqing
;
Liu, Meixian
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/10/04
ligand-target interactions
mass spectrometry
soft ionization
drug discovery
ESI-MS
MALDI-MS
Structural studies and drug discovery of G protein-coupled receptors
期刊论文
OAI收割
Chinese Science Bulletin, 2018, 卷号: 63, 期号: 14, 页码: 1362-1373
作者:
Yang Zhenlin
;
Wu Beili
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
G protein-coupled receptor
drug target
3D structure
ligand
structure-based drug discovery
Counting on natural products for drug design
期刊论文
OAI收割
NATURE CHEMISTRY, 2016, 卷号: 8, 期号: 6, 页码: 531-541
Rodrigues, T
;
Reker, D
;
Schneider, P
;
Schneider, G
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2017/01/12
CATALYTIC ENANTIOSELECTIVE SYNTHESIS
INSPIRED COMPOUND COLLECTION
DIVERSITY-ORIENTED SYNTHESIS
RELEVANT CHEMICAL SPACE
TARGET PREDICTION
MACROMOLECULAR TARGETS
COMBINATORIAL LIBRARY
NETWORK PHARMACOLOGY
MEDICINAL CHEMISTRY
LIGAND DISCOVERY
The Universal Statistical Distributions of the Affinity, Equilibrium Constants, Kinetics and Specificity in Biomolecular Recognition
期刊论文
OAI收割
plos computational biology, 2015, 卷号: 11, 期号: 4, 页码: 5493-5497
作者:
Zheng,Xiliang
;
Wang,Jin
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2016/05/12
SINGLE-MOLECULE DYNAMICS
RANDOM-ENERGY-MODEL
PROTEIN-FOLDING FUNNELS
3-HELIX BUNDLE PROTEIN
DRUG DISCOVERY
COMBINATORIAL TECHNOLOGIES
ENZYMATIC DYNAMICS
INTERFACE BINDING
LANDSCAPE MODEL
LIGAND-BINDING
Identification of a new series of potent diphenol HSP90 inhibitors by fragment merging and structure-based optimization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 11, 页码: 2525—2529
Ren, J
;
Li, J
;
Wang, YQ
;
Chen, WY
;
Shen, AJ
;
Liu, HC
;
Chen, DQ
;
Cao, DY
;
Li, YL
;
Zhang, NX
;
Xu, YC
;
Geng, MY
;
He, JH
;
Xiong, B
;
Shen, JK
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2015/03/13
SHOCK-PROTEIN 90
DRUG DISCOVERY
CHAPERONE
LIGAND
HEAT-SHOCK-PROTEIN-90
DESIGN