中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共17条,第1-10条 帮助

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Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L 期刊论文  OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:  
Li, Xin;  Wu, Xiaowei;  Nie, Shenyou;  Zhao, Jidong;  Yao, Yuan
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/12/19
Characterization of functional transposable element enhancers in acute myeloid leukemia 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2020, 卷号: 63, 期号: 5, 页码: 675-687
作者:  
Zeng, Yingying;  Cao, Yaqiang;  Liu, Denghui;  Zhang, Xiaoli
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/12/21
The Development of Inhibitors Targeting the Mixed Lineage Leukemia 1 (MLL1)-WD Repeat Domain 5 Protein (WDR5) Protein-Protein Interaction 期刊论文  OAI收割
CURRENT MEDICINAL CHEMISTRY, 2020, 卷号: 27, 期号: 33, 页码: 5530-5542
作者:  
Ye, Xiaoqing;  Chen, Gang;  Jin, Jia;  Zhang, Binzhong;  Wang, Yinda
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/12/24
Targeting epigenetic machinery: Emerging novel allosteric inhibitors 期刊论文  OAI收割
PHARMACOLOGY & THERAPEUTICS, 2019, 卷号: 204, 页码: 24
作者:  
Ye, Fei;  Huang, Jing;  Wang, Hongbo;  Luo, Cheng;  Zhao, Kehao
  |  收藏  |  浏览/下载:33/0  |  提交时间:2020/07/01
Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847
作者:  
Wang, Xiaowen;  Su, Mingbo;  Li, You;  Liu, Tongchao;  Wang, Yujie
  |  收藏  |  浏览/下载:22/0  |  提交时间:2020/07/01
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  
Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
  |  收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1751-1758
作者:  
Song, Yakai;  Li, Linjuan;  Chen, Yantao;  Liu, Jingqiu;  Xiao, Senhao
  |  收藏  |  浏览/下载:60/0  |  提交时间:2019/01/08
Piribedil disrupts the MLL1-WDR5 interaction and sensitizes MLL-rearranged acute myeloid leukemia (AML) to doxorubicin-induced apoptosis 期刊论文  OAI收割
CANCER LETTERS, 2018, 卷号: 431, 页码: 150-160
作者:  
Zhang, Xiong;  Zheng, Xingling;  Yang, Hong;  Yan, Juan;  Fu, Xuhong
  |  收藏  |  浏览/下载:46/0  |  提交时间:2019/01/08
Alkaloid constituents from Viola tianschanica 期刊论文  OAI收割
PHYTOCHEMISTRY, 2017, 卷号: 144, 期号: 12, 页码: 233-242
作者:  
Chen, QB (Chen, Qi-Bin)
  |  收藏  |  浏览/下载:32/0  |  提交时间:2018/01/19
Design and synthesis of benzylpiperidine inhibitors targeting the menin-mll1 interface 期刊论文  iSwitch采集
Bioorganic & medicinal chemistry letters, 2016, 卷号: 26, 期号: 18, 页码: 4472-4476
作者:  
Ren, Jing;  Xu, Wei;  Tang, Le;  Su, Minbo;  Chen, Danqi
收藏  |  浏览/下载:42/0  |  提交时间:2019/05/09