中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [78]
大连化学物理研究所 [22]
海洋研究所 [14]
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期刊论文 [196]
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Diazonium-based derivatization for enhanced detection of phosphorylated metabolites by LC-MS in cells
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2025, 卷号: 255, 页码: 7
作者:
Wang, Yikang
;
Lin, Feifei
;
Zhu, Guozheng
;
Zhou, Xiaoxue
;
Hu, Youhong
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/04/01
Phosphorylated metabolite
Derivatization
Chromatographic separation
Quantitative analysis
LC-MS
Mass balance, metabolism, and pharmacokinetics of [
14
C]amdizalisib, a clinical-stage novel oral selective PI3Kδ inhibitor for the treatment of non-hodgkin's lymphoma, in healthy Chinese volunteers
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2024, 卷号: 15, 页码: 13
作者:
Zhao, Chun-Yang
;
Zhang, Li-Jun
;
Sun, Chan
;
Yu, Cheng-Yin
;
Wang, Jian
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2025/01/06
amdizalisib
PI3K delta kinase
metabolism
mass balance
metabolite identification
pharmacokinetics
safety
Molecular basis of enhanced GLP-1 signaling mediated by GLP-1(9-36) in conjunction with LSN3318839
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 11, 页码: 5069-5073
作者:
Li, Jie
;
Li, Guanyi
;
Mai, Yiting
;
Liu, Xiao
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2025/01/06
GLP-1(9-36)
Cryo-electron microscopy
Metabolite
Allosteric modulation
Gardenia jasminoides
Ellis. Polysaccharides Alleviated Cholestatic Liver Injury by Increasing the Production of Butyric Acid and FXR Activation
期刊论文
OAI收割
PHYTOTHERAPY RESEARCH, 2024, 页码: 13
作者:
Wang, Tianming
;
Tian, Tian
;
Zhu, Zhenyun
;
Fang, Su
;
Zhang, Lincong
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/10/21
bile acid
butyric acid
cholestasis
FXR
Gardenia jasminoides Ellis. polysaccharide
intestinal bacterial metabolite
Simultaneous determination of BGT-002 and its acyl glucuronide metabolite ZM326E-M2 in human plasma by liquid chromatography-tandem mass spectrometry and its application to a pharmacokinetic study
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2024, 卷号: 243, 页码: 8
作者:
Zhu, Xueran
;
Cui, Shumin
;
Liu, Xinjing
;
Zhang, Mei
;
Xie, Zhifu
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/05/31
ATP-Citrate Lyase
BGT-002
Acyl glucuronide metabolite
Pseudo-MRM
LC-MS/MS
Pharmacokinetics
Integrated Metagenomic and Metabolomic Analysis on Two Competing Mussels,
Mytella strigata
and
Perna viridis
, in China
期刊论文
OAI收割
ANIMALS, 2024, 卷号: 14, 期号: 6, 页码: 16
作者:
Zuo, Chenxia
;
Ma, Peizhen
;
Ma, Xiaojie
;
Zhu, Yi
;
Yan, Shaojing
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/06/04
biological invasion
intestinal microbiota
metabolite
enzyme activity
Metabolite characterisation of the peptide-drug conjugate LN005 in liver S9s by UHPLC-Orbitrap-HRMS
期刊论文
OAI收割
XENOBIOTICA, 2024, 页码: 9
作者:
Yuan, Yali
;
Wang, Weiqiang
;
Luo, Jing
;
Tang, Chongzhuang
;
Zheng, Yuandong
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/19
peptide-drug conjugate
PDC
LN005
metabolite identification
liver S9s
Metabolomic insights into neurological effects of BDE-47 exposure in the sea cucumber Apostichopus japonicus
期刊论文
OAI收割
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2023, 卷号: 266, 页码: 11
作者:
Ding, Kui
;
Xu, Qinzeng
;
Zhang, Xuelei
;
Liu, Shilin
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/04/07
Apostichopus japonicus
BDE-47
Nervous system
UPLC-Triple-TOF-MS
Metabolite
Neurotoxicity
Pharmacokinetic and metabolite profile of orally administered anemoside B4 in rats with an improved exposure in formulations of rectal suppository
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2023, 卷号: 315, 页码: 11
作者:
Ye, Yaqing
;
Xue, Mingzhen
;
Tian, Xiaoting
;
Gao, Hongwei
;
Hu, Pei
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
Anemoside B4
Pulsatilla chinensis
metabolite identification
Pharmacokinetics
Rectal suppository
Metabolic profiling of
Apostichopus japonicus
body wall exposed to a typical type of PBDEs: potential health risks and impact on sea cucumber health
期刊论文
OAI收割
FRONTIERS IN MARINE SCIENCE, 2023, 卷号: 10, 页码: 15
作者:
Ding, Kui
;
Zhuo, Pengji
;
Ge, Meiling
;
Liao, Xiaomei
;
Mo, Jing
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/11/30
sea cucumber
BDE-47
body wall
metabolite
metabolic pathway