中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
昆明植物研究所 [2]
金属研究所 [1]
新疆理化技术研究所 [1]
合肥物质科学研究院 [1]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2024 [1]
2019 [1]
2018 [1]
2016 [2]
2015 [2]
2014 [2]
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学科主题
Oncology [1]
Pharmacolo... [1]
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浏览/检索结果:
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Identification of YCH2823 as a novel USP7 inhibitor for cancer therapy
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2024, 卷号: 222, 页码: 11
作者:
Cheng, Yong -Jun
;
Zhuang, Zhen
;
Miao, Yu -Ling
;
Song, Shan -Shan
;
Bao, Xu-Bin
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/05/07
YCH2823
USP7 inhibitor
FT671
BCL6
mTOR inhibitor
Practical synthesis of Vistusertib (AZD2014), an ATP competitive mTOR inhibitor
期刊论文
OAI收割
TETRAHEDRON LETTERS, 2019, 卷号: 60, 期号: 52, 页码: 3
作者:
Shen, Guobing
;
Liu, Miaoqing
;
Lu, Jianjun
;
Meng, Tao
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/07/01
Vistusertib
AZD2014
mTOR inhibitor
3-Acetylbenzoic acid
The mTOR inhibitor AZD8055 overcomes tamoxifen resistance in breast cancer cells by down-regulating HSPB8
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1338-1346
作者:
Shi, Jia-jie
;
Chen, Si-meng
;
Guo, Chen-Liang
;
Li, Yi-xue
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
tamoxifen resistance
HSPB8
AZD8055
estrogen receptor
mTOR inhibitor
Molecular regulation of apoptotic machinery and lipid metabolism by mTORC1/mTORC2 dual inhibitors in preclinical models of HER2+/PIK3CAmut breast cancer
期刊论文
OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 67071-67086
作者:
Qian, Jianchang
;
Chen, Yaqing
;
Meng, Tao
;
Ma, Lanping
;
Meng, Lanfang
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2019/01/08
mTOR kinase inhibitor
mTORC2
apoptosis
lipid metabolism
N-Hydroxyphthalimide exhibits antitumor activity by suppressing mTOR signaling pathway in BT-20 and LoVo cells
期刊论文
OAI收割
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2016, 卷号: 35
作者:
Wang, Min
;
Zhou, Ankun
;
An, Tao
;
Kong, Lingmei
;
Yu, Chunlei
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2016/06/27
N-Hydroxyphthalimide
mTOR
Inhibitor
Cancer
Mitochondrial apoptosis
1 T moderate intensity static magnetic field affects Akt/mTOR pathway and increases the antitumor efficacy of mTOR inhibitors in CNE-2Z cells
期刊论文
OAI收割
SCIENCE BULLETIN, 2015, 卷号: 60, 期号: 24, 页码: 2120-2128
作者:
Zhang, Lei
;
Yang, Xingxing
;
Liu, Juanjuan
;
Luo, Yan
;
Li, Zhiyuan
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2017/10/25
Static Magnetic Field
Cell Proliferation
Mtor
Mtor Inhibitor
Feedback Reactivation
mTOR ATP-competitive inhibitor INK128 inhibits neuroblastoma growth via blocking mTORC signaling
期刊论文
OAI收割
APOPTOSIS, 2015, 卷号: 20, 期号: 1, 页码: 50-62
作者:
Zhang, HY (Zhang, Huiyuan)
;
Dou, J (Dou, Jun)
;
Yu, Y (Yu, Yang)
;
Zhao, YL (Zhao, Yanling)
;
Fan, YH (Fan, Yihui)
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2015/03/11
Neuroblastoma
mTOR inhibitor
INK128
Chemotherapy
Drug resistance
HSP90 inhibitor AUY922 abrogates up-regulation of RTKs by mTOR inhibitor AZD8055 and potentiates its antiproliferative activity in human breast cancer
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF CANCER, 2014, 卷号: 135, 期号: 10, 页码: 2462-2474
作者:
Chen, Si-Meng
;
Guo, Chen-Liang
;
Shi, Jia-Jie
;
Xu, Yi-Chao
;
Chen, Yi
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
mTOR kinase inhibitor
HSP90 inhibitor
breast cancer
receptor tyrosine kinases
drug combination
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:
Huang Qiang
;
Fu Qiangqiang
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/02/02
POTENTIAL ANTITUMOR AGENTS
BIOLOGICAL EVALUATION
INHIBITOR
MTOR
Bis(morpholino-1,3,5-triazine)
Design
Anticancer activity
Identification of two novel inhibitors of mTOR signaling pathway based on high content screening
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2013, 卷号: 72, 期号: 4, 页码: 799-808
作者:
Yan, Juming
;
Zhou, Hongyu
;
Kong, Lingmei
;
Zhang, Jing
;
Zhao, Qinshi
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2013/11/12
mTOR signaling
Inhibitor
High content screening
Cancer
Apoptosis