中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共10条,第1-10条 帮助

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Identification of YCH2823 as a novel USP7 inhibitor for cancer therapy 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2024, 卷号: 222, 页码: 11
作者:  
Cheng, Yong -Jun;  Zhuang, Zhen;  Miao, Yu -Ling;  Song, Shan -Shan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/05/07
Practical synthesis of Vistusertib (AZD2014), an ATP competitive mTOR inhibitor 期刊论文  OAI收割
TETRAHEDRON LETTERS, 2019, 卷号: 60, 期号: 52, 页码: 3
作者:  
Shen, Guobing;  Liu, Miaoqing;  Lu, Jianjun;  Meng, Tao
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
The mTOR inhibitor AZD8055 overcomes tamoxifen resistance in breast cancer cells by down-regulating HSPB8 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1338-1346
作者:  
Shi, Jia-jie;  Chen, Si-meng;  Guo, Chen-Liang;  Li, Yi-xue;  Ding, Jian
  |  收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Molecular regulation of apoptotic machinery and lipid metabolism by mTORC1/mTORC2 dual inhibitors in preclinical models of HER2+/PIK3CAmut breast cancer 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 41, 页码: 67071-67086
作者:  
Qian, Jianchang;  Chen, Yaqing;  Meng, Tao;  Ma, Lanping;  Meng, Lanfang
  |  收藏  |  浏览/下载:45/0  |  提交时间:2019/01/08
N-Hydroxyphthalimide exhibits antitumor activity by suppressing mTOR signaling pathway in BT-20 and LoVo cells 期刊论文  OAI收割
JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH, 2016, 卷号: 35
作者:  
Wang, Min;  Zhou, Ankun;  An, Tao;  Kong, Lingmei;  Yu, Chunlei
收藏  |  浏览/下载:41/0  |  提交时间:2016/06/27
1 T moderate intensity static magnetic field affects Akt/mTOR pathway and increases the antitumor efficacy of mTOR inhibitors in CNE-2Z cells 期刊论文  OAI收割
SCIENCE BULLETIN, 2015, 卷号: 60, 期号: 24, 页码: 2120-2128
作者:  
Zhang, Lei;  Yang, Xingxing;  Liu, Juanjuan;  Luo, Yan;  Li, Zhiyuan
收藏  |  浏览/下载:26/0  |  提交时间:2017/10/25
mTOR ATP-competitive inhibitor INK128 inhibits neuroblastoma growth via blocking mTORC signaling 期刊论文  OAI收割
APOPTOSIS, 2015, 卷号: 20, 期号: 1, 页码: 50-62
作者:  
Zhang, HY (Zhang, Huiyuan);  Dou, J (Dou, Jun);  Yu, Y (Yu, Yang);  Zhao, YL (Zhao, Yanling);  Fan, YH (Fan, Yihui)
收藏  |  浏览/下载:46/0  |  提交时间:2015/03/11
HSP90 inhibitor AUY922 abrogates up-regulation of RTKs by mTOR inhibitor AZD8055 and potentiates its antiproliferative activity in human breast cancer 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF CANCER, 2014, 卷号: 135, 期号: 10, 页码: 2462-2474
作者:  
Chen, Si-Meng;  Guo, Chen-Liang;  Shi, Jia-Jie;  Xu, Yi-Chao;  Chen, Yi
  |  收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety 期刊论文  OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:  
Huang Qiang;  Fu Qiangqiang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2021/02/02
Identification of two novel inhibitors of mTOR signaling pathway based on high content screening 期刊论文  OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2013, 卷号: 72, 期号: 4, 页码: 799-808
作者:  
Yan, Juming;  Zhou, Hongyu;  Kong, Lingmei;  Zhang, Jing;  Zhao, Qinshi
收藏  |  浏览/下载:41/0  |  提交时间:2013/11/12