中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共58条,第1-10条 帮助

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JC-010a, a novel selective SHP2 allosteric inhibitor, overcomes RTK/non-RTK-mediated drug resistance in multiple oncogene-addicted cancers 期刊论文  OAI收割
CANCER LETTERS, 2024, 卷号: 582, 页码: 15
作者:  
Lu, Xuxiu;  Yu, Rilei;  Li, Zhen;  Yang, Mengke;  Dai, Jiajia
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/04/07
DCZ5248, a novel dual inhibitor of Hsp90 and autophagy, exerts antitumor activity against colon cancer (vol 42, pg 132, 2021) 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 1
作者:  
Chen, Xiang-ling;  Liu, Peng;  Zhu, Wei-liang;  Lou, Li-guang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/16
Dipyridamole interacts with the N-terminal domain of HSP90 and antagonizes the function of the chaperone in multiple cancer cell lines 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2023, 卷号: 207, 页码: 16
作者:  
Gao, Jing;  Zhou, Chen;  Zhong, Yan;  Shi, Li;  Luo, Xuanyang
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/04/10
7-aminocephalosporanic acid, a novel HSP90 beta inhibitor, attenuates HFD-induced hepatic steatosis 期刊论文  OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2022, 卷号: 622, 页码: 184-191
作者:  
Zhang, Weitao;  Xue, Hanyue;  Zhou, Chen;  Zheng, Zuguo;  Xing, Mingming
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/12/13
HSP90 N-terminal inhibitors target oncoprotein MORC2 for autophagic degradation and suppress MORC2-driven breast cancer progression 期刊论文  OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 18
作者:  
Yang, Fan;  Sun, Rui;  Hou, Zeng;  Zhang, Fang-Lin;  Xiao, Yi
  |  收藏  |  浏览/下载:39/0  |  提交时间:2022/06/15
Discovery of pseudolaric acid A as a new Hsp90 inhibitor uncovers its potential anticancer mechanism 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 112, 页码: 104963
作者:  
Liu,Jiangxin;  Wu,Xing-De;  Li,Wenyan
  |  收藏  |  浏览/下载:15/0  |  提交时间:2022/04/02
Hsp90 inhibitor-loaded IR780 micelles for mitochondria-targeted mild-temperature photothermal therapy in xenograft models of human breast cancer 期刊论文  OAI收割
CANCER LETTERS, 2021, 卷号: 500
作者:  
Zhang, Tao;  Wu, Bihan;  Akakuru, Ozioma Udochukwu;  Yao, Chenyang;  Sun, Shan
  |  收藏  |  浏览/下载:15/0  |  提交时间:2021/12/01
Injectable Magnetic Liquid-solid Phase Transition Material for MR Imaging and Low-temperature Magnetocaloric Therapy of Osteosarcoma 期刊论文  OAI收割
JOURNAL OF INORGANIC MATERIALS, 2020, 期号: 11, 页码: 1277
作者:  
Xu, D;  Zhu, YF;  Zheng, YY;  Luo, Y;  Chen, HR
  |  收藏  |  浏览/下载:28/0  |  提交时间:2020/12/23
Harnessing the targeting potential of differential radiobiological effects of photon versus particle radiation for cancer treatment 期刊论文  OAI收割
JOURNAL OF CELLULAR PHYSIOLOGY, 2020, 页码: 17
作者:  
Zhang, Jinhua;  Si, Jing;  Gan, Lu;  Zhou, Rong;  Guo, Menghuan
  |  收藏  |  浏览/下载:20/0  |  提交时间:2022/01/12
Design, Synthesis, and Biological Evaluation of HSP90 Inhibitor-SN38 Conjugates for Targeted Drug Accumulation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 10, 页码: 5421-5441
作者:  
Zhu, Shulei;  Shen, Qianqian;  Gao, Yinglei;  Wang, Lei;  Fang, Yanfen
  |  收藏  |  浏览/下载:13/0  |  提交时间:2020/12/24