中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [38]
上海营养与健康研究所 [5]
海洋研究所 [3]
昆明植物研究所 [2]
上海应用物理研究所 [2]
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OAI收割 [58]
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期刊论文 [57]
会议论文 [1]
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2024 [1]
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浏览/检索结果:
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JC-010a, a novel selective SHP2 allosteric inhibitor, overcomes RTK/non-RTK-mediated drug resistance in multiple oncogene-addicted cancers
期刊论文
OAI收割
CANCER LETTERS, 2024, 卷号: 582, 页码: 15
作者:
Lu, Xuxiu
;
Yu, Rilei
;
Li, Zhen
;
Yang, Mengke
;
Dai, Jiajia
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2024/04/07
Acquired resistance
Cancer
NSCLC
JC-010a
SHP2
DCZ5248, a novel dual inhibitor of Hsp90 and autophagy, exerts antitumor activity against colon cancer (vol 42, pg 132, 2021)
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 1
作者:
Chen, Xiang-ling
;
Liu, Peng
;
Zhu, Wei-liang
;
Lou, Li-guang
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/01/16
Dipyridamole interacts with the N-terminal domain of HSP90 and antagonizes the function of the chaperone in multiple cancer cell lines
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2023, 卷号: 207, 页码: 16
作者:
Gao, Jing
;
Zhou, Chen
;
Zhong, Yan
;
Shi, Li
;
Luo, Xuanyang
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
HSP90
ATP competitive inhibitors
Tip-based affinity selection-mass spectrometry
Dipyridamole
Cell cycle regulators
7-aminocephalosporanic acid, a novel HSP90 beta inhibitor, attenuates HFD-induced hepatic steatosis
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2022, 卷号: 622, 页码: 184-191
作者:
Zhang, Weitao
;
Xue, Hanyue
;
Zhou, Chen
;
Zheng, Zuguo
;
Xing, Mingming
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/12/13
7-aminocephalosporanic acid
HSP90 beta
NAFLD
de novo lipogenesis
SPR
HSP90 N-terminal inhibitors target oncoprotein MORC2 for autophagic degradation and suppress MORC2-driven breast cancer progression
期刊论文
OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 18
作者:
Yang, Fan
;
Sun, Rui
;
Hou, Zeng
;
Zhang, Fang-Lin
;
Xiao, Yi
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2022/06/15
breast cancer
chaperone-mediated autophagy
HSP90 inhibitor
MORC2
protein degradation
Discovery of pseudolaric acid A as a new Hsp90 inhibitor uncovers its potential anticancer mechanism
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 112, 页码: 104963
作者:
Liu,Jiangxin
;
Wu,Xing-De
;
Li,Wenyan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/04/02
Pseudolaric acid A
Hsp90 inhibitor
Apoptosis
NMR
Structure-activity relationship
Photoaffinity-based probe
Protein-ligand interaction
MOLECULAR CHAPERONE
PROTEIN
TARGET
CANCER
KINASE
NMR
IDENTIFICATION
SELECTIVITY
BINDING
DESIGN
Hsp90 inhibitor-loaded IR780 micelles for mitochondria-targeted mild-temperature photothermal therapy in xenograft models of human breast cancer
期刊论文
OAI收割
CANCER LETTERS, 2021, 卷号: 500
作者:
Zhang, Tao
;
Wu, Bihan
;
Akakuru, Ozioma Udochukwu
;
Yao, Chenyang
;
Sun, Shan
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/12/01
IR-780 DYE
BIIB021
NANOPARTICLES
METABOLISM
DELIVERY
CELLS
Injectable Magnetic Liquid-solid Phase Transition Material for MR Imaging and Low-temperature Magnetocaloric Therapy of Osteosarcoma
期刊论文
OAI收割
JOURNAL OF INORGANIC MATERIALS, 2020, 期号: 11, 页码: 1277
作者:
Xu, D
;
Zhu, YF
;
Zheng, YY
;
Luo, Y
;
Chen, HR
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/12/23
Harnessing the targeting potential of differential radiobiological effects of photon versus particle radiation for cancer treatment
期刊论文
OAI收割
JOURNAL OF CELLULAR PHYSIOLOGY, 2020, 页码: 17
作者:
Zhang, Jinhua
;
Si, Jing
;
Gan, Lu
;
Zhou, Rong
;
Guo, Menghuan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/01/12
DNA damage
DNA repair
particle therapy
photon therapy
radiosensitizer
Design, Synthesis, and Biological Evaluation of HSP90 Inhibitor-SN38 Conjugates for Targeted Drug Accumulation
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 10, 页码: 5421-5441
作者:
Zhu, Shulei
;
Shen, Qianqian
;
Gao, Yinglei
;
Wang, Lei
;
Fang, Yanfen
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24