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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [40]
采集方式
OAI收割 [40]
内容类型
期刊论文 [40]
发表日期
2023 [8]
2022 [4]
2021 [5]
2020 [3]
2019 [2]
2018 [4]
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专题:上海药物研究所
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Five undescribed abietane-type diterpenes of Callicarpa macrophylla
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 170, 页码: 10
作者:
Du, Gao-Xiang
;
Chen, Tong
;
Wang, Ge
;
Liu, Ying-Bo
;
Zheng, Liu
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Callicarpa macrophylla
Verbenaceae
Abietane-type diterpenoids
PCSK9
Macrophypene F -J
Selective Electrochemical Benzylic C(sp(3))-H Oxidations in Fluoroalcohols
期刊论文
OAI收割
CHEMISTRYSELECT, 2023, 卷号: 8, 期号: 27, 页码: 4
作者:
Shen, Haiwei
;
Yang, Bo
;
Lin, Jiusheng
;
Zheng, Mingyue
;
Jiang, Hualiang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
C(sp(3))-H oxidation
electrochemical
aryl aldehydes
fluorinated ethers
eco-friendly
Comparative Characterization of the Ginsenosides from Six Panax Herbal Extracts and Their In Vitro Rat Gut Microbial Metabolites by Advanced Liquid Chromatography-Mass Spectrometry Approaches
期刊论文
OAI收割
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2023, 卷号: 71, 期号: 24, 页码: 9391-9403
作者:
Mi, Yue-Guang
;
Xu, Xiao-Yan
;
Hong, Li-Li
;
Jiang, Mei-Ting
;
Chen, Bo-Xue
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/10/17
Panax
multicomponent characterization
quantitative assay
gut microbiota
in vitro biotransformation
liquid chromatography-massspectrometry
Naphthylisoquinoline alkaloids, a new structural template inhibitor of Nav1.7 sodium channel
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 9
作者:
Wang, Qiao-qiao
;
Wang, Long
;
Zhang, Wen-bo
;
Tang, Chun-ping
;
Chen, Xue-qin
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
Nav1.7 channel
naphthylisoquinolines
Ancistrocladus tectorius
dorsal root ganglion neurons
formalin-induced mouse inflammatory pain model
analgesics
Lnc956-TRIM28-HSP90B1 complex on replication forks promotes CMG helicase retention to ensure stem cell genomic stability and embryogenesis
期刊论文
OAI收割
SCIENCE ADVANCES, 2023, 卷号: 9, 期号: 4, 页码: 19
作者:
Zhang, Weidao
;
Tang, Min
;
Wang, Lin
;
Zhou, Hu
;
Gao, Jing
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/10/17
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors
期刊论文
OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:
Zang, Yi
;
Su, Mingbo
;
Wang, Qingxing
;
Cheng, Xi
;
Zhang, Wenru
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
high-throughput screening
SARS
CoV-2
main
papain-like
proteases
Cryo-EM structures of orphan GPR21 signaling complexes
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 1
作者:
Xi Lin
;
Bo Chen
;
Yiran Wu
;
Yingqi Han
;
Ao Qi
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/05/22
Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:
Xie, Xiong
;
Zheng, Yu-Gui
;
Chen, Huan
;
Li, Jian
;
Luo, Rong-Hua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
(-)-Epigallocatechin Gallate is a Noncompetitive Inhibitor of NAD Kinase
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:
Liu, Tonghai
;
Shi, Wenjia
;
Ding, Yiluan
;
Wu, Qiqi
;
Zhang, Bei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/12/13
NAD kinase inhibitor
(-)-epigallocatechin gallate
hydrogen-deuterium exchange mass spectrometry
KRAS