中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [8]
化学研究所 [2]
长春应用化学研究所 [2]
大连化学物理研究所 [1]
昆明植物研究所 [1]
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OAI收割 [15]
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期刊论文 [15]
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2023 [3]
2022 [1]
2020 [1]
2019 [1]
2017 [1]
2014 [1]
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Discovery of 5-trifluoromethyl-2-aminopyrimidine derivatives as potent dual inhibitors of FLT3 and CHK1
期刊论文
OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 14
作者:
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/19
Design, synthesis and biological evaluation of 2-aminopyrimidine derivatives as potent FLT3 inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 96, 页码: 5
作者:
Lian, Xuanmin
;
Gao, Yue
;
Li, Xuemei
;
Wang, Peipei
;
Tong, Lexian
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/11
2-aminopyrimidine
FLT3 inhibitors
MV4-11
FLT3 mutations
Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Li, Xuemei
;
Wang, Peipei
;
Wang, Chang
;
Jin, Tingting
;
Xu, Ran
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
Identification of 2-Aminopyrimidine Derivatives as FLT3 Kinase Inhibitors with High Selectivity over c-KIT
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 4, 页码: 3229-3248
作者:
Tong, Lexian
;
Wang, Peipei
;
Li, Xuemei
;
Dong, Xiaowu
;
Hu, Xiaobei
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2022/08/16
Design and synthesis of novel desfluoroquinolone-aminopyrimidine hybrids as potent anti-MRSA agents with low hERG activity
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 103, 页码: 10
作者:
Song, Runzhe
;
Wang, Yue
;
Wang, Minghui
;
Gao, Ruixuan
;
Yang, Teng
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2020/12/24
Desfluoroquinolone
Aminopyrimidine
Hybrids
Anti-MRSA
hERG activity
Discovery of novel indoleaminopyrimidine NIK inhibitors based on molecular docking-based support vector regression (SVR) model
期刊论文
OAI收割
CHEMICAL PHYSICS LETTERS, 2019, 卷号: 718, 页码: 38-45
作者:
Ye, Qing
;
Li, Qiu
;
Gao, Anhui
;
Ying, Huazhou
;
Cheng, Gang
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收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/07/01
Synthesis, Crystal Structure and Biological Evaluation of 14-O-[(2-chloroacetamide-6-aminopyrimidine-2-yl)thioacetyl] Mutilin
期刊论文
OAI收割
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2017, 卷号: 36, 页码: 1327-1333
作者:
Zhou Xiang
;
Li Xue-Hu
;
Yi Yun-Peng
;
Lu Xi-Hong
;
Wang Liang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/05/31
pleuromutilin derivative
single-crystal structure
antibacterial activities
Discovery of novel type II c-Met inhibitors based on BMS-777607
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 80, 页码: 254-266
作者:
Zhang, Wei
;
Ai, Jing
;
Shi, Dakuo
;
Peng, Xia
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2019/01/08
c-Met
Synthesis
Kinase inhibitor
Preparation and properties of ionic cross-linked sulfonated copolyimide membranes containing pyrimidine groups
期刊论文
OAI收割
POLYMERS FOR ADVANCED TECHNOLOGIES, 2012, 卷号: 23, 期号: 1, 页码: 31-37
作者:
Jin, Rizhe
;
Li, Yuhan
;
Xing, Wei
;
Qiu, Xuepeng
;
Ji, Xiangling
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/04/09
Ionic Cross-linking
Sulfonated Copolyimide
Pyrimidine Group
Fuel Cell
Preparation and properties of ionic cross-linked sulfonated copolyimide membranes containing pyrimidine groups
期刊论文
OAI收割
polymers for advanced technologies, 2012, 卷号: 23, 期号: 1, 页码: 31-37
Jin RZ
;
Li YH
;
Xing W
;
Qiu XP
;
Ji XL
;
Gao LX
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2013/09/03
PROTON-EXCHANGE MEMBRANES
1H-1
FUEL-CELL APPLICATIONS
2
POLYIMIDE IONOMERS
4-TRIAZOLE
ELECTROLYTE MEMBRANES
ACID
CONDUCTIVITY
DIANHYDRIDE
DIAMINES