中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [4]
昆明植物研究所 [1]
采集方式
OAI收割 [5]
内容类型
期刊论文 [5]
发表日期
2024 [1]
2019 [1]
2015 [2]
2013 [1]
学科主题
Chemistry,... [1]
筛选
浏览/检索结果:
共5条,第1-5条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
提交时间升序
提交时间降序
发表日期升序
发表日期降序
题名升序
题名降序
作者升序
作者降序
Discovery of a 1,6-naphthyridin-4-one-based AXL inhibitor with improved pharmacokinetics and enhanced in vivo antitumor efficacy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 17
作者:
Lan, Yaohan
;
Peng, Xia
;
Ji, Yinchun
;
Su, Yi
;
Duan, Wenhu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/27
AXL inhibitor
In vivo antitumor efficacy
6-Naphthyridin-4-one derivatives
Scaffold hopping
Structure-based drug design
Synthesis and In Vitro Antibacterial Activity of Novel Naphthyridinone Derivatives
期刊论文
OAI收割
CHEMISTRYSELECT, 2019, 卷号: 4, 期号: 21, 页码: 6552-6556
作者:
Sun, Bin
;
Chen, Jianwei
;
Ye, Fei
;
Lu, Yaojia
;
Xu, Guiqing
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/07/01
antibacterial activity
C
violaceum ATCC 12472
naphthyridinone derivatives
quorum sensing inhibitory activity
synthesis
Discovery of potent 1H-imidazo[4,5-b]pyridine-based c-Met kinase inhibitors via mechanism-directed structural optimization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 3, 页码: 708-716
作者:
An, Xiao-De
;
Liu, Hongyan
;
Xu, Zhong-Liang
;
Jin, Yi
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
c-Met tyrosine kinase
Small molecule inhibitor
Imidazonaphthyridinone
Imidazopyridine
Binding mode
Pyridone-3-carboxamide
Cyclopropane-1,1-dicarboxamide
Design and synthesis of new 2-arylnaphthyridin-4-ones as potent antitumor agents targeting tumorigenic cell lines
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 90, 页码: 775-787
作者:
Liu, Chin-Yu
;
Cheng, Yung-Yi
;
Chang, Ling-Chu
;
Huang, Li-Jiau
;
Chou, Li-Chen
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2015/06/29
2-Arylnaphthyridin-4-ones
Antitumor agents
Phosphate prodrug
Investigation on the 1,6-naphthyridine motif: discovery and SAR study of 1H-imidazo[4,5-h][1,6]naphthyridin-2(3H)-one-based c-Met kinase inhibitors
期刊论文
OAI收割
ORGANIC & BIOMOLECULAR CHEMISTRY, 2013, 卷号: 11, 期号: 9, 页码: 1545-1562
作者:
Wang, Yong
;
Xu, Zhong-Liang
;
Ai, Jing
;
Peng, Xia
;
Lin, Jian-Ping
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08