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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
化学研究所 [1]
昆明植物研究所 [1]
过程工程研究所 [1]
青岛生物能源与过程研... [1]
合肥物质科学研究院 [1]
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OAI收割 [13]
内容类型
期刊论文 [13]
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2023 [1]
2020 [1]
2017 [2]
2016 [1]
2015 [1]
2014 [2]
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Chemistry,... [1]
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Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:
Wang, Yujie
;
Xu, Keshi
;
Liu, Hongchun
;
Zhang, Wei
;
Hu, Chun
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/19
Auristatin E
beta-Glucuronidase
Antiproliferation
Tumor microenvironment
Oxygen-enriched Fe3O4/Gd2O3 nanopeanuts for tumor-targeting MRI and ROS-triggered dual-modal cancer therapy through platinum (IV) prodrugs delivery
期刊论文
OAI收割
CHEMICAL ENGINEERING JOURNAL, 2020, 卷号: 388
作者:
Zhang, Guilong
;
Zhang, Li
;
Si, Yuanchun
;
Li, Qingdong
;
Xiao, Jianmin
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2020/10/26
Nanopeanut probe
Theranostics
Superimposed effect
Ferroptosis
Apoptosis
Targeted delivery of a guanidine-pendant Pt(IV)-backboned poly-prodrug by an anisamide-functionalized polypeptide
期刊论文
OAI收割
JOURNAL OF MATERIALS CHEMISTRY B, 2017, 卷号: 5, 期号: 48, 页码: 9546-9557
作者:
Li, Shao-Lu
;
Wang, Yaoyi
;
Zhang, Jingfang
;
Wei, Wei
;
Lu, Hua
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/04/09
Targeted delivery of a guanidine-pendant Pt(IV)-backboned poly-prodrug by an anisamide-functionalized polypeptide
期刊论文
OAI收割
JOURNAL OF MATERIALS CHEMISTRY B, 2017, 卷号: 5, 期号: 48, 页码: 9546-9557
作者:
Li, Shao-Lu
;
Wang, Yaoyi
;
Zhang, Jingfang
;
Wei, Wei
;
Lu, Hua
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2018/01/19
Pharmacokinetics in Vitro and in Vivo of Two Novel Prodrugs of Oleanolic Acid in Rats and Its Hepatoprotective Effects against Liver Injury Induced by CCl4
期刊论文
OAI收割
MOLECULAR PHARMACEUTICS, 2016, 卷号: 13, 期号: 5, 页码: 1699-1710
作者:
Yu, Zongjiang
;
Sun, Weizhi
;
Peng, Weibing
;
Yu, Rilei
;
Li, Guoqiang
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2016/07/12
oleanolic acid (OA)
prodrug
hepatoprotective
pharmacokinetics
biodistribution
Design and synthesis of new 2-arylnaphthyridin-4-ones as potent antitumor agents targeting tumorigenic cell lines
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 90, 页码: 775-787
作者:
Liu, Chin-Yu
;
Cheng, Yung-Yi
;
Chang, Ling-Chu
;
Huang, Li-Jiau
;
Chou, Li-Chen
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2015/06/29
2-Arylnaphthyridin-4-ones
Antitumor agents
Phosphate prodrug
Design, Synthesis, and Structure-Activity Relationship Studies of Novel Thioether Pleuromutilin Derivatives as Potent Antibacterial Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 57, 期号: 11, 页码: 4772-4795
作者:
Ling, Chenyu
;
Fu, Liqiang
;
Gao, Suo
;
Chu, Wenjing
;
Wang, Hui
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
Preclinical Evaluation of Antitumor Activity of Acid-Sensitive PEGylated Doxorubicin
期刊论文
OAI收割
acs applied materials & interfaces, 2014, 卷号: 6, 期号: 23, 页码: 21202-21214
Sun, Diankui
;
Ding, Jianxun
;
Xiao, Chunsheng
;
Chen,Jinjin
;
Zhuang,Xiuli
;
Chen,Xuesi
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2015/06/09
INTRACELLULAR DRUG-DELIVERY
CANCER-THERAPY
POLYPEPTIDE NANOGELS
POLYMERIC MICELLES
TARGETED DELIVERY
RATIONAL DESIGN
IN-VITRO
PH
NANOPARTICLES
ANTICANCER
Application of phosphates and phosphonates prodrugs in drug research and development
期刊论文
OAI收割
Acta Pharmaceutica Sinica, 2013, 卷号: 48, 期号: 5, 页码: 621-634
作者:
Ji Xun
;
Wang Jiang
;
Zhang Lei
;
Zhao Linxiang
;
Jiang Hualiang
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
prodrugs of phosphates and phosphonates
bioavailability
lipophilicity
solubility
stability
HepDirect prodrug
Effects of the novel vascular targeting agent MDS-11P on tumor vascularity and its antitumor activity
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2011, 卷号: 82, 期号: 12, 页码: 1832-1842
作者:
Deng, Zhi-Ting
;
Feng, Teng
;
Wang, Peng
;
Qi, Xin
;
Chen, Xue-Hong
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Vascular disrupting agents
MDS-11P
Antitumor
CA4 derivative
Vascularity