中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共215条,第1-10条 帮助

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Discovery of GPX4 inhibitors through FP-based high-throughput screening 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:  
Cao, Yu;  Wu, Bin;  Xu, Ying;  Wang, Mingchen
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/02/27
Discovery of a novel OGT inhibitor through high-throughput screening based on Homogeneous Time-Resolved Fluorescence (HTRF) 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 139, 页码: 12
作者:  
Wu, Xinyu;  Wang, Mingchen;  Cao, Yu;  Xu, Ying;  Yang, Ziqun
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/02/27
An ATG4B inhibitor blocks autophagy and sensitizes Sorafenib inhibition activities in HCC tumor cells 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 84, 页码: 117262
作者:  
Xie, Yanqiu;  Fan, Shijie;  Ni, Dongxuan;  Wan, Wei;  Xu, Pan
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/03/27
Thimerosal, a competitive thioredoxin reductase 1 (TrxR1) inhibitor discovered via high-throughput screening 期刊论文  OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2023, 卷号: 650, 页码: 117-122
作者:  
Ni, Yicheng;  Luo, Zhongyuan;  Lv, Yixin;  Ma, Shuyuan;  Luo, Cheng
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文  OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:  
Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Simulating androgen receptor selection in designer yeast 期刊论文  OAI收割
SYNTHETIC AND SYSTEMS BIOTECHNOLOGY, 2022, 卷号: 7
作者:  
Zhang, Haoran;  Zhang, Lu;  Xu, Yipeng;  Chen, Shaoyong;  Ma, Zhenyi
  |  收藏  |  浏览/下载:18/0  |  提交时间:2022/12/23
(-)-Epigallocatechin Gallate is a Noncompetitive Inhibitor of NAD Kinase 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:  
Liu, Tonghai;  Shi, Wenjia;  Ding, Yiluan;  Wu, Qiqi;  Zhang, Bei
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/12/13
The discovery of a non-competitive GOT1 inhibitor, hydralazine hydrochloride, via a coupling reaction-based high-throughput screening assay 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 73, 页码: 6
作者:  
Wu, Qiqi;  Sun, Zhongya;  Chen, Zhifeng;  Liu, Jingqiu;  Ding, Hong
  |  收藏  |  浏览/下载:53/0  |  提交时间:2022/08/30
Phosphodiesters as GPR84 Antagonists for the Treatment of Ulcerative Colitis 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 3991-4006
作者:  
Chen, Lin-Hai;  Zhang, Qing;  Xiao, Yu-Feng;  Fang, You-Chen;  Xie, Xin
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/06/15
High-Throughput-Methyl-Reading (HTMR) assay: a solution based on nucleotide methyl-binding proteins enables large-scale screening for DNA/RNA methyltransferases and demethylases 期刊论文  OAI收割
NUCLEIC ACIDS RESEARCH, 2022, 卷号: 50, 期号: 2, 页码: 14
作者:  
Xiao, Senhao;  Guo, Siqi;  Han, Jie;  Sun, Yanli;  Wang, Mingchen
  |  收藏  |  浏览/下载:29/0  |  提交时间:2022/06/15