中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共19条,第1-10条 帮助

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Spermine is a natural suppressor of AR signaling in castration-resistant prostate cancer 期刊论文  OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 7, 页码: 24
作者:  
Li, Xiao;  Li, Fei;  Ye, Fei;  Guo, Haotian;  Chen, Wentao
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/10/17
Simulating androgen receptor selection in designer yeast 期刊论文  OAI收割
SYNTHETIC AND SYSTEMS BIOTECHNOLOGY, 2022, 卷号: 7
作者:  
Zhang, Haoran;  Zhang, Lu;  Xu, Yipeng;  Chen, Shaoyong;  Ma, Zhenyi
  |  收藏  |  浏览/下载:18/0  |  提交时间:2022/12/23
Synthesis of Hydantoin Androgen Receptor Antagonists and Study on Their Antagonistic Activity 期刊论文  OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 18, 页码: 22
作者:  
Ma, Longjun;  Zhou, Yan;  Yang, Dehua;  Wang, Ming-Wei;  Lu, Wei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2022/11/11
Discovery of a Novel Androgen Receptor Antagonist Manifesting Evidence to Disrupt the Dimerization of the Ligand-Binding Domain via Attenuating the Hydrogen-Bonding Network Between the Two Monomers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64
作者:  
Fu, Weitao;  Zhang, Minkui;  Liao, Jianing;  Tang, Qing;  Lei, Yixuan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/03/21
Design, synthesis and biological evaluation of novel thiohydantoin derivatives as potent androgen receptor antagonists for the treatment of prostate cancer 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 31, 页码: 13
作者:  
Wang, Ao;  Wang, Yawan;  Meng, Xin;  Yang, Yushe
  |  收藏  |  浏览/下载:12/0  |  提交时间:2021/05/24
Discovery of Novel Androgen Receptor Ligands by Structure-based Virtual Screening and Bioassays 期刊论文  OAI收割
GENOMICS PROTEOMICS & BIOINFORMATICS, 2019, 卷号: 16, 期号: 6, 页码: 416-427
作者:  
Hou, Tingjun;  Li, Dan;  Chang, Shan;  Xu, Lei;  Sun, Huiyong
  |  收藏  |  浏览/下载:260/0  |  提交时间:2019/06/24
Synthesis of androgen receptor antagonists containing a pentafluorosulfanyl (SF5) moiety 期刊论文  OAI收割
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 11
作者:  
Jin, Jiyu;  Zhou, Yan;  Yang, Dehua;  Zhang, Qiumeng;  Wang, Ming-Wei
  |  收藏  |  浏览/下载:69/0  |  提交时间:2019/01/08
CMKLR1 deficiency attenuates androgen-induced lipid accumulation in mice. 期刊论文  OAI收割
Cellular Physiology and Biochemistry, 2018
作者:  
Zhao Huashan;  Wu Linlin;  Huang Chen;  Xiang Liang;  Wang Baobei
  |  收藏  |  浏览/下载:85/0  |  提交时间:2019/01/31
Evaluation and characterization of anti-estrogenic and anti-androgenic activities in soil samples along the Second Songhua River, China 期刊论文  OAI收割
ENVIRONMENTAL MONITORING AND ASSESSMENT, ENVIRONMENTAL MONITORING AND ASSESSMENT, 2015, 2015, 卷号: 187, 187, 期号: 11, 页码: 724, 724
作者:  
Li, J;  Wang, YF;  Kong, DD;  Wang, JS;  Teng, YG
  |  收藏  |  浏览/下载:35/0  |  提交时间:2016/04/18
Development of beta-amino-carbonyl compounds as androgen receptor antagonists 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 664-673
作者:  
Zhang, Zhi-yun;  Zhu, Yan-hui;  Zhou, Cai-hong;  Liu, Qing;  Lu, Hui-li
  |  收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08