中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [15]
上海营养与健康研究所 [4]
过程工程研究所 [1]
武汉物理与数学研究所 [1]
中国科学院大学 [1]
上海生物化学与细胞生... [1]
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期刊论文 [23]
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Selective PPAR gamma modulator diosmin improves insulin sensitivity and promotes browning of white fat
期刊论文
OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023, 卷号: 299, 期号: 4, 页码: 14
作者:
Yu, Jian
;
Hu, Yepeng
;
Sheng, Maozheng
;
Gao, Mingyuan
;
Guo, Wenxiu
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/10/17
Identification and structural insight of an effective PPAR gamma modulator with improved therapeutic index for anti-diabetic drug discovery
期刊论文
OAI收割
CHEMICAL SCIENCE, 2020, 卷号: 11, 期号: 8, 页码: 2260-2268
作者:
Jiang, Haowen
  |  
收藏
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浏览/下载:22/0
  |  
提交时间:2020/07/01
Peroxisome Proliferator-Activated Receptor gamma and Its Role in Adipocyte Homeostasis and Thiazolidinedione-Mediated Insulin Sensitization
期刊论文
OAI收割
MOLECULAR AND CELLULAR BIOLOGY, 2018, 卷号: 38, 期号: 10, 页码: UNSP e00677
作者:
Wang, Qiong A.
;
Zhang, Fang
;
Ye, Risheng
;
An, Yu
;
Shao, Mengle
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/12/09
C/EBP alpha
insulin sensitization
PPAR gamma
thiazolidinedione
adipocyte
adipose tissue
inducible knockout
mouse model
obesity
Identification of a novel selective PPAR gamma ligand with a unique binding mode and improved therapeutic profile in vitro
期刊论文
OAI收割
Scientific Reports, 2017, 卷号: 7
作者:
Yi, Wei
;
Shi, Jingjing
;
Zhao, Guanguan
;
Zhou, X. Edward
;
Suino-Powell, Kelly
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Bavachinin, as a novel natural pan-PPAR agonist, exhibits unique synergistic effects with synthetic PPAR-gamma and PPAR-alpha agonists on carbohydrate and lipid metabolism in db/db and diet-induced obese mice
期刊论文
OAI收割
DIABETOLOGIA, 2016, 卷号: 59, 期号: 6, 页码: 1276-1286
作者:
Feng, Li
;
Luo, Huan
;
Xu, Zhijian
;
Yang, Zhuo
;
Du, Guoxin
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2019/01/08
Alternative binding site
Bavachinin
Canonical ligand-binding pocket
Carbohydrate metabolism
Lipid metabolism
Pan-PPAR agonist
Synergistic effects
(2S)-7,4 '-dihydroxy-8-prenylflavan stimulates adipogenesis and glucose uptake through p38MAPK pathway in 3T3-L1 cells
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2015, 卷号: 460, 期号: 3, 页码: 578-582
作者:
Ji, Jun
;
Zhu, Jingjie
;
Hu, Xiao
;
Wang, Ting
;
Zhang, Xiaodong
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
(2S)-7,4 '-dihydroxy-8-prenylflavan
Adipogenesis
Glucose uptake
p38MAPK
Type 2 diabetes
Rosiglitazone Causes Cardiotoxicity via Peroxisome Proliferator-Activated Receptor gamma-Independent Mitochondrial Oxidative Stress in Mouse Hearts
期刊论文
OAI收割
TOXICOLOGICAL SCIENCES, 2014, 卷号: 138, 期号: 2, 页码: 468-481
作者:
He, Huamei
;
Tao, Hai
;
Xiong, Hui
;
Duan, ShengZhong(段胜仲)
;
McGowan, Francis X., Jr.
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2015/09/02
Rosiglitazone
PPAR gamma
energy metabolism
cardiac function
mitochondria
oxidative stress
Metabonomic Profiling Revealed an Alteration in Purine Nucleotide Metabolism Associated with Cardiac Hypertrophy in Rats Treated with Thiazolidinediones
期刊论文
OAI收割
JOURNAL OF PROTEOME RESEARCH, 2013, 卷号: 12, 期号: 12, 页码: 5634-5641
作者:
Liu, Yan
;
Yan, Xing
;
Mao, Guangmei
;
Fang, Li
;
Zhao, Beilei
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2015/06/23
thiazolidinediones
PPARy
cardiac hypertrophy
metabonomics
purine nucleotide metabolism
Effects of PPARs Agonists on Cardiac Metabolism in Littermate and Cardiomyocyte-Specific PPAR-gamma - Knockout (CM-PGKO) Mice
期刊论文
OAI收割
PLOS ONE, 2012, 卷号: 7, 期号: 4, 页码: e35999
作者:
Barbieri, Michelangela
;
Di Filippo, Clara
;
Esposito, Antonietta
;
Marfella, Raffaele
;
Rizzo, Maria Rosaria
收藏
  |  
浏览/下载:16/0
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提交时间:2015/09/02