中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [5]
上海营养与健康研究所 [2]
武汉病毒研究所 [1]
昆明植物研究所 [1]
合肥物质科学研究院 [1]
采集方式
OAI收割 [9]
iSwitch采集 [1]
内容类型
期刊论文 [10]
发表日期
2019 [10]
学科主题
Cardiovasc... [1]
Science & ... [1]
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共10条,第1-10条
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发表日期:2019
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Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:
Wang, Jubo
;
Li, Tinghan
;
Zhao, Tengteng
;
Wu, Tizhi
;
Liu, Chuang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
Wogonin
CDK9
AML
Flavonoid
Antitumor
Pharmacological characterization of TQ05310, a potent inhibitor of isocitrate dehydrogenase 2 R140Q and R172K mutants
期刊论文
OAI收割
CANCER SCIENCE, 2019, 页码: 9
作者:
Gao, Mingzhao
;
Zhu, Hongmei
;
Fu, Li
;
Li, Yun
;
Bao, Xubin
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
AG-221
IDH2
leukemia
R140Q
R172K
Discovery of DC_H31 as potential mutant IDH1 inhibitor through NADPH-based high throughput screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3229-3236
作者:
Duan, Zhe
;
Liu, Jingqiu
;
Niu, Liping
;
Wang, Jun
;
Feng, Mingqian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
IDH1 mutation
High-throughput screening
Pan-inhibitor
2-HG
Gliomas
Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433
作者:
Guo, Zuhao
;
Zhang, Zhuqing
;
Yang, Hong
;
Cao, Danyan
;
Xu, Xiaowei
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2020/07/01
Small-Molecule Targeting of Oncogenic FTO Demethylase in Acute Myeloid Leukemia
期刊论文
OAI收割
CANCER CELL, 2019, 卷号: 35, 期号: 4, 页码: 677-+
作者:
Huang, Yue
;
Su, Rui
;
Sheng, Yue
;
Dong, Lei
;
Dong, Ze
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/07/01
Highly functionalized cyclohexanone-monocyclic polyprenylated acylphloroglucinols from Hypericum perforatum induce leukemia cell apoptosis
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 6, 页码: 817-824
作者:
Guo, Yi
;
Tong, Qingyi
;
Zhang, Na
;
Duan, Xueyan
;
Cao, Yunfang
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2019/07/29
Quantitative profiling of cd13 on single acute myeloid leukemia cells by super-resolution imaging and its implication in targeted drug susceptibility assessment
期刊论文
iSwitch采集
Nanoscale, 2019, 卷号: 11, 期号: 4, 页码: 1737-1744
作者:
Xi, Yan
;
Wang, Dianbing
;
Wang, Tingting
;
Huang, Lin
;
Zhang, Xian-En
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2019/05/08
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:
Liang, Xiaofei
;
Wang, Beilei
;
Chen, Cheng
;
Wang, Aoli
;
Hu, Chen
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2020/05/21
TAF1 plays a critical role in AML1-ETO driven leukemogenesis
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2019, 卷号: 10, 期号: -, 页码: 4925
作者:
Xu, Ye
;
Man, Na
;
Karl, Daniel
;
Martinez, Concepcion
;
Liu, Fan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/12/09
Osteoglycin
Angiogenesis
Extracellular matrix
VEGF
VEGFR2
KDM3B suppresses APL progression by restricting chromatin accessibility and facilitating the ATRA-mediated degradation of PML/RAR alpha
期刊论文
OAI收割
CANCER CELL INTERNATIONAL, 2019, 卷号: 19, 期号: 1, 页码: 256
作者:
Wang, Xinrui
;
Fan, Huiyong
;
Xu, Congling
;
Jiang, Guojuan
;
Zhang, Ji
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/12/09
KDM3B
APL
PML
RAR alpha
me2
Chromatin accessibility
Differentiation