中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2019 [10]
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Design of wogonin-inspired selective cyclin-dependent kinase 9 (CDK9) inhibitors with potent in vitro and in vivo antitumor activity 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 782-801
作者:  
Wang, Jubo;  Li, Tinghan;  Zhao, Tengteng;  Wu, Tizhi;  Liu, Chuang
  |  收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
Pharmacological characterization of TQ05310, a potent inhibitor of isocitrate dehydrogenase 2 R140Q and R172K mutants 期刊论文  OAI收割
CANCER SCIENCE, 2019, 页码: 9
作者:  
Gao, Mingzhao;  Zhu, Hongmei;  Fu, Li;  Li, Yun;  Bao, Xubin
  |  收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
AG-221  IDH2  leukemia  R140Q  R172K  
Discovery of DC_H31 as potential mutant IDH1 inhibitor through NADPH-based high throughput screening 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 15, 页码: 3229-3236
作者:  
Duan, Zhe;  Liu, Jingqiu;  Niu, Liping;  Wang, Jun;  Feng, Mingqian
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Design and Synthesis of Potent, Selective Inhibitors of Protein Arginine Methyltransferase 4 against Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 11, 页码: 5414-5433
作者:  
Guo, Zuhao;  Zhang, Zhuqing;  Yang, Hong;  Cao, Danyan;  Xu, Xiaowei
  |  收藏  |  浏览/下载:61/0  |  提交时间:2020/07/01
Small-Molecule Targeting of Oncogenic FTO Demethylase in Acute Myeloid Leukemia 期刊论文  OAI收割
CANCER CELL, 2019, 卷号: 35, 期号: 4, 页码: 677-+
作者:  
Huang, Yue;  Su, Rui;  Sheng, Yue;  Dong, Lei;  Dong, Ze
  |  收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Highly functionalized cyclohexanone-monocyclic polyprenylated acylphloroglucinols from Hypericum perforatum induce leukemia cell apoptosis 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 6, 页码: 817-824
作者:  
Guo, Yi;  Tong, Qingyi;  Zhang, Na;  Duan, Xueyan;  Cao, Yunfang
  |  收藏  |  浏览/下载:62/0  |  提交时间:2019/07/29
Quantitative profiling of cd13 on single acute myeloid leukemia cells by super-resolution imaging and its implication in targeted drug susceptibility assessment 期刊论文  iSwitch采集
Nanoscale, 2019, 卷号: 11, 期号: 4, 页码: 1737-1744
作者:  
Xi, Yan;  Wang, Dianbing;  Wang, Tingting;  Huang, Lin;  Zhang, Xian-En
收藏  |  浏览/下载:62/0  |  提交时间:2019/05/08
Discovery of N-(4-(6-Acetamidopyrimidin-4-yloxy)phenyl)-2-(2-(trifluoromethyl)phenyl)acetamide (CHMFL-FLT3-335) as a Potent FMS-like Tyrosine Kinase 3 Internal Tandem Duplication (FLT3-ITD) Mutant Selective Inhibitor for Acute Myeloid Leukemia 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 2, 页码: 875-892
作者:  
Liang, Xiaofei;  Wang, Beilei;  Chen, Cheng;  Wang, Aoli;  Hu, Chen
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/05/21
TAF1 plays a critical role in AML1-ETO driven leukemogenesis 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2019, 卷号: 10, 期号: -, 页码: 4925
作者:  
Xu, Ye;  Man, Na;  Karl, Daniel;  Martinez, Concepcion;  Liu, Fan
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/12/09
KDM3B suppresses APL progression by restricting chromatin accessibility and facilitating the ATRA-mediated degradation of PML/RAR alpha 期刊论文  OAI收割
CANCER CELL INTERNATIONAL, 2019, 卷号: 19, 期号: 1, 页码: 256
作者:  
Wang, Xinrui;  Fan, Huiyong;  Xu, Congling;  Jiang, Guojuan;  Zhang, Ji
  |  收藏  |  浏览/下载:39/0  |  提交时间:2020/12/09