中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2021 [155]
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An overview of kinase downregulators and recent advances in discovery approaches 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6
作者:  
  |  收藏  |  浏览/下载:63/0  |  提交时间:2022/01/25
Macrocephatriolides A and B: Two Guaianolide Trimers from Ainsliaea macrocephala as PTP1B Inhibitors and Insulin Sensitizers 期刊论文  OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 24, 页码: 17782-17789
作者:  
Ren, Yong-Mei;  Zhang, Rui;  Feng, Zheling;  Ke, Chang-Qiang;  Yao, Sheng
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 6
作者:  
Yang, Xiangbo;  Lu, Huimin;  Xie, Hang;  Zhang, Binbin;  Nie, Tianqing
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/01/18
LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo 期刊论文  OAI收割
CANCER SCIENCE, 2021, 页码: 12
作者:  
Liu, Yingqiang;  Lai, Mengzhen;  Li, Shan;  Wang, Yanan;  Feng, Fang
  |  收藏  |  浏览/下载:87/0  |  提交时间:2022/01/18
Nanopore detects.-radiation inhibited HIV-1 protease activity 期刊论文  OAI收割
BIOSENSORS & BIOELECTRONICS, 2021, 卷号: 194, 页码: 5
作者:  
Li, Minghan;  Li, Wei;  Xiao, Yicen;  Liu, Qianshan;  Liang, Liyuan
  |  收藏  |  浏览/下载:66/0  |  提交时间:2021/11/26
Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 52, 页码: 12
作者:  
Ding, Hong;  Pei, Yuan;  Li, Yuanqing;  Xu, Wen;  Mei, Lianghe
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/06/15
A nomogram model based on peripheral blood lymphocyte subsets to assess the prognosis of non-small cell lung cancer patients treated with immune checkpoint inhibitors 期刊论文  OAI收割
TRANSLATIONAL LUNG CANCER RESEARCH, 2021
作者:  
Xu, Xiaoling;  Wang, Ding;  Chen, Wei;  Li, Na;  Suwinski, Rafal
  |  收藏  |  浏览/下载:75/0  |  提交时间:2022/02/14
FK228 potentiates topotecan activity against small cell lung cancer cells via induction of SLFN11 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021
作者:  
Yin, Yan-ping;  Ma, Li-ying;  Cao, Guo-zhen;  Hua, Jing-han
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/01/10
Transcriptomic Response to Perkinsus marinus in Two Crassostrea Oysters Reveals Evolutionary Dynamics of Host-Parasite Interactions 期刊论文  OAI收割
FRONTIERS IN GENETICS, 2021, 卷号: 12, 页码: 16
作者:  
Chan, Jiulin;  Wang, Lu;  Li, Li;  Mu, Kang;  Bushek, David
  |  收藏  |  浏览/下载:51/0  |  提交时间:2022/04/12
Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1 期刊论文  OAI收割
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:  
Zhang, Chun;  Sun, Yi-Tao;  Gao, Li-Xin;  Feng, Bo;  Yan, Xue
  |  收藏  |  浏览/下载:47/0  |  提交时间:2022/01/18