中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
采集方式
OAI收割 [20]
内容类型
期刊论文 [20]
发表日期
2016 [20]
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发表日期:2016
专题:上海药物研究所
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Identification and biochemical characterization of DC07090 as a novel potent small molecule inhibitor against human enterovirus 71 3C protease by structure-based virtual screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 124, 页码: 981-991
作者:
Ma, Guang-Hui
;
Ye, Yan
;
Zhang, Dan
;
Xu, Xin
;
Si, Pei
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
HFMD
EV71 3C(Pro)
Non-peptidyl inhibitor
Virtual screening
Pterostilbene Inhibits Human Multiple Myeloma Cells via ERK1/2 and JNK Pathway In Vitro and In Vivo
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2016, 卷号: 17, 期号: 11
作者:
Xie, Bingqian
;
Xu, Zhijian
;
Hu, Liangning
;
Chen, Gege
;
Wei, Rong
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
multiple myeloma
pterostilbene
apoptosis
cell cycle
ERK1/2
JNK
Facile Synthesis of 7-epi-Taxane and Its Derivatives and Preliminary Evaluation of Anticancer Activity
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2016, 卷号: 34, 期号: 11, 页码: 1165-1176
作者:
Li, Zhao
;
Feng, Jia
;
Zou, Kun
;
Yang, Zhuo
;
Zhang, Yong
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
taxane
7-epi-taxane
silver oxide
amino acid
C-13 derivative of taxane
anticancer activity
Small-Molecule Targeting of E3 Ligase Adaptor SPOP in Kidney Cancer
期刊论文
OAI收割
CANCER CELL, 2016, 卷号: 30, 期号: 3, 页码: 474-484
作者:
Guo, Zhong-Qiang
;
Zheng, Tong
;
Chen, Baoen
;
Luo, Cheng
;
Ouyang, Sisheng
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
Absorption mechanism of neobavaisoflavone in Caco-2 cell monolayer mode
期刊论文
OAI收割
Zhongguo Zhong yao za zhi = Zhongguo zhongyao zazhi = China journal of Chinese materia medica, 2016, 卷号: 41, 期号: 15, 页码: 2922-2926
作者:
Xu, Xiao-Kun
;
Chen, Zhi-Yong
;
Li, Zhuo-Qing
;
Zhang, Yi-Min
;
Liao, Li-Ping
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Structural mechanism of ligand activation in human calcium-sensing receptor
期刊论文
OAI收割
ELIFE, 2016, 卷号: 5
作者:
Geng, Yong
;
Mosyak, Lidia
;
Kurinov, Igor
;
Zuo, Hao
;
Sturchler, Emmanuel
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2019/01/08
Effects of alisol B 23-acetate on ovarian cancer cells: G1 phase cell cycle arrest, apoptosis, migration and invasion inhibition
期刊论文
OAI收割
PHYTOMEDICINE, 2016, 卷号: 23, 期号: 8, 页码: 800-809
作者:
Zhang, Le-Le
;
Xu, Yu-Lian
;
Tang, Zheng-Hai
;
Xu, Xiao-Huang
;
Chen, Xin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Ovarian cancer
Alisol B 23-acetate
Cell cycle arrest
Apoptosis
Migration
Invasion
Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b] [1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 239-251
作者:
Zhan, Zhengsheng
;
Peng, Xia
;
Liu, Qiufeng
;
Chen, Fang
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:48/0
  |  
提交时间:2019/01/08
Antitumor
c-Met
Kinase inhibitor
Triazolotriazines
Discovery of Benzocycloalkane Derivatives Efficiently Blocking Bacterial Virulence for the Treatment of Methicillin-Resistant S. aureus (MRSA) Infections by Targeting Diapophytoene Desaturase (CrtN)
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 10, 页码: 4831-4848
作者:
Wang, Youxin
;
Di, Hongxia
;
Chen, Feifei
;
Xu, Yong
;
Xiao, Qiang
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2019/01/08
Design and synthesis of novel triazole derivatives containing gamma-lactam as potential antifungal agents
期刊论文
OAI收割
CHINESE CHEMICAL LETTERS, 2016, 卷号: 27, 期号: 5, 页码: 703-706
作者:
Xu, Yuan-Yuan
;
Qian, An-Ran
;
Cao, Xu-Feng
;
Ling, Chen-Yu
;
Cao, Yong-Bing
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Synthesis
Triazole
gamma-Lactam
Antifungal activity