中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
采集方式
OAI收割 [20]
内容类型
期刊论文 [20]
发表日期
2023 [2]
2022 [3]
2021 [1]
2020 [4]
2019 [2]
2016 [1]
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专题:上海药物研究所
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Intranasal delivery of replicating mRNA encoding hACE2-targeting antibody against SARS-CoV-2 Omicron infection in the hamster
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2023, 卷号: 209, 页码: 9
作者:
Zhang, Ya-Nan
;
Zhang, Hong-Qing
;
Wang, Gui-Feng
;
Zhang, Zhe-Rui
;
Li, Jia-Qi
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Omicron
VEEV VRP
Replicable mRNA
Therapeutic drug monitoring of caffeine and its primary metabolites in plasma using LC-ESI-MS/MS for apnea of prematurity treatment: Evaluation of ultrapure water as a surrogate matrix
期刊论文
OAI收割
BIOMEDICAL CHROMATOGRAPHY, 2022, 卷号: 36, 期号: 11, 页码: e5462
作者:
Long, Jia-Yi
;
Hu, Ya-Hui
;
Xia, Ying
;
Du, Fei-Fei
;
Dai, Hao-Ran
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/21
apnea of prematurity
caffeine
LC-ESI-MS
MS
preterm infants
surrogate matrix
therapeutic drug monitoring
Identification and evaluation of a lipid-lowering small compound in preclinical models and in a Phase I trial
期刊论文
OAI收割
CELL METABOLISM, 2022, 卷号: 34, 期号: 5, 页码: 667-+
作者:
Wang, Jiang
;
Zhao, Jing
;
Yan, Cong
;
Xi, Cong
;
Wu, Chenglin
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2022/08/16
Computational and Structure-Based Development of High Potent Cell-Active Covalent Inhibitor Targeting the Peptidyl-Prolyl Isomerase NIMA-Interacting-1 (Pin1)
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 3, 页码: 2174-2190
作者:
Liu, Liping
;
Zhu, Rui
;
Li, Jiacheng
;
Pei, Yuan
;
Wang, Shuangshuang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/08/16
Design, synthesis, and biological evaluation of tetrahydroisoquinolines derivatives as novel, selective PDE4 inhibitors for antipsoriasis treatment
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 211, 页码: 20
作者:
Zhang, Rui
;
Li, Heng
;
Zhang, Xianglei
;
Li, Jian
;
Su, Haixia
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/24
PDE4 inhibitors
Tetrahydroisoquinoline
Antipsoriasis
Therapy for Apnoea of Prematurity: A Retrospective Study on Effects of Standard Dose and Genetic Variability on Clinical Response to Caffeine Citrate in Chinese Preterm Infants
期刊论文
OAI收割
ADVANCES IN THERAPY, 2020, 页码: 20
作者:
He, Xin
;
Qiu, Jin-Chun
;
Lu, Ke-Yu
;
Guo, Hong-Li
;
Li, Ling
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/12/24
Adenosine receptors
AHR
AOP
Caffeine
Phosphodiesterase
Polymorphism
Therapeutic drug monitoring
Anti-hepatitis B virus activity of swertisin isolated from Iris tectorum Maxim
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2020, 卷号: 257, 页码: 9
作者:
Xu, Hong-Yan
;
Ren, Ji-Hua
;
Su, Yu
;
Ren, Fang
;
Zhou, Yu-Jiao
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
Iris tectorum Maxim
Swertisin
Hepatitis B virus
HBsAg
HBeAg
DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:
Li, Heng
;
Li, Jian
;
Zhang, Xianglei
;
Feng, Chunlan
;
Fan, Chen
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2020/12/24
DC591017
PDE4
Inflammation
Macrophages
Dendritic cells
Psoriasis
DC591017, a phosphodiesterase-4 (PDE4) inhibitor with robust anti-inflammation through regulating PKA-CREB signaling
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 15
作者:
Li, Heng
;
Li, Jian
;
Zhang, Xianglei
;
Feng, Chunlan
;
Fan, Chen
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
DC591017
PDE4
Inflammation
Macrophages
Dendritic cells
Psoriasis