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Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [106]
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Pharmacological inhibition of Kir4.1 evokes rapid-onset antidepressant responses 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2024, 页码: 29
作者:  
Zhou, Xiaoyu;  Zhao, Cheng;  Xu, Haiyan;  Xu, Yixiang;  Zhan, Li
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Conserved class B GPCR activation by a biased intracellular agonist 期刊论文  OAI收割
NATURE, 2023, 页码: 25
作者:  
Zhao, Li-Hua;  He, Qian;  Yuan, Qingning;  Gu, Yimin;  He, Xinheng
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/10/17
Antiandrogen treatment induces stromal cell reprogramming to promote castration resistance in cancer 期刊论文  OAI收割
CANCER CELL, 2023, 卷号: 41, 期号: 7, 页码: 1345-+
作者:  
Wang, Hanling;  Li, Ni;  Liu, Qiuli;  Guo, Jiacheng
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
Design, Synthesis and Bioactivity of [3.3.3]Propellane-Based Voltage-Gated Calcium Channel alpha 2 delta Subunit Ligands 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 6, 页码: 2226-2238
作者:  
He Jinyan;  Tian Fuyun;  Wu Qingqing;  Zheng Yueming;  Chen Yuting
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/10/17
Selective PPAR gamma modulator diosmin improves insulin sensitivity and promotes browning of white fat 期刊论文  OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2023, 卷号: 299, 期号: 4, 页码: 14
作者:  
Yu, Jian;  Hu, Yepeng;  Sheng, Maozheng;  Gao, Mingyuan;  Guo, Wenxiu
  |  收藏  |  浏览/下载:23/0  |  提交时间:2023/10/17
Discovery of a Potent, Cooperative, and Selective SOS1 PROTAC ZZ151 with In Vivo Antitumor Efficacy in KRAS-Mutant Cancers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 6, 页码: 4197-4214
作者:  
Zhou, Zehui;  Zhou, Guizhen;  Zhou, Chuan;  Fan, Zisheng;  Cui, Rongrong
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
Design, Synthesis, and Bioevaluation of Pyrido[2,3-d]pyrimidin-7-ones as Potent SOS1 Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 页码: 183-190
作者:  
Liu, Meiying;  Zhou, Guizhen;  Su, Wenhong;  Gu, Yuejiao;  Gao, Mingshan
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/03/27
Mannosylated engineered trichosanthin-legumain protein vaccine hydrogel for breast cancer immunotherapy 期刊论文  OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2022, 卷号: 223, 页码: 1485-1494
作者:  
Chen, Guihua;  Xiong, Wei;  Gu, Zeyun;  Gao, Yanrong;  Hou, Jiazhen
  |  收藏  |  浏览/下载:10/0  |  提交时间:2023/10/17
Diversity-oriented synthesis of marine polybrominated diphenyl ethers as potential KCNQ potassium channel activators 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 126, 页码: 105909
作者:  
Liu, Lai-Xin;  Gu, Ru-Rong;  Jin, Yang;  Chen, Xue-Qin;  Li, Xu-Wen
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/03/21