中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [25]
采集方式
OAI收割 [25]
内容类型
期刊论文 [25]
发表日期
2023 [2]
2022 [5]
2021 [3]
2020 [3]
2019 [1]
2017 [1]
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学科主题
Chemistry [1]
Pharmacolo... [1]
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专题:上海药物研究所
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Autoimmune diseases: targets, biology, and drug discovery
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 12
作者:
Li, Shu-jie
;
Wu, Yan-li
;
Chen, Juan-hua
;
Shen, Shi-yi
;
Duan, Jia
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/26
autoimmune disease
autoantigen
immunotherapy
type 1 diabetes
insulin
drug discovery
Conserved class B GPCR activation by a biased intracellular agonist
期刊论文
OAI收割
NATURE, 2023, 页码: 25
作者:
Zhao, Li-Hua
;
He, Qian
;
Yuan, Qingning
;
Gu, Yimin
;
He, Xinheng
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
Molecular recognition of two endogenous hormones by the human parathyroid hormone receptor-1
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 11
作者:
Zhao, Li-hua
;
Yuan, Qing-ning
;
Dai, An-tao
;
He, Xin-heng
;
Chen, Chuan-wei
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/04/10
G protein- coupled receptors
parathyroid hormone
PTH-related peptide
PTH receptor-1
cryo-electron microscopy structure
osteoporosis
Structure insights into selective coupling of G protein subtypes by a class B G protein-coupled receptor
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 13
作者:
Zhao, Li-Hua
;
Lin, Jingyu
;
Ji, Su-Yu
;
Zhou, X. Edward
;
Mao, Chunyou
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/04/10
AlphaFold2 versus experimental structures: evaluation on G protein-coupled receptors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 7
作者:
He, Xin-heng
;
You, Chong-zhao
;
Jiang, Hua-liang
;
Jiang, Yi
;
Xu, H. Eric
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/08/16
G protein-coupled receptors
AlphaFold2
protein structure prediction
drug design
structural biology
Molecular insights into ligand recognition and activation of chemokine receptors CCR2 and CCR3
期刊论文
OAI收割
CELL DISCOVERY, 2022, 卷号: 8, 期号: 1, 页码: 11
作者:
Shao, Zhehua
;
Tan, Yangxia
;
Shen, Qingya
;
Hou, Li
;
Yao, Bingpeng
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/08/16
A distinctive ligand recognition mechanism by the human vasoactive intestinal polypeptide receptor 2
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 10
作者:
Xu, Yingna
;
Feng, Wenbo
;
Zhou, Qingtong
;
Liang, Anyi
;
Li, Jie
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2022/06/15
Identification and mechanism of G protein-biased ligands for chemokine receptor CCR1
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 页码: 24
作者:
Shao, Zhehua
;
Shen, Qingya
;
Yao, Bingpeng
;
Mao, Chunyou
;
Chen, Li-Nan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/06/15
Constitutive signal bias mediated by the human GHRHR splice variant 1
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:
Cong, Zhaotong
;
Zhou, Fulai
;
Zhang, Chao
;
Zou, Xinyu
;
Zhang, Huibing
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/12/01
class B1 GPCR
receptor bias
cancer
cell proliferation
A multi-targeting drug design strategy for identifying potent anti-SARS-CoV-2 inhibitors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Ren, Peng-xuan
;
Shang, Wei-juan
;
Yin, Wan-chao
;
Ge, Huan
;
Wang, Lin
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2021/06/11
SARS-CoV-2 inhibitors
RdRp
host ribosome
Virus RNA