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Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [40]
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Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11
作者:  
Zhao, Yitian;  Zhang, Min;  Hou, Xudong;  Han, Jiaxin;  Qin, Xiaoya
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/10/17
Chloroquine enhances the efficacy of chemotherapy drugs against acute myeloid leukemia by inactivating the autophagy pathway 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 11
作者:  
Wang, Han-lin;  Li, Jia-nan;  Kan, Wei-juan;  Xu, Gao-ya;  Luo, Guang-hao
  |  收藏  |  浏览/下载:18/0  |  提交时间:2023/10/17
High-throughput screening of SARS-CoV-2 main and papain-like protease inhibitors 期刊论文  OAI收割
PROTEIN & CELL, 2023, 卷号: 14, 期号: 1, 页码: 17-27
作者:  
Zang, Yi;  Su, Mingbo;  Wang, Qingxing;  Cheng, Xi;  Zhang, Wenru
  |  收藏  |  浏览/下载:2/0  |  提交时间:2024/03/27
(-)-Epigallocatechin Gallate is a Noncompetitive Inhibitor of NAD Kinase 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:  
Liu, Tonghai;  Shi, Wenjia;  Ding, Yiluan;  Wu, Qiqi;  Zhang, Bei
  |  收藏  |  浏览/下载:24/0  |  提交时间:2022/12/13
Spiroarborin, an ent-Clerodane Homodimer from Callicarpa arborea as an Inhibitor of the Eleven-Nineteen Leukemia (ENL) Protein by the YEATS Domain 期刊论文  OAI收割
JOURNAL OF NATURAL PRODUCTS, 2022, 卷号: 85, 期号: 2, 页码: 317-326
作者:  
Pu, De-Bing;  Guo, Si-Qi;  Ni, Dong-Xuan;  Lin, Jing;  Gao, Jun-Bo
  |  收藏  |  浏览/下载:22/0  |  提交时间:2022/06/15
Discovery of highly potent SARS-CoV-2 M-pro inhibitors based on benzoisothiazolone scaffold 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 58, 页码: 6
作者:  
Chen, Weixiong;  Feng, Bo;  Han, Sheng;  Wang, Peipei;  Chen, Wuhong
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/06/15
Dual-Channel Fluorescent Probe for the Simultaneous Monitoring of Peroxynitrite and Adenosine-5 '-triphosphate in Cellular Applications 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2021, 页码: 10
作者:  
Wu, Luling;  Liu, Jihong;  Tian, Xue;  Groleau, Robin R.;  Feng, Beidou
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/06/15
Discovery of High-Affinity Inhibitors of the BPTF Bromodomain 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12075-12088
作者:  
Lu, Tian;  Lu, Haibo;  Duan, Zhe;  Wang, Jun;  Han, Jie
  |  收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
Competitive CatSper Activators of Progesterone from Rhynchosia volubilis 期刊论文  OAI收割
PLANTA MEDICA, 2021, 页码: 10
作者:  
Xiang, Jin;  Kang, Hang;  Li, Hong-Gang;  Shi, Yu-Long;  Zhang, Ya-Li
  |  收藏  |  浏览/下载:47/0  |  提交时间:2021/11/04
Pharmacodynamic, pharmacokinetic, and phase 1a study of bisthianostat, a novel histone deacetylase inhibitor, for the treatment of relapsed or refractory multiple myeloma 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  
Zhou, Yu-bo;  Zhang, Yang-ming;  Huang, Hong-hui;  Shen, Li-jing;  Han, Xiao-feng
  |  收藏  |  浏览/下载:67/0  |  提交时间:2021/11/04