中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [84]
采集方式
OAI收割 [84]
内容类型
期刊论文 [84]
发表日期
2024 [1]
2023 [6]
2022 [9]
2021 [11]
2020 [8]
2019 [6]
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浏览/检索结果:
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专题:上海药物研究所
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Proteogenomic characterization of small cell lung cancer identifies biological insights and subtype-specific therapeutic strategies
期刊论文
OAI收割
CELL, 2024, 卷号: 187, 期号: 1, 页码: 49
作者:
Liu, Qian
;
Zhang, Jing
;
Guo, Chenchen
;
Wang, Mengcheng
;
Wang, Chenfei
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/02/27
The enzyme activity of sortase A is regulated by phosphorylation in Staphylococcus aureus
期刊论文
OAI收割
VIRULENCE, 2023, 卷号: 14, 期号: 1, 页码: 2171641
作者:
Chen, Feifei
;
Di, Hongxia
;
Wang, Yanhui
;
Peng, Chao
;
Chen, Rongrong
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
Staphylococcus aureus
Sortase A
protein phosphorylation
virulence
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:
Fang, Feifei
;
Dai, Yang
;
Wang, Hao
;
Ji, Yinchun
;
Liang, Xuewu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
derivatives
Antitumor drug development
Potential AXL inhibitor
Antitumor activity
Structure-based drug design
Fused-pyrazolone carboxamide
DCZ5248, a novel dual inhibitor of Hsp90 and autophagy, exerts antitumor activity against colon cancer (vol 42, pg 132, 2021)
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 1
作者:
Chen, Xiang-ling
;
Liu, Peng
;
Zhu, Wei-liang
;
Lou, Li-guang
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/01/16
Effect of an Herbal-Based Injection on 28-Day Mortality in Patients With Sepsis The EXIT-SEP Randomized Clinical Trial
期刊论文
OAI收割
JAMA INTERNAL MEDICINE, 2023, 卷号: 183, 期号: 7, 页码: 647-655
作者:
Liu, Songqiao
;
Yao, Chen
;
Xie, Jianfeng
;
Liu, Hong
;
Wang, Hongliang
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/27
Squamabietenols A-F, undescribed abietane-O-abietane dimeric diterpenoids from the ornamental conifer Juniperus squamata and their ATP-citrate lyase inhibitory activities
期刊论文
OAI收割
PHYTOCHEMISTRY, 2023, 卷号: 210, 页码: 14
作者:
Liang, Kai -Yuan
;
Li, Hao
;
Zhou, Peng-Jun
;
Zhao, Ze-Yu
;
Zang, Yi
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
Juniperus squamata Buch
-ham ex D
don
Cupressaceae
Conifer
Phytochemistry
Chemotaxonomy
Abietane
O -Abietane
Dimeric
mono-diterpenoids
Squamabietenols a -f
ATP -Citrate lyase
Molecular docking
AXL antibody and AXL-ADC mediate antitumor efficacy via targeting AXL in tumor-intrinsic epithelial-mesenchymal transition and tumor-associated M2-like macrophage
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 14
作者:
Pei, Jin-peng
;
Wang, Yue
;
Ma, Lan-ping
;
Wang, Xin
;
Liu, Liang
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/04/10
AXL
NSCLC
TNBC
M2-macrophage
antibody-drug conjugate
Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:
Xie, Xiong
;
Zheng, Yu-Gui
;
Chen, Huan
;
Li, Jian
;
Luo, Rong-Hua
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
Identification of a class of potent USP25/28 inhibitors with broad-spectrum anti-cancer activity
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 3
作者:
Peng, Jin
;
Jiang, Kun
;
Sun, Xiao
;
Wu, Lingzhi
;
Wang, Jiewei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Synthesis and pharmacological validation of fluorescent diarylsulfonylurea analogues as NLRP3 inhibitors and imaging probes
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 237, 页码: 13
作者:
Zhao, Jiannan
;
Li, Yongling
;
Ma, Jing
;
Liu, Jingting
;
Xiao, Ruoxuan
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/08/16
NLRP3
Inflammasome
Inhibitor
Fluorescence imaging
Sulfonylurea