中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [20]
采集方式
OAI收割 [20]
内容类型
期刊论文 [20]
发表日期
2023 [6]
2022 [2]
2021 [2]
2020 [3]
2018 [2]
2017 [1]
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专题:上海药物研究所
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Discovery of 2-Aminopyrimidine Derivatives as Potent Dual FLT3/CHK1 Inhibitors with Significantly Reduced hERG Inhibitory Activities
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 23
作者:
Li, Xuemei
;
Wang, Peipei
;
Wang, Chang
;
Jin, Tingting
;
Xu, Ran
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
Chloroquine enhances the efficacy of chemotherapy drugs against acute myeloid leukemia by inactivating the autophagy pathway
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 11
作者:
Wang, Han-lin
;
Li, Jia-nan
;
Kan, Wei-juan
;
Xu, Gao-ya
;
Luo, Guang-hao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/10/17
acute myeloid leukemia
cytarabine
daunorubicin
idarubicin
drug resistant
multi-omics
autophagy
chloroquine phosphate
Recent advances of activation techniques-based discovery of new compounds from marine fungi
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 167, 页码: 14
作者:
Zou, Ran
;
Chen, Bao
;
Sun, Jie
;
Guo, Yue-Wei
;
Xu, Baofu
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
Marine fungi
Silent
Biosynthetic gene clusters
Activation techniques
Scalarane sesterterpenes from the South China Sea sponge Hyrtios erecta and their PTP1B inhibitory activity
期刊论文
OAI收割
TETRAHEDRON, 2023, 卷号: 137, 页码: 5
作者:
Sun, Li-Li
;
Shen, Yi-Ran
;
Li, Jia
;
Wang, Jian-Rong
;
Li, Xu-Wen
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/10/17
Sponge
Hyrtios erecta
Scalarane-type sesterterpene
Configuration
PTP1B
Bioactive compounds from Huashi Baidu decoction possess both antiviral and anti-inflammatory effects against COVID-19
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 18, 页码: 11
作者:
Xu, Haiyu
;
Li, Shufen
;
Liu, Jiayuan
;
Cheng, Jinlong
;
Kang, Liping
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/10/17
COVID-19
traditional Chinese medicine
TCMT-NDRD
antivirus
anti-inflammation
Targeting C/EBP alpha overcomes primary resistance and improves the efficacy of FLT3 inhibitors in acute myeloid leukaemia
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 18
作者:
Wang, Hanlin
;
Luo, Guanghao
;
Hu, Xiaobei
;
Xu, Gaoya
;
Wang, Tao
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Therapeutic drug monitoring of caffeine and its primary metabolites in plasma using LC-ESI-MS/MS for apnea of prematurity treatment: Evaluation of ultrapure water as a surrogate matrix
期刊论文
OAI收割
BIOMEDICAL CHROMATOGRAPHY, 2022, 卷号: 36, 期号: 11, 页码: e5462
作者:
Long, Jia-Yi
;
Hu, Ya-Hui
;
Xia, Ying
;
Du, Fei-Fei
;
Dai, Hao-Ran
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/21
apnea of prematurity
caffeine
LC-ESI-MS
MS
preterm infants
surrogate matrix
therapeutic drug monitoring
p Proteogenomic characterization identifies clinically relevant subgroups of intrahepatic cholangiocarcinoma
期刊论文
OAI收割
CANCER CELL, 2022, 卷号: 40, 期号: 1, 页码: 70-+
作者:
Dong, Liangqing
;
Lu, Dayun
;
Chen, Ran
;
Lin, Youpei
;
Zhu, Hongwen
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/06/15
Rescue of maternal immune activation-induced behavioral abnormalities in adult mouse offspring by pathogen-activated maternal T-reg cells
期刊论文
OAI收割
NATURE NEUROSCIENCE, 2021, 页码: 33
作者:
Xu, Zhipeng
;
Zhang, Xiaoyun
;
Chang, Hao
;
Kong, Yue
;
Ni, Yangyue
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2021/05/24
SL010110, a lead compound, inhibits gluconeogenesis via SIRT2-p300-mediated PEPCK1 degradation and improves glucose homeostasis in diabetic mice
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Ren, Yu-ran
;
Ye, Yang-liang
;
Feng, Ying
;
Xu, Ti-fei
;
Shen, Yu
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/05/24
SL010110
gluconeogenesis
primary mouse hepatocytes
PEPCK1
acetylation
degradation