中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [672]
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Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-d]pyrimidin-7(6H)-one" Scaffold for the Treatment of B Cell Lymphoma 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2884-2906
作者:  
Liang, Xuewu;  Yu, Haolan;  Liang, Renwen;  Feng, Zhuanghui;  Saidahmatov, Abdusaid
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/04/09
Molecular features of the ligand-free GLP-1R, GCGR and GIPR in complex with Gs proteins 期刊论文  OAI收割
CELL DISCOVERY, 2024, 卷号: 10, 期号: 1, 页码: 13
作者:  
Cong, Zhaotong;  Zhao, Fenghui;  Li, Yang;  Luo, Gan;  Mai, Yiting
  |  收藏  |  浏览/下载:22/0  |  提交时间:2024/03/13
Development and Validation of an ADA-Tolerant Assay for Quantification of an Exatecan-Based ADC in Monkey Plasma 期刊论文  OAI收割
MOLECULES, 2024, 卷号: 29, 期号: 3, 页码: 14
作者:  
Tao, Yimin;  Lu, Wei;  Gao, Jinli;  Yang, Shuangshuang;  Ruan, Chaoyi
  |  收藏  |  浏览/下载:15/0  |  提交时间:2024/03/13
Bioorthogonal chemistry mediated cell engineering for advanced cell and cell-derived vesicle therapies: Principles, progresses, and remaining challenges 期刊论文  OAI收割
CHEMICAL ENGINEERING JOURNAL, 2024, 卷号: 480, 页码: 19
作者:  
Pan, Chao;  Jiang, Xiuxian;  Liu, Chang;  Wei, Junchao;  Wang, Yang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/02/27
Revisiting the Role of Valeric Acid in Manipulating Ulcerative Colitis 期刊论文  OAI收割
INFLAMMATORY BOWEL DISEASES, 2024, 页码: 12
作者:  
Liu, Moting;  Zhang, Yao;  Liu, Jia;  Xiang, Caigui;  Lu, Qiukai
  |  收藏  |  浏览/下载:7/0  |  提交时间:2024/02/19
The promise and challenges of combination therapies with antibody-drug conjugates in solid tumors 期刊论文  OAI收割
JOURNAL OF HEMATOLOGY & ONCOLOGY, 2024, 卷号: 17, 期号: 1, 页码: 32
作者:  
Wei, Qing;  Li, Peijing;  Yang, Teng;  Zhu, Jiayu;  Sun, Lu
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/02/27
Structure-Guided Design, Synthesis, and Antivirulence Assessment of Covalent Staphylococcus aureus Sortase A Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1127-1146
作者:  
Yue, Chuan;  Yuan, Ziqi;  Xu, Guobin;  Guan, Xiang-Na;  Wei, Bingyan
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/02/27
Reversible SAHH inhibitor ameliorates MIA-induced osteoarthritis of rats through suppressing MEK/ERK pathway 期刊论文  OAI收割
BIOMEDICINE & PHARMACOTHERAPY, 2024, 卷号: 170, 页码: 6
作者:  
Fan, Shu-Hui;  Chang, Yuan;  Xiong, Xiao-Yu;  Xiang, Mai;  Yuan, Wen-Long
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/02/27
Epigenetic-based combination therapy and liposomal codelivery overcomes osimertinib-resistant NSCLC via repolarizing tumor-associated macrophages 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 12
作者:  
Lin, Ting-ting;  Xiong, Wei;  Chen, Gui-hua;  He, Yang;  Long, Li
  |  收藏  |  浏览/下载:6/0  |  提交时间:2024/01/26
FMRP phosphorylation modulates neuronal translation through YTHDF1 期刊论文  OAI收割
MOLECULAR CELL, 2023, 卷号: 83, 期号: 23
作者:  
Zou, Zhongyu;  Wei, Jiangbo;  Chen, Yantao;  Kang, Yunhee;  Shi, Hailing
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/03/27