中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [47]
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Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:  
Wang, Pingyuan;  Zhu, Wen-Ting;  Wang, Yajing;  Song, Shan-Shan;  Xi, Yong
  |  收藏  |  浏览/下载:58/0  |  提交时间:2023/10/17
Thioparib inhibits homologous recombination repair, activates the type I IFN response, and overcomes olaparib resistance 期刊论文  OAI收割
EMBO MOLECULAR MEDICINE, 2023, 页码: 24
作者:  
Wang, Li-Min;  Wang, Pingyuan;  Chen, Xiao-Min
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/04/10
Targeting UHRF1-SAP30-MXD4 axis for leukemia initiating cell eradication in myeloid leukemia 期刊论文  OAI收割
CELL RESEARCH, 2022, 页码: 19
作者:  
Hu, Cheng-Long;  Chen, Bing-Yi;  Li, Zijuan;  Yang, Tianbiao;  Xu, Chun-Hui
  |  收藏  |  浏览/下载:31/0  |  提交时间:2022/12/13
Mass spectrometry imaging: new eyes on natural products for drug research and development 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 16
作者:  
Hou, Jin-jun;  Zhang, Zi-jia;  Wu, Wen-yong;  He, Qing-qing;  Zhang, Teng-qian
  |  收藏  |  浏览/下载:29/0  |  提交时间:2022/11/11
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:  
Kayumov, Muzaffar;  Jia, Li;  Pardaev, Azizbek;  Song, Shan-Shan;  Mirzaakhmedov, Sharafitdin
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/21
SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy 期刊论文  OAI收割
NEOPLASIA, 2022, 卷号: 32, 页码: 12
作者:  
Zhou, Li-Na;  Xiong, Chaodong;  Cheng, Yong-Jun;  Song, Shan-Shan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/04/10
Chemo- and Site-Selective Lysine Modification of Peptides and Proteins under Native Conditions Using the Water-Soluble Zolinium 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 14
作者:  
Sun, Haiguo;  Xi, Mengyu;  Jin, Qiang;  Zhu, Zhengdan;  Zhang, Yani
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/09/30
CoVac501, a self-adjuvanting peptide vaccine conjugated with TLR7 agonists, against SARS-CoV-2 induces protective immunity 期刊论文  OAI收割
CELL DISCOVERY, 2022, 卷号: 8, 期号: 1, 页码: 16
作者:  
Long, Yiru;  Sun, Jianhua;  Song, Tian-Zhang;  Liu, Tingting;  Tang, Feng
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/06/15
DCZ0014, a novel compound in the therapy of diffuse large B-cell lymphoma via the B cell receptor signaling pathway 期刊论文  OAI收割
NEOPLASIA, 2022, 卷号: 24, 期号: 1, 页码: 50-61
作者:  
Chang, Shuaikang;  Li, Bo;  Xie, Yongsheng;  Wang, Yingcong;  Xu, Zhijian
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target 期刊论文  OAI收割
CELL RESEARCH, 2021, 页码: 14
作者:  
Xia, Bingqing;  Shen, Xurui;  He, Yang;  Pan, Xiaoyan;  Liu, Feng-Liang
  |  收藏  |  浏览/下载:74/0  |  提交时间:2021/08/17