中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [70]
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期刊论文 [174]
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pH-responsive nanogels with enhanced antioxidant and antitumor activities on drug delivery and smart drug release
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2024, 卷号: 257, 页码: 16
作者:
Ma, Bing
;
Li, Qing
;
Mi, Yingqi
;
Zhang, Jingjing
;
Tan, Wenqiang
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
Benzimidazole-chitosan quaternary ammonium
salt
Nanogels
pH-responsive
Antioxidant activity
Antitumor activity
Structure-based drug discovery of novel fused- pyrazolone carboxamide derivatives as potent and selective AXL inhibitors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 12, 页码: 4918-4933
作者:
Fang, Feifei
;
Dai, Yang
;
Wang, Hao
;
Ji, Yinchun
;
Liang, Xuewu
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
derivatives
Antitumor drug development
Potential AXL inhibitor
Antitumor activity
Structure-based drug design
Fused-pyrazolone carboxamide
Preparation of imidazole acids grafted chitosan with enhanced antioxidant, antibacterial and antitumor activities
期刊论文
OAI收割
CARBOHYDRATE POLYMERS, 2023, 卷号: 315, 页码: 16
作者:
Ma, Bing
;
Zhang, Jingjing
;
Mi, Yingqi
;
Miao, Qin
;
Tan, Wenqiang
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/11/15
Imidazole acids grafted chitosan
Antioxidant activity
Antibacterial activity
Antitumor activity
Antitumor Cembrane Diterpenoids from the South China Sea Soft Coral Lobophytum sp.
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 卷号: 20, 期号: 4
作者:
Song, Yu-Ting
;
Yu, Dan-Dan
;
Zhi Su, Ming
;
Luo, Hui
;
Cao, Jian-Guo
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/03/27
soft coral
Lobophytum sp
cembranoids
configuration determination
antitumor activity
Synthesis and Biological Evaluation of Sclareolide-Indole Conjugates and Their Derivatives
期刊论文
OAI收割
MOLECULES, 2023, 卷号: 28, 期号: 4, 页码: 1737
作者:
Cheng, Ying
;
Lyu, Xilin
;
Liu, Chen
;
Wang, Xiancheng
;
Cheng, Jing
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/03/27
sclareolide
indole
polyphenol
acetal
antitumor activity
Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:
Li, Ennian
;
Wang, Kai
;
Zhang, Bei
;
Guo, Siqi
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/08/16
DNMT1 inhibitor
A549 cell lines
HCT116 cell lines
antitumor activity
pharmacokinetic
Preparation of Doxorubicin-Loaded Carboxymethyl-beta-Cyclodextrin/Chitosan Nanoparticles with Antioxidant, Antitumor Activities and pH-Sensitive Release
期刊论文
OAI收割
MARINE DRUGS, 2022, 卷号: 20, 期号: 5, 页码: 18
作者:
Mi, Yingqi
;
Zhang, Jingjing
;
Tan, Wenqiang
;
Miao, Qin
;
Li, Qing
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/07/26
chitosan nanoparticles
cyclodextrin
antioxidant activity
antitumor activity
drug release
Discovery of PHGDH inhibitors by virtual screening and preliminary structure-activity relationship study
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 121, 页码: 13
作者:
Zhang, Fu-Mao
;
Yuan, Liang
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/06/15
Virtual screening
PHGDH
Structure-activity relationships
Antitumor
Efficient Synthesis and Biological Evaluation of 6-Trifluoroethoxy Functionalized Pteridine Derivatives as EGFR Inhibitors
期刊论文
OAI收割
MEDICINAL CHEMISTRY, 2022, 卷号: 18, 期号: 3, 页码: 353-363
作者:
Lin, Jin
;
Zhang, Zemin
;
Lin, Xiongqiang
;
Chen, Zhendong
;
Luc, Tian
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
Pteridine
derivatives
EGFR
inhibitor
2,2,2-trifluoroethoxy
antitumor activity
TNKS inhibitors potentiate proliferative inhibition of BET inhibitors via reducing beta-Catenin in colorectal cancer cells
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2022, 卷号: 12, 期号: 3, 页码: 1069-+
作者:
Wu, Qian
;
Xuan, Yi-Fei
;
Su, Ai-Ling
;
Bao, Xu-Bin
;
Miao, Ze-Hong
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
BET inhibitor
Tankyrases inhibitor
beta-Catenin
antitumor activity
combination therapy