中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [11]
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Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Chen, Xuetao
;
Wu, Tingting
;
Du, Zhiyan
;
Kang, Wenjing
;
Xu, Rujun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/02/27
BET
BD1
Bromodomain
Brain-permeable
Multiple sclerosis
Evolution of pore structure and adsorption-desorption in oil shale formation rocks after compression
期刊论文
OAI收割
ENERGY, 2023, 卷号: 278, 页码: 127913
作者:
Huang XF(黄先富)
;
Zhao YP(赵亚溥)
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/09/05
Shale oil and shale gas
Adsorption -desorption ishotherms
BET specific surface area
Total pore volume
Fractal dimension
Carbon sequestration
Cyclization strategy leads to highly potent Bromodomain and extra-terminal (BET) Bromodomain inhibitors for the treatment of acute liver injury
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 13
作者:
Chen, Chao
;
Lu, Tian
;
Chen, Panyu
;
Li, Zizhou
;
Yang, Yaxi
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2023/04/10
BET Bromodomains
Acute liver injury
Anti-inflammatory activity
Inhibitors
Tetracyclic compounds
Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 13
作者:
Luo, Menglan
;
Wu, Qian
;
Yang, Yueyue
;
Sun, Lin
;
Huan, Xiajuan
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2022/08/30
BET inhibitor
BRD4
Bivalent inhibitor
Anticancer
Selective bromodomain and extra-terminal bromodomain inhibitor inactivates macrophages and hepatic stellate cells to inhibit liver inflammation and fibrosis
期刊论文
OAI收割
BIOENGINEERED, 2022, 卷号: 13, 期号: 4, 页码: 10914-10930
作者:
Fu, Rong
;
Zu, Shi-Jia
;
Liu, Yan-Jun
;
Li, Jia-Cheng
;
Dang, Wen-Zhen
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2022/06/15
BET inhibitor
macrophage
hepatic stellate cell
inflammation
fibrosis
Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma
期刊论文
OAI收割
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:
Chen, Zi-qi
;
Cao, Zhe-rui
;
Wang, Yi
;
Zhang, Xi
;
Xu, Lan
  |  
收藏
  |  
浏览/下载:54/0
  |  
提交时间:2021/12/16
CYH33
MYC
P300
BET
B cell lymphoma
PI3K
TNKS inhibitors potentiate proliferative inhibition of BET inhibitors via reducing beta-Catenin in colorectal cancer cells
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2022, 卷号: 12, 期号: 3, 页码: 1069-+
作者:
Wu, Qian
;
Xuan, Yi-Fei
;
Su, Ai-Ling
;
Bao, Xu-Bin
;
Miao, Ze-Hong
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
BET inhibitor
Tankyrases inhibitor
beta-Catenin
antitumor activity
combination therapy
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells
期刊论文
OAI收割
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:
Liu, Yuwei
;
Xue, Mengzhu
;
Cao, Danyan
;
Qin, Lihuai
;
Wang, Ying
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2021/08/17
Multi-omics
BET inhibitor responses
WNT pathway
Liver cancer
Precise therapy
Novel bivalent BET inhibitor N2817 exhibits potent anticancer activity and inhibits TAF1
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 185, 页码: 14
作者:
Wu, Qian
;
Chen, Dan-Qi
;
Sun, Lin
;
Huan, Xia-Juan
;
Bao, Xu-Bin
  |  
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2021/05/24
N2817
Bivalent BET inhibitors
Monovalent BET inhibitors
TAF1
Anticancer activity
The MYC Paralog-PARP1 Axis as a Potential TherapeuticTarget in MYC Paralog-Activated Small Cell Lung Cancer
期刊论文
OAI收割
FRONTIERS IN ONCOLOGY, 2020, 卷号: 10
作者:
Bian, Xing
;
Wang, Xiaolin
;
Zhang, Qiuyan
;
Ma, Liying
;
Cao, Guozhen
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2020/11/30
small cell lung cancer
MYCparalog
PARP1
BET
DNA damage response