中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共62条,第1-10条 帮助

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Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:  
Chen, Xuetao;  Wu, Tingting;  Du, Zhiyan;  Kang, Wenjing;  Xu, Rujun
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/02/27
Evolution of pore structure and adsorption-desorption in oil shale formation rocks after compression 期刊论文  OAI收割
ENERGY, 2023, 卷号: 278, 页码: 127913
作者:  
Huang XF(黄先富);  Zhao YP(赵亚溥)
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/09/05
Cyclization strategy leads to highly potent Bromodomain and extra-terminal (BET) Bromodomain inhibitors for the treatment of acute liver injury 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 247, 页码: 13
作者:  
Chen, Chao;  Lu, Tian;  Chen, Panyu;  Li, Zizhou;  Yang, Yaxi
  |  收藏  |  浏览/下载:23/0  |  提交时间:2023/04/10
Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 239, 页码: 13
作者:  
Luo, Menglan;  Wu, Qian;  Yang, Yueyue;  Sun, Lin;  Huan, Xiajuan
  |  收藏  |  浏览/下载:40/0  |  提交时间:2022/08/30
Selective bromodomain and extra-terminal bromodomain inhibitor inactivates macrophages and hepatic stellate cells to inhibit liver inflammation and fibrosis 期刊论文  OAI收割
BIOENGINEERED, 2022, 卷号: 13, 期号: 4, 页码: 10914-10930
作者:  
Fu, Rong;  Zu, Shi-Jia;  Liu, Yan-Jun;  Li, Jia-Cheng;  Dang, Wen-Zhen
  |  收藏  |  浏览/下载:33/0  |  提交时间:2022/06/15
Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文  OAI收割
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  
Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
  |  收藏  |  浏览/下载:54/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
TNKS inhibitors potentiate proliferative inhibition of BET inhibitors via reducing beta-Catenin in colorectal cancer cells 期刊论文  OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2022, 卷号: 12, 期号: 3, 页码: 1069-+
作者:  
Wu, Qian;  Xuan, Yi-Fei;  Su, Ai-Ling;  Bao, Xu-Bin;  Miao, Ze-Hong
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/06/15
Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells 期刊论文  OAI收割
GENOMICS, 2021, 卷号: 113, 期号: 3, 页码: 1057-1069
作者:  
Liu, Yuwei;  Xue, Mengzhu;  Cao, Danyan;  Qin, Lihuai;  Wang, Ying
  |  收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
Novel bivalent BET inhibitor N2817 exhibits potent anticancer activity and inhibits TAF1 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 185, 页码: 14
作者:  
Wu, Qian;  Chen, Dan-Qi;  Sun, Lin;  Huan, Xia-Juan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:39/0  |  提交时间:2021/05/24
The MYC Paralog-PARP1 Axis as a Potential TherapeuticTarget in MYC Paralog-Activated Small Cell Lung Cancer 期刊论文  OAI收割
FRONTIERS IN ONCOLOGY, 2020, 卷号: 10
作者:  
Bian, Xing;  Wang, Xiaolin;  Zhang, Qiuyan;  Ma, Liying;  Cao, Guozhen
  |  收藏  |  浏览/下载:32/0  |  提交时间:2020/11/30