中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共83条,第1-10条 帮助

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Structure-based optimization of indoline-containing compounds as second generation inhibitors of NF-KB-inducing kinase (NIK) 期刊论文  OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1295, 页码: 19
作者:  
Cheng, Jing;  Yan, Ziqin;  Li, Xinzhi;  Liu, Chen;  Tong, Linjiang
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/12/08
Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1079-1092
作者:  
Qin, Shaozhao;  Feng, Lijian;  Zhao, Qingyi
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/02/27
Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:  
Cheng, Jing;  Yan, Ziqin;  Jiang, Kailong;  Liu, Chen;  Xu, Dehua
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/02/19
Design, Construction, and Screening of Diversified Pyrimidine-Focused DNA-Encoded Libraries 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 14, 期号: 8, 页码: 1073-1078
作者:  
Seydimemet, Mengnisa;  Yang, Yixuan;  Lv, Yuhan;  Liu, Jiaxiang;  Yan, Ziqin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/10/17
Selective degradation of cellular BRD3 and BRD4-L promoted by PROTAC molecules in six cancer cell lines 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 17
作者:  
Yan, Ziqin;  Lyu, Xilin;  Lin, Dongze;  Wu, Gaoxing;  Gong, Yang
  |  收藏  |  浏览/下载:25/0  |  提交时间:2023/10/17
VideoFusion: Decomposed Diffusion Models for High-Quality Video Generation 会议论文  OAI收割
加拿大温和华, 2023-6
作者:  
Luo, Zhengxiong;  Chen, Dayou;  Zhang, Yingya;  Huang, Yan;  Wang, Liang
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/06/09
Norgestrel causes digestive gland injury in the clam Mactra veneriformis: An integrated histological, transcriptomics, and metabolomics study 期刊论文  OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2023, 卷号: 871, 页码: 13
作者:  
Zhao, Xiaoran;  Wang, Qing;  Li, Xiangfei;  Xu, Hua;  Ren, Chuanbo
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/11/15
Synthesis and Biological Evaluation of Sclareolide-Indole Conjugates and Their Derivatives 期刊论文  OAI收割
MOLECULES, 2023, 卷号: 28, 期号: 4, 页码: 1737
作者:  
Cheng, Ying;  Lyu, Xilin;  Liu, Chen;  Wang, Xiancheng;  Cheng, Jing
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/03/27
PRMT6 promotes tumorigenicity and cisplatin response of lung cancer through triggering 6PGD/ENO1 mediated cell metabolism 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 1, 页码: 157-173
作者:  
Sun, Mingming;  Li, Leilei;  Niu, Yujia;  Wang, Yingzhi;  Yan, Qi
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/03/27
A chemical perspective on the modulation of TEAD transcriptional activities: Recent progress, challenges, and opportunities 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 31
作者:  
Lou, Jianfeng;  Lu, Yuhang;  Cheng, Jing;  Zhou, Feilong;  Yan, Ziqin
  |  收藏  |  浏览/下载:27/0  |  提交时间:2022/12/13