中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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金属研究所 [37]
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LPS exacerbates TRPV4-mediated itch through the intracellular TLR4-PI3K signalling
期刊论文
OAI收割
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2024, 卷号: 28, 期号: 13, 页码: 9
作者:
Hao, Yanping
;
Wu, Liyan
;
Wang, Yuhui
;
Shan, Dongmei
;
Liu, Yifei
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/08/22
itch sensitization
LPS
PI3K
TLR4
TRPV4
Effect of constraint on fracture performance of Ti6Al4V alloy fabricated by laser powder bed fusion
期刊论文
OAI收割
THEORETICAL AND APPLIED FRACTURE MECHANICS, 2024, 卷号: 131, 页码: 11
作者:
Xiao YM(肖应梦)
;
Sun JY(孙经雨)
;
Qian GA(钱桂安)
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/07/04
Laser powder bed fusion
Fracture property
Constraint effect
Ti6Al4V alloy
K-T-11-T-33 method
Discovery of a novel 53BP1 inhibitor through AlphaScreen-based high-throughput screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 34, 页码: 116054
作者:
Sun, Yanli
;
Lu, Haibo
;
Fang, Xueyu
;
Xiao, Senhao
;
Yang, Feng
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2024/03/21
53BP1-TTD
H4K2Ome2
AlphaScreen
HTS
Novel inhibitor
Discovery of 2-(5-(quinolin-6-yl)-1,3,4-oxadiazol-2-yl)acetamide derivatives as novel PI3K alpha inhibitors via docking-based virtual screening
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 9
作者:
Gu, Dongyan
;
Cheng, Gang
;
Zhang, Mengmeng
;
Zhou, Yu-Bo
;
Li, Jia
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/24
PI3K alpha inhibitors
Virtual screening
2-(5-(quinolin-6-yl)-1,3,4 oxadiazol-2-yl)acetamide
Molecular dynamics
Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:
Xiang, Hao-Yue
;
Wang, Xiang
;
Chen, Yan-Hong
;
Zhang, Xi
;
Tan, Cun
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/05/24
PI3K
Pyrrolo[2,1-f][1,2,4]triazine
Anti-cancer
Target therapy
Enhancing the denitration performance and anti-K poisoning ability of CeO2-TiO2/P25 catalyst by H2SO4 pretreatment: Structure-activity relationship and mechanism study
期刊论文
OAI收割
APPLIED CATALYSIS B-ENVIRONMENTAL, 2020, 卷号: 269, 页码: 13
作者:
Yao, Xiaojiang
;
Kang, Keke
;
Cao, Jun
;
Chen, Li
;
Luo, Wen
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/08/24
CeO2-TiO2/P25 catalyst
H2SO4 pretreatment
Denitration performance
Anti-K poisoning ability
NH3-SCR reaction
Design, synthesis and antiproliferative activity evaluation of a series of pyrrolo [2,1-f] [1,2,4] triazine derivatives
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 12, 页码: 4
作者:
Xiang, Hao-Yue
;
Chen, Yan-Hong
;
Wang, Yi
;
Zhang, Xi
;
Ding, Jian
  |  
收藏
  |  
浏览/下载:40/0
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提交时间:2020/07/01
Antiproliferative
Cancer
Therapy
PI3K inhibitors
Pyrrolo [2,1-f][1,2,4] triazine
Kinase
Discovery of 6 '-chloro-N-methyl-5 '-(phenylsulfonamido)-[3,3 '-bipyridine]-5-carboxamide (CHMFL-PI4K-127) as a novel Plasmodium falciparum PI(4)K inhibitor with potent antimalarial activity against both blood and liver stages of Plasmodium
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 188
作者:
Liang, Xiaofei
;
Jiang, Zongru
;
Huang, Zhenghui
;
Li, Feng
;
Chen, Cheng
  |  
收藏
  |  
浏览/下载:46/0
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提交时间:2020/11/26
PI4K kinase
Kinase inhibitor
Malaria
Blood stage
Liver stage
Enhanced electrodeposition and separation of metallic Cr from soluble K2CrO4 on a liquid Zn cathode
期刊论文
OAI收割
JOURNAL OF ENERGY CHEMISTRY, 2020, 卷号: 40, 页码: 204-211
作者:
Weng, Wei
;
Wang, Zhi
;
Guo, Zhancheng
;
Jiao, Shuqiang
;
Wang, Mingyong
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2020/03/24
Molten salt electrolysis
Liquid Zn cathode
Carbon contamination
K2CrO4
Metallic Cr
Lithium recovery from lepidolite roasted with potassium compounds
期刊论文
OAI收割
MINERALS ENGINEERING, 2020, 卷号: 145, 页码: 9
作者:
Su, Hui
;
Ju, Jiaying
;
Zhang, Jian
;
Yi, Aifei
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2020/03/24
Lepidolite
Lithium
K2SO4
KOH
Roasting
Water leaching