中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
昆明植物研究所 [5]
上海药物研究所 [3]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2024 [1]
2023 [1]
2022 [2]
2021 [1]
2019 [1]
2009 [1]
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学科主题
Chemistry,... [1]
Chemistry,... [1]
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Structure-based development of potent and selective type-II kinase inhibitors of RIPK1
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 1, 页码: 319-334
作者:
Qin, Ying
;
Li, Dekang
;
Qi, Chunting
;
Xiang, Huaijiang
;
Meng, Huyan
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2024/03/06
RIPK1
Necroptosis
Type-II kinase inhibitors
Rational design
Lead optimization
Structure-activity relationship
Anti-inflammation
Preclinical drug discovery
Optimization of potent, selective and orally bioavailable biphenyl scaffold as FABP4 inhibitors for anti-inflammation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 253, 页码: 16
作者:
He, Yulong
;
Li, Shunyi
;
Zhu, Yueyue
;
Wang, Yujie
;
Chen, Yuqi
  |  
收藏
  |  
浏览/下载:85/0
  |  
提交时间:2023/10/17
Structure-activity relationship
FABP4 inhibitor
Biphenyl scaffold
Selectivity
Oral bioavailability
Anti-inflammation
Anti-Inflammatory Effects of Camellia fascicularis Polyphenols via Attenuation of NF-kappa B and MAPK Pathways in LPS-Induced THP-1 Macrophages
期刊论文
OAI收割
JOURNAL OF INFLAMMATION RESEARCH, 2022, 卷号: 15, 页码: 851-864
作者:
Gao, Miaozi
;
Peng, Xiaowei
;
Tang, Junrong
;
Deng, Jia
;
Wang, Fang
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/04/30
Camellia fascicularis
polyphenols
anti-inflammatory activity
NF-kappa B
MAPK
LIPOPOLYSACCHARIDE-INDUCED INFLAMMATION
OXIDATIVE STRESS
CELLS
SUPPRESSION
ANTIOXIDANT
ACTIVATION
NRF2/HO-1
RESPONSES
PROTEIN
CANCER
Anti-Adipogenic Lanostane-Type Triterpenoids from the Edible and Medicinal Mushroom Ganoderma applanatum
期刊论文
OAI收割
JOURNAL OF FUNGI, 2022, 卷号: 8, 期号: 4, 页码: 331
作者:
Peng, Xing-Rong
;
Wang, Qian
;
Su, Hai-Guo
;
Zhou, Lin
;
Xiong, Wen-Yong
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/04/30
Ganoderma applanatum
lanostane triterpenoid
Mosher's method
anti-adipogenesis activity
structure-activity relationship
APOPTOSIS
LUCIDUM
INFLAMMATION
METABOLISM
EXTRACTS
PROVIDE
BODY
Diversity-oriented synthesis of cembranoid derivatives as potential anti-inflammatory agents
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 111, 页码: 8
作者:
Zhang, Cong
;
Li, Heng
;
Liu, Jin
;
Liu, Moting
;
Zhang, Hao
  |  
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2021/08/17
Marine natural product
Cembranoid
Anti-inflammation
molecular docking
structuremodification
Structure Activity Relationship
The polymer iridoid glucosides isolated from Dipsacus asper
期刊论文
OAI收割
PHYTOCHEMISTRY LETTERS, 2019, 卷号: 33, 页码: 17-21
作者:
Duan, Xiao-Yan
;
Ai, Lun-Qiang
;
Qian, Cheng-Zhen
;
Zhang, Mei-De
;
Mei, Ren-Qiang
  |  
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2019/12/20
Dipsacus asper
Tetrairidoid glucosides
Bis-iridoid glucosides
Anti-inflammation activity
Anti-inflammatory activity of lansais from endophytic Streptomyces sp SUC1 in LPS-induced RAW 264.7 cells
期刊论文
OAI收割
FOOD AND AGRICULTURAL IMMUNOLOGY, 2009, 卷号: 20, 期号: 1, 页码: 67-77
Taechowisan, Thongchai
;
Wanbanjob, Asawin
;
Tuntiwachwuttikul, Pittaya
;
Liu, Jikai
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2012/10/12
anti-inflammatory activity
endophytic Streptomyces
lansai C
RAW 264
7 cells
NITRIC-OXIDE PRODUCTION
MACROPHAGES
LIPOPOLYSACCHARIDE
CYCLOOXYGENASE-2
INFLAMMATION
CYTOKINES
PAIN
In vitro anti-inflammatory activity of 4-arylcoumarins from endophytic Streptomyces aureofaciens CMUAc130 in murine macrophage RAW 264.7 cells
期刊论文
OAI收割
NATURAL PRODUCT RESEARCH, 2007, 卷号: 21, 期号: 12, 页码: 1104-1113
Taechowisan, Thongchai
;
Lu, Chunhua
;
Shen, Yuemao
;
Lumyong, Saisamorn
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2012/10/12
4-arylcoumarins
anti-inflammatory activity
endophytic streptomyces
murine macrophage RAW 264.7 cells
HUMAN-LEUKOCYTE ELASTASE
COUMARIN DERIVATIVES
ANTIFUNGAL ACTIVITY
INHIBITORS
LIPOPOLYSACCHARIDE
CYCLOOXYGENASE-2
INFLAMMATION
ENZYME
ACID