中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共17条,第1-10条 帮助

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The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer 期刊论文  OAI收割
CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:  
He, Ting;  Gao, Yinglei;  Fang, Yanfen;  Zhang, Yangming;  Zhang, Shuwei
  |  收藏  |  浏览/下载:27/0  |  提交时间:2024/03/21
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:  
Lu, Dong;  Yan, Juan
  |  收藏  |  浏览/下载:58/0  |  提交时间:2019/01/08
Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b] [1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 239-251
作者:  
Zhan, Zhengsheng;  Peng, Xia;  Liu, Qiufeng;  Chen, Fang;  Ji, Yinchun
  |  收藏  |  浏览/下载:58/0  |  提交时间:2019/01/08
Simm530, a novel and highly selective c-Met inhibitor, blocks c-Met-stimulated signaling and neoplastic activities 期刊论文  OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 25, 页码: 38091-38104
作者:  
Wang, Ying;  Zhan, Zhengsheng;  Jiang, Xifei;  Peng, Xia;  Shen, Yanyan
  |  收藏  |  浏览/下载:67/0  |  提交时间:2019/01/08
Pyridazinone derivatives displaying highly potent and selective inhibitory activities against c-Met tyrosine kinase 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 322-333
作者:  
Liu, Yang;  Jin, Shiyu;  Peng, Xia;  Lu, Dong;  Zeng, Limin
  |  收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Enhancing the cellular anti-proliferation activity of pyridazinones as c-met inhibitors using docking analysis 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 95, 页码: 302-312
作者:  
Xing, Weiqiang;  Ai, Jing;  Jin, Shiyu;  Shi, Zhangxing;  Peng, Xia
  |  收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Imidazo[1,2-a]pyridine Derivatives as Potent c-Met Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 507-512
作者:  
Li, Chunpu;  Ai, Jing;  Zhang, Dengyou;  Peng, Xia;  Chen, Xi
  |  收藏  |  浏览/下载:24/0  |  提交时间:2019/01/08
Discovery and SAR study of c-Met kinase inhibitors bearing an 3-amino-benzo[d] isoxazole or 3-aminoindazole scaffold 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 3, 页码: 564-578
作者:  
Jiang, Xiaolong;  Liu, Hongyan
  |  收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Discovery of potent 1H-imidazo[4,5-b]pyridine-based c-Met kinase inhibitors via mechanism-directed structural optimization 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 3, 页码: 708-716
作者:  
An, Xiao-De;  Liu, Hongyan;  Xu, Zhong-Liang;  Jin, Yi;  Peng, Xia
  |  收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Discovery of novel type II c-Met inhibitors based on BMS-777607 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 80, 页码: 254-266
作者:  
Zhang, Wei;  Ai, Jing;  Shi, Dakuo;  Peng, Xia;  Ji, Yinchun
  |  收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08