中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
上海药物研究所 [15]
金属研究所 [2]
采集方式
OAI收割 [17]
内容类型
期刊论文 [17]
发表日期
2022 [1]
2017 [1]
2016 [3]
2015 [4]
2014 [5]
2013 [3]
更多
学科主题
筛选
浏览/检索结果:
共17条,第1-10条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
题名升序
题名降序
提交时间升序
提交时间降序
作者升序
作者降序
发表日期升序
发表日期降序
The HDAC inhibitor GCJ-490A suppresses c-Met expression through IKK? and overcomes gefitinib resistance in non-small cell lung cancer
期刊论文
OAI收割
CANCER BIOLOGY & MEDICINE, 2022, 卷号: 19, 期号: 8, 页码: 1172-1192
作者:
He, Ting
;
Gao, Yinglei
;
Fang, Yanfen
;
Zhang, Yangming
;
Zhang, Shuwei
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2024/03/21
HDAC inhibitor
c-Met
IKK?
NSCLC
gefitinib
Design, Synthesis, and Biological Evaluation of the First c-Met/HDAC Inhibitors Based on Pyridazinone Derivatives
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 8, 期号: 8, 页码: 830-834
作者:
Lu, Dong
;
Yan, Juan
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2019/01/08
Dual c-Met/HDAC inhibitor
hybrid
designed multiple ligand (DML)
Discovery of 6-(difluoro(6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b] [1,2,4]triazin-3-yl)methyl)quinoline as a highly potent and selective c-Met inhibitor
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 116, 页码: 239-251
作者:
Zhan, Zhengsheng
;
Peng, Xia
;
Liu, Qiufeng
;
Chen, Fang
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2019/01/08
Antitumor
c-Met
Kinase inhibitor
Triazolotriazines
Simm530, a novel and highly selective c-Met inhibitor, blocks c-Met-stimulated signaling and neoplastic activities
期刊论文
OAI收割
ONCOTARGET, 2016, 卷号: 7, 期号: 25, 页码: 38091-38104
作者:
Wang, Ying
;
Zhan, Zhengsheng
;
Jiang, Xifei
;
Peng, Xia
;
Shen, Yanyan
  |  
收藏
  |  
浏览/下载:67/0
  |  
提交时间:2019/01/08
c-Met
kinase inhibitor
Simm530
Pyridazinone derivatives displaying highly potent and selective inhibitory activities against c-Met tyrosine kinase
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 108, 页码: 322-333
作者:
Liu, Yang
;
Jin, Shiyu
;
Peng, Xia
;
Lu, Dong
;
Zeng, Limin
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2019/01/08
Pyridazinone
c-Met inhibitor
Cyclization strategy
Antitumor
Enhancing the cellular anti-proliferation activity of pyridazinones as c-met inhibitors using docking analysis
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 95, 页码: 302-312
作者:
Xing, Weiqiang
;
Ai, Jing
;
Jin, Shiyu
;
Shi, Zhangxing
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Pyridazinone
c-Met inhibitor
Anticancer
Docking study
Design, Synthesis, and Biological Evaluation of Novel Imidazo[1,2-a]pyridine Derivatives as Potent c-Met Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 5, 页码: 507-512
作者:
Li, Chunpu
;
Ai, Jing
;
Zhang, Dengyou
;
Peng, Xia
;
Chen, Xi
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Receptor tyrosine kinase
c-Met inhibitor
imidazo[1,2-a]pyridine
metabolic stability
Discovery and SAR study of c-Met kinase inhibitors bearing an 3-amino-benzo[d] isoxazole or 3-aminoindazole scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 3, 页码: 564-578
作者:
Jiang, Xiaolong
;
Liu, Hongyan
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
c-Met kinase
Inhibitor
3-Amino-benzo[d]isoxazole
3-Aminoindazole
Non-small cell lung cancer
Discovery of potent 1H-imidazo[4,5-b]pyridine-based c-Met kinase inhibitors via mechanism-directed structural optimization
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 3, 页码: 708-716
作者:
An, Xiao-De
;
Liu, Hongyan
;
Xu, Zhong-Liang
;
Jin, Yi
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
c-Met tyrosine kinase
Small molecule inhibitor
Imidazonaphthyridinone
Imidazopyridine
Binding mode
Pyridone-3-carboxamide
Cyclopropane-1,1-dicarboxamide
Discovery of novel type II c-Met inhibitors based on BMS-777607
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 80, 页码: 254-266
作者:
Zhang, Wei
;
Ai, Jing
;
Shi, Dakuo
;
Peng, Xia
;
Ji, Yinchun
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
c-Met
Synthesis
Kinase inhibitor