中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2022 [22]
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Structure-Based Design of Tropane Derivatives as a Novel Series of CCR5 Antagonists with Broad-Spectrum Anti-HIV-1 Activities and Improved Oral Bioavailability 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 24, 页码: 16526-16540
作者:  
Xie, Xiong;  Zheng, Yu-Gui;  Chen, Huan;  Li, Jian;  Luo, Rong-Hua
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10
Facile Synthesis of Benzimidazoles via N-Arylamidoxime Cyclization 期刊论文  OAI收割
ACS OMEGA, 2022, 页码: 10
作者:  
Qin, Hongjian;  Odilov, Abdullajon;  Bonku, Emmanuel Mintah;  Zhu, Fuqiang;  Hu, Tianwen
  |  收藏  |  浏览/下载:24/0  |  提交时间:2023/04/10
Simulating androgen receptor selection in designer yeast 期刊论文  OAI收割
SYNTHETIC AND SYSTEMS BIOTECHNOLOGY, 2022, 卷号: 7
作者:  
Zhang, Haoran;  Zhang, Lu;  Xu, Yipeng;  Chen, Shaoyong;  Ma, Zhenyi
  |  收藏  |  浏览/下载:19/0  |  提交时间:2022/12/23
Olanzapine for the Prevention and Treatment of Chemotherapy-Induced Nausea and Vomiting: A Review to Identify the Best Way to Administer the Drug 期刊论文  OAI收割
CURRENT ONCOLOGY, 2022, 卷号: 29
作者:  
Zhang, Xiao-Ling;  Ying, Jie-Er
  |  收藏  |  浏览/下载:19/0  |  提交时间:2022/12/23
Upregulation of dynorphin/kappa opioid receptor system in the dorsal hippocampus contributes to morphine withdrawal-induced place aversion 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 8
作者:  
Chen, Yan;  Wang, Chen-yao;  Zan, Gui-ying;  Yao, Song-yu;  Deng, Ying-zhi
  |  收藏  |  浏览/下载:22/0  |  提交时间:2022/11/11
Discovery of Betulinic Acid Derivatives as Potent Intestinal Farnesoid X Receptor Antagonists to Ameliorate Nonalcoholic Steatohepatitis 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 21
作者:  
Zhang, Chenlu;  Liu, Yameng;  Wang, Ying;  Ge, Xie;  Jiao, Tingying
  |  收藏  |  浏览/下载:35/0  |  提交时间:2022/11/11
Synthesis of Hydantoin Androgen Receptor Antagonists and Study on Their Antagonistic Activity 期刊论文  OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 18, 页码: 22
作者:  
Ma, Longjun;  Zhou, Yan;  Yang, Dehua;  Wang, Ming-Wei;  Lu, Wei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2022/11/11
Key Considerations in Targeted Protein Degradation Drug Discovery and Development 期刊论文  OAI收割
FRONTIERS IN CHEMISTRY, 2022, 卷号: 10
作者:  
Qin, Liena;  Dai, Han;  Wang, Junfeng
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/12/23
Structural insights into ligand recognition and selectivity of somatostatin receptors 期刊论文  OAI收割
CELL RESEARCH, 2022, 页码: 12
作者:  
Zhao, Wenli;  Han, Shuo;  Qiu, Na;  Feng, Wenbo;  Lu, Mengjie
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/08/16
Identification of a Subtype-Selective Allosteric Inhibitor of GluN1/GluN3 NMDA Receptors 期刊论文  OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 13
作者:  
Zeng, Yue;  Zheng, Yueming;  Zhang, Tongtong;  Ye, Fei;  Zhan, Li
  |  收藏  |  浏览/下载:18/0  |  提交时间:2022/08/16