中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [186]
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Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 25
作者:  
Zhang, Yinyong;  Zhang, Dan;  Zhao, Wenhao;  Li, Hongyuan;  Lu, Zhengyu
  |  收藏  |  浏览/下载:0/0  |  提交时间:2024/05/22
Chemical and biosynthetic potential of Penicillium shentong XL-F41 期刊论文  OAI收割
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 2024, 卷号: 20, 页码: 597-606
作者:  
Zou, Ran;  Li, Xin;  Chen, Xiaochen;  Guo, Yue-Wei;  Xu, Baofu
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/05/07
Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:  
Zhuo, Ning;  Yun, Ying;  Zhang, Chenlu;  Guo, Shimeng;  Yin, Jianpeng
  |  收藏  |  浏览/下载:17/0  |  提交时间:2024/03/25
Pharmacological inhibition of Kir4.1 evokes rapid-onset antidepressant responses 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2024, 页码: 29
作者:  
Zhou, Xiaoyu;  Zhao, Cheng
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/03/25
Discovery and exploration of novel somatostatin receptor subtype 5 (SSTR5) antagonists for the treatment of cholesterol gallstones 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 264, 页码: 16
作者:  
Han, Fanghui;  Zhao, Tingting;  Zhang, Yanglong;  Yun, Ying;  Xu, Yuanyuan
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/02/19
Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 96, 页码: 12
作者:  
Song, Zhaoxiang;  Lu, Dan;  Sun, Jun;  Ye, Yangliang;  Fang, Jiahui
  |  收藏  |  浏览/下载:31/0  |  提交时间:2024/01/16
GPR35  IBD  Lodoxamide  
A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects 期刊论文  OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:  
Yang, Xin-Mei;  Yang, Yang;  Yao, Bu-Fan;  Ye, Pan-Pan;  Xu, Yan
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/12/11
The aminosteroid U73122 promotes oligodendrocytes generation and myelin formation 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 12
作者:  
Cui, Shi-hao;  Suo, Na;  Yang, Ying;  Wu, Xuan;  Guo, Shi-meng
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/12/11
Design and Synthesis Studies of α-Methylene-γ-butyrolactones Antagonists of GPR52 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 43, 期号: 11, 页码: 3916-3929
作者:  
Shen, Donghang;  Li, Xin;  Guo, Shimeng;  Xie, Xin;  Nan, Fajun
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/02/27
Ligand recognition and G protein coupling of the human itch receptor MRGPRX1 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 12
作者:  
Guo, Lulu;  Zhang, Yumu;  Fang, Guoxing;  Tie, Lu;  Zhuang, Yuming
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/01/16