中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [91]
采集方式
OAI收割 [91]
内容类型
期刊论文 [90]
会议论文 [1]
发表日期
2024 [3]
2023 [7]
2022 [11]
2021 [12]
2020 [5]
2019 [9]
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Biochemist... [1]
Chemistry [1]
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浏览/检索结果:
共91条,第1-10条
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专题:上海药物研究所
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Discovery of a Covalent Inhibitor Selectively Targeting the Autophosphorylation Site of c-Src Kinase
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2024, 页码: 12
作者:
Zhang, Huimin
;
Xu, Dounan
;
Huang, Hongchan
;
Jiang, Hao
;
Hu, Linghao
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Structure-based design of pan-coronavirus inhibitors targeting host cathepsin L and calpain-1
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2024, 卷号: 9, 期号: 1, 页码: 14
作者:
Xie, Xiong
;
Lan, Qiaoshuai
;
Zhao, Jinyi
;
Zhang, Sulin
;
Liu, Lu
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Limonoids and alkaloids from
Tetradium
austrosinense
(Hand.-Mazz.) TG Hartley
期刊论文
OAI收割
FITOTERAPIA, 2024, 卷号: 172, 页码: 5
作者:
Han, Feng
;
Yao, Jia-Ying
;
Tan, Jun-Jie
;
Qin, Nan
;
Jiang, Yu-Xia
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2024/02/19
Rutaceae
Tetradium austrosinense
Limonoids
Alkaloids
TDDFT-ECD calculation
Anti-inflammation
Ginsenoside Rg3 endows liposomes with prolonged blood circulation and reduced accelerated blood clearance
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2023, 卷号: 364, 页码: 23-36
作者:
Xia, Jiaxuan
;
Chen, Chen
;
Dong, Meichen
;
Zhu, Ying
;
Wang, Anni
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/01/16
Ginsenoside Rg3
Liposomes
Polyethylene glycol
Long circulation
Accelerated blood clearance (ABC)
IgM antibody
Complement activation
Natural product P57 induces hypothermia through targeting pyridoxal kinase
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 15
作者:
Wang, Ruina
;
Xiao, Lei
;
Pan, Jianbo
;
Bao, Guangsen
;
Zhu, Yunmei
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/02/19
B-seco Limonoids with anti-inflammatory activity from Tetradium fraxinifolium (Hook.) TGHartley
期刊论文
OAI收割
FITOTERAPIA, 2023, 卷号: 169, 页码: 6
作者:
Jiang, Yu-Xia
;
Yao, Jia-Ying
;
Qin, Nan
;
Tan, Jun-Jie
;
Han, Feng
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17
Tetradium fraxinifolium
Rutaceae
seco limonoids
Anti-inflammation
RAW264
7 cells
ETCM v2.0: An update with comprehensive resource and rich annotations for traditional Chinese medicine
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 6, 页码: 2559-2571
作者:
Zhang, Yanqiong
;
Li, Xin
;
Shi, Yulong
;
Chen, Tong
;
Xu, Zhijian
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/10/17
Traditional Chinese medicine
Database
Target identification
Network visualization
New drug research and development
Molecular mechanism
Quality marker
Drug repurposing
SYK-mediated epithelial cell state is associated with response to c-Met inhibitors in c-Met-overexpressing lung cancer
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 13
作者:
Zhou, Ji
;
Zhang, Xu-Chao
;
Xue, Shan
;
Dai, Mengdi
;
Wang, Yueliang
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Optimization of carbazole carboxamide RORγt agonists: Challenges in improving the metabolic stability and maintaining the agonistic activity
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 251, 页码: 115213
作者:
Sun, Nannan
;
Yu, Mingcheng
;
Jiang, Zhengyuan
;
Yang, Feng
;
Lu, Lixue
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/27
ROR?t agonists
Carbazole carboxamide
Agonistic activity
Metabolic stability
Co-crystallization
Molecular docking
Rucaparib cocrystal: Improved solubility and bioavailability over camsylate
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2023, 卷号: 631, 页码: 10
作者:
Xia, Mengyuan
;
Jiang, Yihua
;
Cheng, Yinxiang
;
Dai, Wenjuan
;
Rong, Xiaoyi
  |  
收藏
  |  
浏览/下载:63/0
  |  
提交时间:2023/04/10
Rucaparib
Cocrystal
Solubility
Dissolution
Bioavailability