中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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机构
上海药物研究所 [14]
上海生物化学与细胞生... [8]
中国科学院大学 [2]
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期刊论文 [26]
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2022 [2]
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Learning with uncertainty to accelerate the discovery of histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitors
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2022, 页码: 14
作者:
Wang, Dong
;
Wu, Zhenxing
;
Shen, Chao
;
Bao, Lingjie
;
Luo, Hao
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
uncertainty estimation
graph neural network
KDM1A
LSD1 inhibitors
upper confidence bound method
virtual screening
Structure-Activity Relationship Study of Indolin-5-yl-cyclopropanamine Derivatives as Selective Lysine Specific Demethylase 1 (LSD1) Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 5, 页码: 4335-4349
作者:
Li, Chunpu
;
Su, Mingbo
;
Zhu, Wei
;
Kan, Weijuan
;
Ge, Tianpeng
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/06/15
Divalent tranylcypromine derivative as lysine-specific demethylase 1 inhibitor
期刊论文
OAI收割
MEDICINAL CHEMISTRY RESEARCH, 2021, 页码: 8
作者:
Sun, Yin
;
Li, Na
;
Su, Mingbo
;
Wang, Xiaowen
;
Zhao, Dongmei
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/05/24
Divalent tranylcypromine
LSD1 inhibitor
MV4-11 antiproliferative activity
CD86 mRNA expression
Linker
Selectivity
USP28 and USP25 are downregulated by Vismodegib in vitro and in colorectal cancer cell lines
期刊论文
OAI收割
FEBS JOURNAL, 2020, 页码: 18
作者:
Wang, Hui
;
Meng, Qian
;
Ding, Yiluan
;
Xiong, Muya
;
Zhu, Mengying
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
colorectal cancer
HDX-MS
inhibitor
USP25
USP28
Vismodegib
Sepiapterin reductase promotes hepatocellular carcinoma progression via FoxO3a/Bim signaling in a nonenzymatic manner
期刊论文
OAI收割
CELL DEATH & DISEASE, 2020, 卷号: 11, 期号: 4, 页码: 14
作者:
Wu, Yao
;
Du, Hongzhi
;
Zhan, Meixiao
;
Wang, Hongxv
;
Chen, Peng
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
Biological roles of LSD1 beyond its demethylase activity
期刊论文
OAI收割
CELLULAR AND MOLECULAR LIFE SCIENCES, 2020
作者:
Gu, Feiying
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/11/26
LSD1
Demethylase
Ubiquitylation
FBXW7
Non-catalytic
SET8 prevents excessive DNA methylation by methylation-mediated degradation of UHRF1 and DNMT1
期刊论文
OAI收割
NUCLEIC ACIDS RESEARCH, 2019, 卷号: 47, 期号: 17, 页码: 9053-9068
作者:
Zhang, Huifang
;
Gao, Qinqin
;
Tan, Shuo
;
You, Jia
;
Lyu, Cong
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/09/10
Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847
作者:
Wang, Xiaowen
;
Su, Mingbo
;
Li, You
;
Liu, Tongchao
;
Wang, Yujie
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/07/01
LSD1 inhibitor
Tranylcypromine
Menin-MLL1 protei n-protein interaction inhibitor
MV4-11 antiproliferative activity
Structure activity relationship
Kdm1a promotes SCLC progression by transcriptionally silencing the tumor suppressor Rest
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2019, 卷号: 515, 期号: 1, 页码: 214-221
作者:
Jin, Yujuan
;
Ma, Dingailu
;
Gramyk, Tobin
;
Fang, Rui
;
Shi, Yujiang Geno
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2020/12/21
CELL LUNG-CANCER
REPRESSOR
DIFFERENTIATION
Histone demethylase LSD1 regulates bone mass by controlling WNT7B and BMP2 signaling in osteoblasts
期刊论文
OAI收割
BONE RESEARCH, 2018, 卷号: 6, 期号: 14, 页码: -
作者:
Sun, Jun
;
Niu, Ningning
;
Yan, Guang
;
Yang, Yang
;
Zou, Weiguo
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/04/28
Mesenchymal Stem-cells
Brachydactyly Type A2
Gene-expression
Differentiation
Activation
Mouse
Methylation
Repression
Mutations
Leukemia