中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共437条,第1-10条 帮助

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Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:  
Cheng, Jing;  Yan, Ziqin;  Jiang, Kailong;  Liu, Chen;  Xu, Dehua
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/02/19
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study 期刊论文  OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:  
Zhao, Tian-Tian;  Hu, Hao-Jie;  Gao, Li-Xin;  Zhou, Yu-Bo;  Zhu, Yun-Long
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Discovery, Structure-Activity Relationship and In Vitro Anticancer Activity of Small-Molecule Inhibitors of the Protein-Protein Interactions between AF9/ENL and AF4 or DOT1L 期刊论文  OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 28
作者:  
Li, Xin;  Wu, Xiaowei;  Nie, Shenyou;  Zhao, Jidong;  Yao, Yuan
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/19
Discovery of novel cGAS inhibitors based on natural flavonoids 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 140, 页码: 14
作者:  
Li, Jiameng;  Xiong, Muya;  Liu, Jiayuan;  Zhang, Fengping
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/08
Development of SV2A Ligands for Epilepsy Treatment: A Review of Levetiracetam, Brivaracetam, and Padsevonil 期刊论文  OAI收割
NEUROSCIENCE BULLETIN, 2023, 页码: 15
作者:  
Wu, Peng-Peng;  Cao, Bi-Rong;  Tian, Fu-Yun;  Gao, Zhao-Bing
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/08
Loops Mediate Agonist-Induced Activation of the Stimulator of Interferon Genes Protein 期刊论文  OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2023, 页码: 9
作者:  
Li, Rui;  Chen, Lin;  He, Xinheng;  Cao, Duanhua;  Zhang, Zehong
  |  收藏  |  浏览/下载:7/0  |  提交时间:2023/12/11
Risk of drug-drug interactions in China's fight against COVID-19 and beyond 期刊论文  OAI收割
PHARMACOLOGICAL RESEARCH, 2023, 卷号: 196, 页码: 2
作者:  
Zhang, Qingpeng;  Yang, Jiannan;  Zeng, Daniel Dajun;  Feng, Yibin;  Wong, Ian C. K.
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/03/26
Deciphering the functional landscape of phosphosites with deep neural network 期刊论文  OAI收割
CELL REPORTS, 2023, 卷号: 42, 期号: 9, 页码: 23
作者:  
Liang, Zhongjie;  Liu, Tonghai;  Li, Qi;  Zhang, Guangyu;  Zhang, Bei
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/12/08
Screening and optimization of phage display cyclic peptides against the WDR5 WBM site 期刊论文  OAI收割
RSC MEDICINAL CHEMISTRY, 2023, 页码: 10
作者:  
Song, Lingyu;  Cao, Jiawen;  Chen, Lin;  Du, Zhiyan
  |  收藏  |  浏览/下载:6/0  |  提交时间:2023/10/17
Sequence-based drug design as a concept in computational drug design 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 21
作者:  
Chen, Lifan;  Fan, Zisheng;  Chang, Jie;  Yang, Ruirui;  Hou, Hui
  |  收藏  |  浏览/下载:17/0  |  提交时间:2023/10/17