中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [19]
新疆理化技术研究所 [1]
合肥物质科学研究院 [1]
采集方式
OAI收割 [21]
内容类型
期刊论文 [21]
发表日期
2020 [21]
学科主题
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A unique hormonal recognition feature of the human glucagon-like peptide-2 receptor
期刊论文
OAI收割
CELL RESEARCH, 2020, 页码: 11
作者:
Sun, Wen
;
Chen, Li-Nan
;
Zhou, Qingtong
;
Zhao, Li-Hua
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:113/0
  |  
提交时间:2020/12/24
Automated design and optimization of multitarget schizophrenia drug candidates by deep learning
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 204, 页码: 16
作者:
Tan, Xiaoqin
;
Jiang, Xiangrui
;
He, Yang
;
Zhong, Feisheng
;
Li, Xutong
  |  
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2020/12/21
Schizophrenia
Multitarget antipsychotic drugs
Recurrent neural network
Multitask deep neural network
Automated drug design
Anti-inflammatory signaling through G protein-coupled receptors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:
Ge, Yun-jun
;
Liao, Qi-wen
;
Xu, Ye-chun
;
Zhao, Qiang
;
Wu, Bei-li
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2020/12/21
Evaluation of biased agonism mediated by dual agonists of the GLP-1 and glucagon receptors
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 180, 页码: 16
作者:
Darbalaei, Sanaz
;
Yuliantie, Elita
;
Dai, Antao
;
Chang, Rulue
;
Zhao, Peishen
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2020/12/21
G protein-coupled receptor
Glucagon-like peptide-1 receptor
Glucagon receptor
Biased agonism
Unimolecular dual agonist
GPR91, a critical signaling mechanism in modulating pathophysiologic processes in chronic illnesses
期刊论文
OAI收割
FASEB JOURNAL, 2020, 页码: 15
作者:
Li, Xinyi
;
Xie, Li
;
Qu, Xiangli
;
Zhao, Bangyi
;
Fu, Wei
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
G protein-coupled receptor
innate immunity
metabolic regulation
succinate
SUCNR1
GABA(B) receptor pas de deux: insights from high-resolution structures
期刊论文
OAI收割
CELL RESEARCH, 2020, 页码: 2
作者:
Jiang, Yi
;
Xu, H. Eric
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2020/12/24
Mechanochemical Activation of Class-B G-Protein-Coupled Receptor upon Peptide-Ligand Binding
期刊论文
OAI收割
NANO LETTERS, 2020, 卷号: 20, 期号: 7, 页码: 5575-5582
作者:
Lo Giudice, Cristina
;
Zhang, Haonan
;
Wu, Beili
;
Alsteens, David
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/12/24
Atomic force microscopy
single-molecule force spectroscopy
human glucagon receptor
G-protein-coupled receptors
mechanotransduction
Pharmacological characterization of mono-, dual- and tri-peptidic agonists at GIP and GLP-1 receptors
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 13
作者:
Yuliantie, Elita
;
Darbalaei, Sanaz
;
Dai, Antao
;
Zhao, Peishen
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2020/12/24
G protein-coupled receptor
Glucose-dependent insulinotropic peptide receptor
Glucagon-like peptide-1 receptor
Biased agonist
GPCR signaling
A genetically encoded small-size fluorescent pair reveals allosteric conformational changes of G proteins upon its interaction with GPCRs by fluorescence lifetime based FRET
期刊论文
OAI收割
CHEMICAL COMMUNICATIONS, 2020, 卷号: 56
作者:
Shi, Pan
;
Zhang, Yanan
;
Lv, Pei
;
Fang, Wei
;
Ling, Shenglong
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/10/26
Update of P2Y receptor pharmacology: IUPHAR Review 27
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 11, 页码: 2413-2433
作者:
Jacobson, Kenneth A.
;
Delicado, Esmerilda G.
;
Gachet, Christian
;
Kennedy, Charles
;
von Kuegelgen, Ivar
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/07/01