中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
采集方式
内容类型
发表日期
学科主题
筛选

浏览/检索结果: 共21条,第1-10条 帮助

条数/页: 排序方式:
Tail engagement of arrestin at the glucagon receptor 期刊论文  OAI收割
NATURE, 2023, 页码: 21
作者:  
Chen, Kun;  Zhang, Chenhui;  Lin, Shuling;  Yan, Xinyu;  Cai, Heng
  |  收藏  |  浏览/下载:15/0  |  提交时间:2023/10/17
Effects of site-directed mutagenesis of GLP-1 and glucagon receptors on signal transduction activated by dual and triple agonists 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 13
作者:  
Darbalaei, Sanaz;  Chang, Ru-lue;  Zhou, Qing-tong;  Chen, Yan;  Dai, An-tao
  |  收藏  |  浏览/下载:20/0  |  提交时间:2022/09/30
Structural basis of peptidomimetic agonism revealed by small-molecule GLP-1R agonists Boc5 and WB4-24 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 20, 页码: 10
作者:  
Cong, Zhaotong;  Zhou, Qingtong;  Li, Yang;  Chen, Li-Nan;  Zhang, Zi-Chen
  |  收藏  |  浏览/下载:29/0  |  提交时间:2022/09/30
Structural insights into multiplexed pharmacological actions of tirzepatide and peptide 20 at the GIP, GLP-1 or glucagon receptors 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:  
Zhao, Fenghui;  Zhou, Qingtong;  Cong, Zhaotong;  Hang, Kaini;  Zou, Xinyu
  |  收藏  |  浏览/下载:38/0  |  提交时间:2022/06/15
Insights into agonist-elicited activation of the human glucose-dependent insulinotropic polypeptide receptor 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2021, 卷号: 192, 页码: 16
作者:  
Yuliantie, Elita;  van der Velden, Wijnand J. C.;  Labroska, Viktorija;  Dai, Antao;  Zhao, Fenghui
  |  收藏  |  浏览/下载:94/0  |  提交时间:2021/11/04
G protein-coupled receptors: structure- and function-based drug discovery 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 27
作者:  
Yang, Dehua;  Zhou, Qingtong;  Labroska, Viktorija;  Qin, Shanshan;  Darbalaei, Sanaz
  |  收藏  |  浏览/下载:29/0  |  提交时间:2021/05/24
Evaluation of biased agonism mediated by dual agonists of the GLP-1 and glucagon receptors 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 180, 页码: 16
作者:  
Darbalaei, Sanaz;  Yuliantie, Elita;  Dai, Antao;  Chang, Rulue;  Zhao, Peishen
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/12/21
Cryo-electron microscopy structure of the glucagon receptor with a dual-agonist peptide 期刊论文  OAI收割
JOURNAL OF BIOLOGICAL CHEMISTRY, 2020, 卷号: 295, 期号: 28, 页码: 9313-9325
作者:  
Chang, Rulue;  Zhang, Xin;  Qiao, Anna;  Dai, Antao;  Belousoff, Matthew J.
  |  收藏  |  浏览/下载:40/0  |  提交时间:2020/12/24
Pharmacological characterization of mono-, dual- and tri-peptidic agonists at GIP and GLP-1 receptors 期刊论文  OAI收割
BIOCHEMICAL PHARMACOLOGY, 2020, 卷号: 177, 页码: 13
作者:  
Yuliantie, Elita;  Darbalaei, Sanaz;  Dai, Antao;  Zhao, Peishen;  Yang, Dehua
  |  收藏  |  浏览/下载:23/0  |  提交时间:2020/12/24
Discovery of 3-((dimethylamino)methyl)-4-hydroxy-4-(3-methoxypheny1)-N-phenylpiperidine-1-carboxamide as novel potent analgesic 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 189, 页码: 14
作者:  
Huang, Huoming;  Wang, Wenli;  Xu, Xuejun;  Zhu, Chen;  Wang, Yujun
  |  收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01